WAY‐318068: a novel, potent and selective noradrenaline re‐uptake inhibitor with activity in rodent models of pain and depression von Whiteside, GT, Dwyer, JM, Harrison, JE, Beyer, CE, Cummons, T, Manzino, L, Mark, L, Johnston, GH, Strassle, BW, Adedoyin, A, Lu, P, Piesla, MJ, Pulicicchio, CM, Erve, JCL, Platt, BJ, Hughes, ZA, Rogers, KE, Deecher, DC, Trybulski, EJ, Kennedy, JD, Zhang, P, Leventhal, L

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The design, synthesis and physical chemical properties of novel human vasopressin V2-receptor antagonists optimized for parenteral delivery von ASHWELL, M. A, BAGLI, J. F, WILLIAMS, D. K, CAGGIANO, T. J, CHAN, P. S, MOLINARI, A. J, PALKA, C, PARK, C. H, ROGERS, J. F, SHERMAN, M, TRYBULSKI, E. J

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The synthesis and biochemical pharmacology of enantiomerically pure methylated oxotremorine derivatives von Trybulski, Eugene J, Zhang, Jing, Kramss, Richard H, Mangano, Richard M

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Chemical and biochemical studies of 2-propynylpyrrolidine derivatives. Restricted-rotation analogs of N-methyl-N-(1-methyl-4-pyrrolidino-2-butynyl)acetamide (BM-5) von Trybulski, Eugene J, Kramss, Richard H, Mangano, Richard M, Rusinko, Andrew

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2-Benzazepines. 9. Synthesis and chemistry of 3H-2-benzazepine and pyrimido[4,5-d][2]benzazepine derivatives von Trybulski, E. J, Fryer, R. I, Reeder, E, Vitone, S, Todaro, L

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Anti-arrhythmic agents von Trybulski, Eugene J

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Synthesis and activity of a new class of pathway-selective estrogen receptor ligands: Hydroxybenzoyl-3,4-dihydroquinoxalin-2(1 H)-ones von Mahaney, Paige E., Webb, Michael B., Ye, Fei, Sabatucci, Joseph P., Steffan, Robert J., Chadwick, Christopher C., Harnish, Douglas C., Trybulski, Eugene J.

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Pyridobenzodiazepines: A novel class of orally active, vasopressin V 2 receptor selective agonists von Failli, Amedeo A., Shumsky, Jay S., Steffan, Robert J., Caggiano, Thomas J., Williams, David K., Trybulski, Eugene J., Ning, Xiaoping, Lock, Yeungwai, Tanikella, Tarak, Hartmann, David, Chan, Peter S., Park, C.H.

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2-Benzazepines. 4. [1,2,3]Triazolo[4,5-d][2]benzazepines and dibenzo[c,f][1,2,3]triazolo[3,4-a]azepines: synthesis and evaluation as central nervous system agents von Trybulski, E J, Benjamin, L, Vitone, S, Walser, A, Fryer, R I

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2-Benzazepines. 6. Synthesis and pharmacological properties of the metabolites of 9-chloro-7-(2-chlorophenyl)-5H-pyrimido[5,4-d][2]benzazepine von Trybulski, Eugene J, Fryer, R. Ian, Reeder, Earl, Walser, Armin, Blount, John

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Quinazolines and 1,4-benzodiazepines. 90. Structure-activity relationship between substituted 2-amino-N-(2-benzoyl-4-chlorophenyl)acetamides and 1,4-benzodiazepinones von Fryer, R I, Leimgruber, W, Trybulski, E J

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2-Benzazepines. [1,2,3]Triazolo[4,5-d][2]benzazepines and dibenzo[c,f][1,2,3]triazolo[3,4-a]azepines. Synthesis and evaluation as central nervous system agents von Trybulski, E. J, Benjamin, L, Vitone, S, Walser, A, Fryer, R. I

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2-Benzazepines. 5. Synthesis of pyrimido[5,4-d][2]benzazepines and their evaluation as anxiolytic agents von Trybulski, Eugene J, Benjamin, Louis E, Earley, James V, Fryer, R. Ian, Gilman, Norman W, Reeder, Earl, Walser, Armin, Davidson, Arnold B, Horst, W. Dale

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2-Benzazepines. 2. Thiazolo[5,4-d][2]benzazepines von Benjamin, Louis E, Fryer, R. Ian, Gilman, Norman W, Trybulski, Eugene J

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The design, synthesis and physical chemical properties of novel human vasopressin V 2 -receptor antagonists optimized for parenteral delivery von Ashwell, M.A, Bagli, J.F, Caggiano, T.J, Chan, P.S, Molinari, A.J, Palka, C, Park, C.H, Rogers, J.F, Sherman, M, Trybulski, E.J, Williams, D.K

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A new protecting group for the carbonyl function von Corey, E.J., Trybulski, E.J., William Suggs, J.

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Synthetic approach to the skeleton of histrionicotoxin von Tufariello, Joseph J, Trybulski, Eugene J

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Synthesis in the tropane class of alkaloids. Pseudotropine and dl-cocaine von Tufariello, Joseph J, Mullen, George B, Tegeler, John J, Trybulski, Eugene J, Wong, Shing Chun, Ali, S. Asrof

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Total synthesis of erythromycins. 4. Total synthesis of erythronolide B von Corey, E. J, Kim, Sunggak, Yoo, Sung-Eun, Nicolaou, K. C, Melvin, Lawrence S, Brunelle, Daniel J, Falck, J. R, Trybulski, Eugene J, Lett, Robert, Sheldrake, Peter W

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The synthesis and structure activity relationships of enantiomerically pure hydroxylated oxotremorine derivatives von Trybulski, Eugene J., Kramss, Richard H., Mangano, Richard M., Brabander, Herbert J., Francisco, Gerardo

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