Nine-Step Stereoselective Synthesis of Islatravir from Deoxyribose von Nawrat, Christopher C, Whittaker, Aaron M, Huffman, Mark A, McLaughlin, Mark, Cohen, Ryan D, Andreani, Teresa, Ding, Bangwei, Li, Hongming, Weisel, Mark, Tschaen, David M

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A Mild Cu(I)-Catalyzed Oxidative Aromatization of Indolines to Indoles von Peng, Feng, McLaughlin, Mark, Liu, Yizhou, Mangion, Ian, Tschaen, David M, Xu, Yingju

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Synthesis of Islatravir Enabled by a Catalytic, Enantioselective Alkynylation of a Ketone von Patel, Niki R., Nawrat, Christopher C., McLaughlin, Mark, Xu, Yingju, Huffman, Mark A., Yang, Hao, Li, Hongming, Whittaker, Aaron M., Andreani, Teresa, Lévesque, François, Fryszkowska, Anna, Brunskill, Andrew, Tschaen, David M., Maloney, Kevin M.

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Oxidation of Primary Alcohols to Carboxylic Acids with Sodium Chlorite Catalyzed by TEMPO and Bleach von Zhao, Mangzhu, Li, Jing, Mano, Eiichi, Song, Zhiguo, Tschaen, David M, Grabowski, Edward J. J, Reider, Paul J

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Practical Asymmetric Synthesis of an Endothelin Receptor Antagonist von Song, Zhiguo J, Zhao, Mangzhu, Desmond, Richard, Devine, Paul, Tschaen, David M, Tillyer, Richard, Frey, Lisa, Heid, Richard, Xu, Feng, Foster, Bruce, Li, Jing, Reamer, Robert, Volante, Ralph, Dolling, Ulf H, Reider, Paul J, Okada, Shigemitsu, Kato, Yoshiaki, Mano, Eiichi

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Merck’s Reaction Review Policy: An Exercise in Process Safety von Bassan, Ephraim, Ruck, Rebecca T, Dienemann, Erik, Emerson, Khateeta M, Humphrey, Guy R, Raheem, Izzat T, Tschaen, David M, Vickery, Thomas P, Wood, Harold B, Yasuda, Nobuyoshi

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Highly Selective Cascade Couplings for the Syntheses of Functionalized Piperidinones and Bispidines von Xu, Feng, Corley, Edward, Murry, Jerry A, Tschaen, David M

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Practical Synthesis of A Macrocyclic HCV Protease Inhibitor: A High-Yielding Macrolactam Formation von Song, Zhiguo J, Tellers, David M, Dormer, Peter G, Zewge, Daniel, Janey, Jacob M, Nolting, Andrew, Steinhuebel, Dietrich, Oliver, Steven, Devine, Paul N, Tschaen, David M

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Efficient Synthesis of Losartan, A Nonpeptide Angiotensin II Receptor Antagonist von Larsen, Robert D, King, Anthony O, Chen, Cheng Y, Corley, Edward G, Foster, Bruce S, Roberts, F. Edward, Yang, Chunhua, Lieberman, David R, Reamer, Robert A, Tschaen, David M, Verhoeven, Thomas R, Reider, Paul J, Lo, Young S, Rossano, Lucius T, Brookes, A. Sidney, Meloni, David, Moore, James R, Arnett, John F

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Practical Asymmetric Synthesis of a Selective Endothelin A Receptor (ETA) Antagonist von Song, Zhiguo J, Zhao, Matthew, Frey, Lisa, Li, Jing, Tan, Lushi, Chen, Cheng Y, Tschaen, David M, Tillyer, Richard, Grabowski, Edward J. J, Volante, Ralph, Reider, Paul J, Kato, Yoshiaki, Okada, Shigemitsu, Nemoto, Takayuki, Sato, Hiroki, Akao, Atsushi, Mase, Toshiaki

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Practical synthesis of a potent indolocarbazole-based, DNA topoisomerase inhibitor von Akao, Atsushi, Hiraga, Shouichi, Iida, Takehiko, Kamatani, Asayuki, Kawasaki, Masashi, Mase, Toshiaki, Nemoto, Takayuki, Satake, Nobuya, Weissman, Steven A, Tschaen, David M, Rossen, Kai, Petrillo, Daniel, Reamer, Robert A, Volante, R.P

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Correction to Synthesis of Vaniprevir (MK-7009): Lactamization To Prepare a 22-Membered Macrocycle von Song, Zhiguo J, Tellers, David M, Journet, Michel, Kuethe, Jeffrey T, Lieberman, David, Humphrey, Guy, Zhang, Fei, Peng, Zhihui, Waters, Marjorie S, Zewge, Daniel, Nolting, Andrew, Zhao, Dalian, Reamer, Robert A, Dormer, Peter G, Belyk, Kevin M, Davies, Ian W, Devine, Paul N, Tschaen, David M

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Preparative Chromatography with Extreme Productivity: HPLC Preparation of an Isomerically Pure Drug Intermediate on Multikilogram Scale von Welch, Christopher J, Henderson, Derek W, Tschaen, David M, Miller, Ross A

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Efficient Synthesis of a Highly Selective NPY-5 Receptor Antagonist:  A Drug Candidate for the Treatment of Obesity von Itoh, Takahiro, Kato, Shinji, Nonoyama, Nobuaki, Wada, Toshihiro, Maeda, Kenji, Mase, Toshiaki, Zhao, Matthew M, Song, Jake Z, Tschaen, David M, McNamara, James M

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Asymmetric Synthesis of MK-0499 von Tschaen, David M, Abramson, Lee, Cai, Dongwei, Desmond, Richard, Dolling, Ulf-H, Frey, Lisa, Karady, Sandor, Shi, Yao-Jun, Verhoeven, Thomas R

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Stereoselective synthesis of 2-aryloxy esters: An asymmetric approach to fluoxetine, tomoxetine and nisoxetine von Devine, Paul N, Heid, Richard M, Tschaen, David M

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