Sequential Cross-Coupling of 1,4-Bissilylbutadienes:  Synthesis of Unsymmetrical 1,4-Disubstituted 1,3-Butadienes von Denmark, Scott E., Tymonko, Steven A.

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Mechanistic Significance of the Si–O–Pd Bond in the Palladium-Catalyzed Cross-Coupling Reactions of Alkenylsilanolates von Tymonko, Steven A, Smith, Russell C, Ambrosi, Andrea, Denmark, Scott E

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Mechanistic Significance of the Si–O–Pd Bond in the Palladium-Catalyzed Cross-Coupling Reactions of Arylsilanolates von Tymonko, Steven A, Smith, Russell C, Ambrosi, Andrea, Ober, Michael H, Wang, Hao, Denmark, Scott E

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Phosphine oxides as stabilizing ligands for the palladium-catalyzed cross-coupling of potassium aryldimethylsilanolates von Denmark, Scott E., Smith, Russell C., Tymonko, Steven A.

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Syn-Selective Synthesis of β‑Branched α‑Amino Acids by Alkylation of Glycine-Derived Imines with Secondary Sulfonates von Lou, Sha, McKenna, Grace M, Tymonko, Steven A, Ramirez, Antonio, Benkovics, Tamas, Conlon, David A, González-Bobes, Francisco

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A Scalable Synthesis of (R,R)‑2,6-Dimethyldihydro‑2H‑pyran-4(3H)‑one von Young, Ian S, Haley, Matthew W, Tam, Annie, Tymonko, Steven A, Xu, Zhongmin, Hanson, Ronald L, Goswami, Animesh

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A Qualitative Examination of the Effects of Silicon Substituents on the Efficiency of Cross-Coupling Reactions von Denmark, Scott E, Neuville, Luc, Christy, Matthew E. L, Tymonko, Steven A

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Development of a Practical Synthesis of Functionalized Azaxanthene-Derived Nonsteroidal Glucocorticoid Receptor Modulators von Conlon, David A, Natalie, Kenneth J, Cuniere, Nicolas, Razler, Thomas M, Zhu, Jason, de Mas, Nuria, Tymonko, Steven, Fraunhoffer, Kenneth J, Sortore, Eric, Rosso, Victor W, Xu, Zhongmin, Adams, Monica L, Patel, Anisha, Huang, Jun, Gong, Hua, Weinstein, David S, Quiroz, Fernando, Chen, Doris C

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Cross-Coupling of Alkynylsilanols with Aryl Halides Promoted by Potassium Trimethylsilanolate von Denmark, Scott E, Tymonko, Steven A

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Impact of ICH Q11 Questions and Answers on the Outcome of Active Pharmaceutical Ingredient Starting Material Proposal Acceptance by ICH Regulatory Members von Tymonko, Steven, Burke, Brenda J., Crochard, Jean-Philippe, Dirat, Olivier, Fraunhoffer, Kenneth J., Harrison, Cristian, Kramer, Timothy, Lee, Heewon, Liberman, Vlad, Sidhu, Kanwar P. S., Smith, Randi, Strotman, Neil A., Tandogan, Nil, Triman, Alan, Zhang, Haitao

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Development of a Commercial Process for Deucravacitinib, a Deuterated API for TYK2 Inhibition von Treitler, Daniel S, Soumeillant, Maxime C, Simmons, Eric M, Lin, Dong, Inankur, Bahar, Rogers, Amanda J, Dummeldinger, Michael, Kolotuchin, Sergei, Chan, Collin, Li, Jun, Freitag, Adam, Lora Gonzalez, Federico, Smith, Michael J, Sfouggatakis, Chris, Wang, Jianji, Benkovics, Tamas, Deerberg, Joerg, Simpson, James H, Chen, Ke, Tymonko, Steven

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Oxidation of benzoins to benzils using bismuth(III) nitrate-copper(II) acetate von Tymonko, Steven A., Nattier, Bryce A., Mohan, Ram S.

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A Scalable Synthesis of ( R , R )-2,6-Dimethyldihydro-2 H -pyran-4(3 H )-one von Young, Ian S., Haley, Matthew W., Tam, Annie, Tymonko, Steven A., Xu, Zhongmin, Hanson, Ronald L., Goswami, Animesh

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The Delivery of Flexibility from the Application of QbD to API Development von Popkin, Matt E., Borman, Phil J., Omer, Batool Ahmed, Seibert, Kevin D., Srivastava, Sushil, Lepore, John V., Hobson, Lindsay, Donaubauer, John, Curran, Timothy, Ide, Nathan, Tymonko, Steven, Looker, Adam, Kallemeyn, Jeffrey M.

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Formation of scalemic α,β-epoxysulfones von Dorow, R.L., Tymonko, Steven A.

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ChemInform Abstract: A Scalable Synthesis of (R,R)‐2,6‐Dimethyldihydro‐2H‐pyran‐4(3H)‐one von Young, Ian S., Haley, Matthew W., Tam, Annie, Tymonko, Steven A., Xu, Zhongmin, Hanson, Ronald L., Goswami, Animesh

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PROCESS FOR THE PREPARATION OF 6-(CYCLOPROPANEAMIDO)-4-((2-METHOXY-3-(1-METHYL-1H-1,2,4-TRIAZOL-3-YL)PHENYL)AMINO)-N-(METHYL-D3)PYRIDAZINE-3-CARBOXAMIDE von SOUMEILLANT, Maxime C. D, TREITLER, Daniels S, WANG, Jianji, ROGERS, Amanda J, KOLOTUCHIN, Sergei V, CHEN, Ke, LI, Jun, BENKOVICS, Tamas, ROSSO, Victor W, TYMONKO, Steven, ZHENG, Bin, INANKUR, Bahar, SMITH, Michael J, DEERBERG, Joerg, LIN, Dong, DUMMELDINGER, Michael, SIMMONS, Eric M, STROTMAN, Neil A

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PROCESS FOR THE PREPARATION OF 6-(CYCLOPROPANEAMIDO)-4-((2-METHOXY-3-(1-METHYL-1H-1,2,4-TRIAZOL-3-YL)PHENYL)AMINO)-N-(METHYL-D3)PYRIDAZINE-3-CARBOXAMIDE von SOUMEILLANT, Maxime C. D, TREITLER, Daniels S, WANG, Jianji, ROGERS, Amanda J, KOLOTUCHIN, Sergei V, CHEN, Ke, LI, Jun, BENKOVICS, Tamas, ROSSO, Victor W, TYMONKO, Steven, ZHENG, Bin, INANKUR, Bahar, SMITH, Michael J, DEERBERG, Joerg, LIN, Dong, DUMMELDINGER, Michael, SIMMONS, Eric M, STROTMAN, Neil A

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PROCESS FOR THE PREPARATION OF 6-(CYCLOPROPANEAMIDO)-4-((2-METHOXY-3-(1-METHYL-1H-1,2,4-TRIAZOL-3-YL)PHENYL)AMINO)-N-(METHYL-D3)PYRIDAZINE-3-CARBOXAMIDE von TREITLER, Daniel S, SOUMEILLANT, Maxime C. D, WANG, Jianji, ROGERS, Amanda J, KOLOTUCHIN, Sergei V, CHEN, Ke, LI, Jun, BENKOVICS, Tamas, ROSSO, Victor W, TYMONKO, Steven, ZHENG, Bin, INANKUR, Bahar, SMITH, Michael J, DEERBERG, Joerg, LIN, Dong, DUMMELDINGER, Michael, SIMMONS, Eric M, STROTMAN, Neil A

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PROCESS FOR THE PREPARATION OF 6-(CYCLOPROPANEAMIDO)-4-((2-METHOXY-3-(1-METHYL-1H-1,2,4-TRIAZOL-3-YL)PHENYL)AMINO)-N-(METHYL-D3)PYRIDAZINE-3-CARBOXAMIDE von Inankur, Bahar, Treitler, Daniel S, Dummeldinger, Michael, Rogers, Amanda J, Zheng, Bin, Lin, Dong, Benkovics, Tamas, Strotman, Neil A, Chen, Ke, Simmons, Eric M, Soumeillant, Maxime C.D, Smith, Michael J, Rosso, Victor W, Kolotuchin, Sergei, Tymonko, Steven, Deerberg, Joerg, Wang, Jianji, Li, Jun

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