Discovery of (1R,2S)‑2-{[(2,4-Dimethylpyrimidin-5-yl)oxy]methyl}-2-(3-fluorophenyl)‑N‑(5-fluoropyridin-2-yl)cyclopropanecarboxamide (E2006): A Potent and Efficacious Oral Orexin Re... von Yoshida, Yu, Naoe, Yoshimitsu, Terauchi, Taro, Ozaki, Fumihiro, Doko, Takashi, Takemura, Ayumi, Tanaka, Toshiaki, Sorimachi, Keiichi, Beuckmann, Carsten T, Suzuki, Michiyuki, Ueno, Takashi, Ozaki, Shunsuke, Yonaga, Masahiro

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Synthesis and Evaluation of Novel Radioligands for Positron Emission Tomography Imaging of the Orexin‑2 Receptor von Oi, Norihito, Suzuki, Michiyuki, Terauchi, Taro, Tokunaga, Masaki, Nakatani, Yosuke, Yamamoto, Noboru, Fukumura, Toshimitsu, Zhang, Ming-Rong, Suhara, Tetsuya, Higuchi, Makoto

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Synthesis and pharmacological profile of serofendic acids A and B von Terauchi, Taro, Asai, Naoki, Doko, Takashi, Taguchi, Ryota, Takenaka, Osamu, Sakurai, Hideki, Yonaga, Masahiro, Kimura, Teiji, Kajiwara, Akiharu, Niidome, Tetsuhiro, Kume, Toshiaki, Akaike, Akinori, Sugimoto, Hachiro

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Isolation of a Diterpenoid Substance with Potent Neuroprotective Activity from Fetal Calf Serum von Kume, Toshiaki, Asai, Naoki, Nishikawa, Hiroyuki, Mano, Nariyasu, Terauchi, Taro, Taguchi, Ryota, Shirakawa, Hisashi, Osakada, Fumitaka, Mori, Hiroki, Asakawa, Naoki, Yonaga, Masahiro, Nishizawa, Yukio, Sugimoto, Hachiro, Shimohama, Shun, Katsuki, Hiroshi, Kaneko, Shuji, Akaike, Akinori

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Synthetic studies on altohyrtins (spongistatins): synthesis of the C15–C28 (CD) spiroacetal portion von Terauchi, Takeshi, Terauchi, Taro, Sato, Ippei, Tsukada, Tomoharu, Kanoh, Naoki, Nakata, Masaya

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Synthesis and absolute configuration of serofendic acids von Terauchi, Taro, Asai, Naoki, Yonaga, Masahiro, Kume, Toshiaki, Akaike, Akinori, Sugimoto, Hachiro

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Discovery of a New Class of mGluR2 Selective Group II mGluR NAM PET Tracer von Li, Zizhong, Hagiwara, Hiroaki, Takaishi, Mamoru, Teceno, Tyler, Krause, Stephen, sasaki, Takeo, McCracken, Paul, Koyama, Akihiko, Terauchi, Taro

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Design, synthesis, and structure–activity relationships of a series of novel N-aryl-2-phenylcyclopropanecarboxamide that are potent and orally active orexin receptor antagonists von Yoshida, Yu, Terauchi, Taro, Naoe, Yoshimitsu, Kazuta, Yuji, Ozaki, Fumihiro, Beuckmann, Carsten T., Nakagawa, Makoto, Suzuki, Michiyuki, Kushida, Ikuo, Takenaka, Osamu, Ueno, Takashi, Yonaga, Masahiro

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Design, synthesis and structure–activity relationships of 5-alkylaminolquinolines as a novel series of CRF1 receptor antagonists von Takeda, Kunitoshi, Terauchi, Taro, Shin, Kogyoku, Ino, Mitsuhiro, Shibata, Hisashi, Yonaga, Masahiro

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Design, synthesis, and structure–activity relationships of a series of 2-Ar-8-methyl-5-alkylaminoquinolines as novel CRF1 receptor antagonists von Takeda, Kunitoshi, Terauchi, Taro, Hashizume, Minako, Shin, Kogyoku, Ino, Mitsuhiro, Shibata, Hisashi, Yonaga, Masahiro

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Corrigendum to “Design, synthesis, and structure–activity relationships of a series of novel N-aryl-2-phenylcyclopropanecarboxamide that are potent and orally active orexin recepto... von Yoshida, Yu, Terauchi, Taro, Naoe, Yoshimitsu, Kazuta, Yuji, Ozaki, Fumihiro, Beuckmann, Carsten T., Nakagawa, Makoto, Suzuki, Michiyuki, Kushida, Ikuo, Takenaka, Osamu, Ueno, Takashi, Yonaga, Masahiro

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Design, Synthesis, and Structure–Activity Relationships of Novel Pyrazolo[5,1‑b]thiazole Derivatives as Potent and Orally Active Corticotropin-Releasing Factor 1 Receptor Antagonis... von Takahashi, Yoshinori, Hashizume, Minako, Shin, Kogyoku, Terauchi, Taro, Takeda, Kunitoshi, Hibi, Shigeki, Murata-Tai, Kaoru, Fujisawa, Masae, Shikata, Kodo, Taguchi, Ryota, Ino, Mitsuhiro, Shibata, Hisashi, Yonaga, Masahiro

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創薬科学賞受賞　AMPA型グルタミン酸受容体拮抗剤ペランパネルの創薬研究: (長戸　哲氏（代表研究者)，花田敬久氏，上野貢嗣氏，上野正孝氏，竹中　理氏）... von 寺内, 太朗

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Synthesis and structure–activity relationships of 8-substituted-2-aryl-5-alkylaminoquinolines: Potent, orally active corticotropin-releasing factor-1 receptor antagonists von Takeda, Kunitoshi, Terauchi, Taro, Hashizume, Minako, Shikata, Kohdoh, Taguchi, Ryota, Murata-Tai, Kaoru, Fujisawa, Masae, Takahashi, Yoshinori, Shin, Kogyoku, Ino, Mitsuhiro, Shibata, Hisashi, Yonaga, Masahiro

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Synthesis and neuroprotective effects of serofendic acid analogues von Terauchi, Taro, Doko, Takashi, Yonaga, Masahiro, Kajiwara, Akiharu, Niidome, Tetsuhiro, Taguchi, Ryota, Kume, Toshiaki, Akaike, Akinori, Sugimoto, Hachiro

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Formal total synthesis of altohyrtin C (spongistatin 2). Part 1: Aldol approach to unite AB and CD spiroacetals von Terauchi, Takeshi, Terauchi, Taro, Sato, Ippei, Shoji, Wataru, Tsukada, Tomoharu, Tsunoda, Takashi, Kanoh, Naoki, Nakata, Masaya

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Serofendic acid prevents acute glutamate neurotoxicity in cultured cortical neurons von Taguchi, Ryota, Nishikawa, Hiroyuki, Kume, Toshiaki, Terauchi, Taro, Kaneko, Shuji, Katsuki, Hiroshi, Yonaga, Masahiro, Sugimoto, Hachiro, Akaike, Akinori

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Formal total synthesis of altohyrtin C (spongistatin 2). Part 2: Construction of fully elaborated ABCD and EF fragments von Terauchi, Takeshi, Tanaka, Taisaku, Terauchi, Taro, Morita, Masataka, Kimijima, Kyoko, Sato, Ippei, Shoji, Wataru, Nakamura, Yasuhiro, Tsukada, Tomoharu, Tsunoda, Takashi, Hayashi, Gouichirou, Kanoh, Naoki, Nakata, Masaya

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O1F-3-5 Synthesis and Evaluation of Novel Radioligands for Positron Emission Tomography Imaging of the Orexin-2 Receptor von Norihito Oi, Michiyuki Suzuki, Taro Terauchi, Masaki Tokunaga, Yosuke Nakatani, Noboru Ymamoto, Toshimitsu Fukumura, Ming-Rong Zhang, tetsuya Suhara, Makoto Higuchi

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METHODS AND COMPOUNDS USEFUL IN THE SYNTHESIS OF OREXIN-2 RECEPTOR ANTAGONISTS von WILCOXEN, Annie, TAKEMURA, Ayumi, SORIMACHI, Keiichi, MONIZ, George, YOSHIDA, Yu, NAOE, Yoshimitsu, KAZUTA, Yuji, ZHANG, Huiming, LEE, Jaemoon, BENAYOUD, Farid, TERAUCHI, Taro, TANAKA, Toshiaki

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