Residue-wise local quality estimation for protein models from cryo-EM maps von Terashi, Genki, Wang, Xiao, Maddhuri Venkata Subramaniya, Sai Raghavendra, Tesmer, John J. G., Kihara, Daisuke

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Hitchhiking on the heptahelical highway: structure and function of 7TM receptor complexes von Tesmer, John J. G.

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Molecular basis for Gβγ-mediated activation of phosphoinositide 3-kinase γ von Chen, Chun-Liang, Syahirah, Ramizah, Ravala, Sandeep K., Yen, Yu-Chen, Klose, Thomas, Deng, Qing, Tesmer, John J. G.

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Structure and function of lysosomal phospholipase A2 and lecithin:cholesterol acyltransferase von Glukhova, Alisa, Hinkovska-Galcheva, Vania, Kelly, Robert, Abe, Akira, Shayman, James A., Tesmer, John J. G.

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Structure of adenylyl cyclase 5 in complex with Gβγ offers insights into ADCY5-related dyskinesia von Yen, Yu-Chen, Li, Yong, Chen, Chun-Liang, Klose, Thomas, Watts, Val J., Dessauer, Carmen W., Tesmer, John J. G.

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Structure and Function of Heterotrimeric G Protein-Regulated Rho Guanine Nucleotide Exchange Factors von Aittaleb, Mohamed, Boguth, Cassandra A, Tesmer, John J G

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Structure-Based Design, Synthesis, and Biological Evaluation of Highly Selective and Potent G Protein-Coupled Receptor Kinase 2 Inhibitors von Waldschmidt, Helen V, Homan, Kristoff T, Cruz-Rodríguez, Osvaldo, Cato, Marilyn C, Waninger-Saroni, Jessica, Larimore, Kelly M, Cannavo, Alessandro, Song, Jianliang, Cheung, Joseph Y, Kirchhoff, Paul D, Koch, Walter J, Tesmer, John J. G, Larsen, Scott D

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GRK2 inhibitors, paroxetine and CCG258747, attenuate IgE-mediated anaphylaxis but activate mast cells via MRGPRX2 and MRGPRB2 von Thapaliya, Monica, Amponnawarat, Aetas, Tesmer, John J G, Ali, Hydar

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GRK2 kinases in the primary cilium initiate SMOOTHENED-PKA signaling in the Hedgehog cascade von Walker, Madison F, Zhang, Jingyi, Steiner, William, Ku, Pei-I, Zhu, Ju-Fen, Michaelson, Zachary, Yen, Yu-Chen, Lee, Annabel, Long, Alyssa B, Casey, Mattie J, Poddar, Abhishek, Nelson, Isaac B, Arveseth, Corvin D, Nagel, Falko, Clough, Ryan, LaPotin, Sarah, Kwan, Kristen M, Schulz, Stefan, Stewart, Rodney A, Tesmer, John J G, Caspary, Tamara, Subramanian, Radhika, Ge, Xuecai, Myers, Benjamin R

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G Protein-Coupled Receptor Kinase 2 (GRK2) and 5 (GRK5) Exhibit Selective Phosphorylation of the Neurotensin Receptor in Vitro von Inagaki, Sayaka, Ghirlando, Rodolfo, Vishnivetskiy, Sergey A, Homan, Kristoff T, White, Jim F, Tesmer, John J. G, Gurevich, Vsevolod V, Grisshammer, Reinhard

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Molecular mechanism of selectivity among G protein-coupled receptor kinase 2 inhibitors von Thal, David M, Yeow, Raymond Y, Schoenau, Christian, Huber, Jochen, Tesmer, John J G

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Identification and Structure–Function Analysis of Subfamily Selective G Protein-Coupled Receptor Kinase Inhibitors von Homan, Kristoff T, Larimore, Kelly M, Elkins, Jonathan M, Szklarz, Marta, Knapp, Stefan, Tesmer, John J. G

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Structural and Functional Analysis of the Regulator of G Protein Signaling 2-Gαq Complex von Nance, Mark R., Kreutz, Barry, Tesmer, Valerie M., Sterne-Marr, Rachel, Kozasa, Tohru, Tesmer, John J.G.

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Monomeric Rhodopsin Is Sufficient for Normal Rhodopsin Kinase (GRK1) Phosphorylation and Arrestin-1 Binding von Bayburt, Timothy H., Vishnivetskiy, Sergey A., McLean, Mark A., Morizumi, Takefumi, Huang, Chih-chin, Tesmer, John J.G., Ernst, Oliver P., Sligar, Stephen G., Gurevich, Vsevolod V.

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Molecular Mechanism for Inhibition of G Protein-Coupled Receptor Kinase 2 by a Selective RNA Aptamer von Tesmer, Valerie M., Lennarz, Sabine, Mayer, Günter, Tesmer, John J.G.

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Structural Basis of Lysosomal Phospholipase A2 Inhibition by Zn2 von Bouley, Renee A, Hinkovska-Galcheva, Vania, Shayman, James A, Tesmer, John J. G

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Structure of the C-terminal guanine nucleotide exchange factor module of Trio in an autoinhibited conformation reveals its oncogenic potential von Bandekar, Sumit J, Arang, Nadia, Tully, Ena S, Tang, Brittany A, Barton, Brenna L, Li, Sheng, Gutkind, J Silvio, Tesmer, John J G

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Structure-Based Design of Highly Selective and Potent G Protein-Coupled Receptor Kinase 2 Inhibitors Based on Paroxetine von Waldschmidt, Helen V, Homan, Kristoff T, Cato, Marilyn C, Cruz-Rodríguez, Osvaldo, Cannavo, Alessandro, Wilson, Michael W, Song, Jianliang, Cheung, Joseph Y, Koch, Walter J, Tesmer, John J. G, Larsen, Scott D

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Structural insights into G protein-coupled receptor kinase function von Homan, Kristoff T, Tesmer, John JG

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Molecular Basis for Small Molecule Inhibition of G Protein-Coupled Receptor Kinases von Homan, Kristoff T, Tesmer, John J. G

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