Structure-Based Design, Synthesis, and Biological Evaluation of Irreversible Human Rhinovirus 3C Protease Inhibitors. 6. Structure−Activity Studies of Orally Bioavailable, 2-Pyrido... von Dragovich, Peter S, Prins, Thomas J, Zhou, Ru, Brown, Edward L, Maldonado, Fausto C, Fuhrman, Shella A, Zalman, Leora S, Tuntland, Tove, Lee, Caroline A, Patick, Amy K, Matthews, David A, Hendrickson, Thomas F, Kosa, Maha B, Liu, Bo, Batugo, Minerva R, Gleeson, Jean-Paul R, Sakata, Sylvie K, Chen, Lijian, Guzman, Mark C, Meador, James W, Ferre, Rose Ann, Worland, Stephen T

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Benzothiophene containing Rho kinase inhibitors: Efficacy in an animal model of glaucoma von Davis, Robert L., Kahraman, Mehmet, Prins, Thomas J., Beaver, Yan, Cook, Travis G., Cramp, Jessica, Cayanan, Charmagne S., Gardiner, Elisabeth M.M., McLaughlin, Marsha A., Clark, Abbot F., Hellberg, Mark R., Shiau, Andrew K., Noble, Stewart A., Borchardt, Allen J.

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Structure-Based Design, Synthesis, and Biological Evaluation of Irreversible Human Rhinovirus 3C Protease Inhibitors. 8. Pharmacological Optimization of Orally Bioavailable 2-Pyrid... von Dragovich, Peter S, Prins, Thomas J, Zhou, Ru, Johnson, Theodore O, Hua, Ye, Luu, Hiep T, Sakata, Sylvie K, Brown, Edward L, Maldonado, Fausto C, Tuntland, Tove, Lee, Caroline A, Fuhrman, Shella A, Zalman, Leora S, Patick, Amy K, Matthews, David A, Wu, Ellen Y, Guo, Ming, Borer, Bennett C, Nayyar, Naresh K, Moran, Terence, Chen, Lijian, Rejto, Paul A, Rose, Peter W, Guzman, Mark C, Dovalsantos, Elena Z, Lee, Steven, McGee, Kevin, Mohajeri, Michael, Liese, Andreas, Tao, Junhua, Kosa, Maha B, Liu, Bo, Batugo, Minerva R, Gleeson, Jean-Paul R, Wu, Zhen Ping, Liu, Jia, Meador, James W, Ferre, Rose Ann

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Structure-Based Design, Synthesis, and Biological Evaluation of Irreversible Human Rhinovirus 3C Protease Inhibitors. 4. Incorporation of P1 Lactam Moieties as l-Glutamine Replacem... von Dragovich, Peter S, Prins, Thomas J, Zhou, Ru, Webber, Stephen E, Marakovits, Joseph T, Fuhrman, Shella A, Patick, Amy K, Matthews, David A, Lee, Caroline A, Ford, Clifford E, Burke, Benjamin J, Rejto, Paul A, Hendrickson, Thomas F, Tuntland, Tove, Brown, Edward L, Meador, James W, Ferre, Rose Ann, Harr, James E. V, Kosa, Maha B, Worland, Stephen T

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Structure-Based Design, Synthesis, and Biological Evaluation of Irreversible Human Rhinovirus 3C Protease Inhibitors. Part 7: Structure–Activity Studies of Bicyclic 2-Pyridone-Cont... von Dragovich, Peter S., Prins, Thomas J., Zhou, Ru, Johnson, Theodore O., Brown, Edward L., Maldonado, Fausto C., Fuhrman, Shella A., Zalman, Leora S., Patick, Amy K., Matthews, David A., Hou, Xinjun, Meador, James W., Ferre, Rose Ann, Worland, Stephen T.

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Synthesis of an Optically Active, Bicyclic 2-Pyridone Dipeptide Mimetic von Dragovich, Peter S., Zhou, Ru, Prins, Thomas J.

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Structure-Based Design, Synthesis, and Biological Evaluation of Irreversible Human Rhinovirus 3C Protease Inhibitors. 3. Structure−Activity Studies of Ketomethylene-Containing Pept... von Dragovich, Peter S, Prins, Thomas J, Zhou, Ru, Fuhrman, Shella A, Patick, Amy K, Matthews, David A, Ford, Clifford E, Meador, James W, Ferre, Rose Ann, Worland, Stephen T

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Structure-based design of ketone-containing, tripeptidyl human rhinovirus 3C protease inhibitors von DRAGOVICH, P. S, RU ZHOU, MEADOR, J. W, PATICK, A. K, FORD, C. E, BROTHERS, M. A, BINFORD, S. L, MATTHEWS, D. A, FERRE, R. A, WORLAND, S. T, WEBBER, S. E, PRINS, T. J, KWOK, A. K, OKANO, K, FUHRMAN, S. A, ZALMAN, L. S, MALDONADO, F. C, BROWN, E. L

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Chemoenzymic synthesis of 2-amino-3-(2,2'-bipyridinyl)propanoic acids von Imperiali, Barbara, Prins, Thomas J, Fisher, Stewart L

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Structure-Based Design of Novel, Urea-Containing FKBP12 Inhibitors von Dragovich, Peter S, Barker, John E, French, Judy, Imbacuan, Michael, Kalish, Vincent J, Kissinger, Charles R, Knighton, Daniel R, Lewis, Cristina T, Moomaw, Ellen W, Parge, Hans E, Pelletier, Laura A. K, Prins, Thomas J, Showalter, Richard E, Tatlock, John H, Tucker, Kathleen D, Villafranca, J. Ernest

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Palladium Catalyzed, Regioselective Reduction of 1,2-Epoxides by Ammonium Formate von Dragovich, Peter S, Prins, Thomas J, Zhou, Ru

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An optical thin film assay incorporating rhinovirus protease inhibitors as detector reagents von Ettinger, Anna, Ostroff, Rachel, Rhihanek, Marynette, Dragovich, Peter S, Zalman, Leora S, Patick, Amy K, Prins, Thomas J, Fuhrman, Shella A, Brown, Edward L, Worland, Stephen T, Polisky, Barry

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Structure-based design of irreversible, tripeptidyl human rhinovirus 3C protease inhibitors containing N-methyl amino acids von Dragovich, Peter S, Webber, Stephen E, Prins, Thomas J, Zhou, Ru, Marakovits, Joseph T, Tikhe, Jayashree G, Fuhrman, Shella A, Patick, Amy K, Matthews, David A, Ford, Clifford E, Brown, Edward L, Binford, Susan L, Meador, James W, Ferre, Rose Ann, Worland, Stephen T

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Design and synthesis of irreversible depsipeptidyl human rhinovirus 3C protease inhibitors von Webber, Stephen E., Marakovits, Joseph T., Dragovich, Peter S., Prins, Thomas J., Zhou, Ru, Fuhrman, Shella A., Patick, Amy K., Matthews, David A., Lee, Caroline A., Srinivasan, Babu, Moran, Terry, Ford, Clifford E., Brothers, Mary A., Harr, James E.V., Meador, James W., Ferre, Rose Ann, Worland, Stephen T.

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Formal, Stereoselective Synthesis of Hydroxyethylene Dipeptide Isosteres Utilizing Pseudoephedrine Amides von Dragovich, Peter S, Prins, Thomas J, Zhou, Ru

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Structure-Based Design, Synthesis, and Biological Evaluation of Irreversible Human Rhinovirus 3C Protease Inhibitors. 4. Incorporation of P 1 Lactam Moieties as l -Glutamine Replac... von Dragovich, Peter S., Prins, Thomas J., Zhou, Ru, Webber, Stephen E., Marakovits, Joseph T., Fuhrman, Shella A., Patick, Amy K., Matthews, David A., Lee, Caroline A., Ford, Clifford E., Burke, Benjamin J., Rejto, Paul A., Hendrickson, Thomas F., Tuntland, Tove, Brown, Edward L., Meador, James W., Ferre, Rose Ann, Harr, James E. V., Kosa, Maha B., Worland, Stephen T.

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Structure-Based Design, Synthesis, and Biological Evaluation of Irreversible Human Rhinovirus 3C Protease Inhibitors. 1. Michael Acceptor Structure−Activity Studies von Dragovich, Peter S, Webber, Stephen E, Babine, Robert E, Fuhrman, Shella A, Patick, Amy K, Matthews, David A, Lee, Caroline A, Reich, Siegfried H, Prins, Thomas J, Marakovits, Joseph T, Littlefield, Ethel S, Zhou, Ru, Tikhe, Jayashree, Ford, Clifford E, Wallace, Michael B, Meador, James W, Ferre, Rose Ann, Brown, Edward L, Binford, Susan L, Harr, James E. V, DeLisle, Dorothy M, Worland, Stephen T

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Structure-Based Design, Synthesis, and Biological Evaluation of Irreversible Human Rhinovirus 3C Protease Inhibitors. 2. Peptide Structure−Activity Studies von Dragovich, Peter S, Webber, Stephen E, Babine, Robert E, Fuhrman, Shella A, Patick, Amy K, Matthews, David A, Reich, Siegfried H, Marakovits, Joseph T, Prins, Thomas J, Zhou, Ru, Tikhe, Jayashree, Littlefield, Ethel S, Bleckman, Ted M, Wallace, Michael B, Little, Thomas L, Ford, Clifford E, Meador, James W, Ferre, Rose Ann, Brown, Edward L, Binford, Susan L, DeLisle, Dorothy M, Worland, Stephen T

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Cyclopentadienyl(allyl)(butadiene)hafnium compounds. Synthesis, crystal structure, and dynamics of cyclopentadienyl(1,2,3-trimethylallyl)(1,2-dimethylbutadiene)hafnium and cyclopen... von Prins, Thomas J, Hauger, Bryan E, Vance, Peter J, Wemple, Michael E, Kort, David A, O'Brien, Jonathan P, Silver, Michael E, Huffman, John C

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Chemoenzymatic synthesis of 2-amino-3-(2,2'-bipyridinyl)propanoic acids von IMPERIALI, B, PRINS, T. J, FISHER, S. L

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