Unifying Family A GPCR Theories of Activation von TEHAN, Benjamin G, BORTOLATO, Andrea, BLANEY, Frank E, WEIR, Malcolm P, MASON, Jonathan S

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Acetylcholine prioritises direct synaptic inputs from entorhinal cortex to CA1 by differential modulation of feedforward inhibitory circuits von Palacios-Filardo, Jon, Udakis, Matt, Brown, Giles A., Tehan, Benjamin G., Congreve, Miles S., Nathan, Pradeep J., Brown, Alastair J. H., Mellor, Jack R.

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Comparison of Orexin 1 and Orexin 2 Ligand Binding Modes Using X‑ray Crystallography and Computational Analysis von Rappas, Mathieu, Ali, Ammar A. E, Bennett, Kirstie A, Brown, Jason D, Bucknell, Sarah J, Congreve, Miles, Cooke, Robert M, Cseke, Gabriella, de Graaf, Chris, Doré, Andrew S, Errey, James C, Jazayeri, Ali, Marshall, Fiona H, Mason, Jonathan S, Mould, Richard, Patel, Jayesh C, Tehan, Benjamin G, Weir, Malcolm, Christopher, John A

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Structure of Class B GPCRs: new horizons for drug discovery von Bortolato, Andrea, Doré, Andrew S, Hollenstein, Kaspar, Tehan, Benjamin G, Mason, Jonathan S, Marshall, Fiona H

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Fragment and Structure-Based Drug Discovery for a Class C GPCR: Discovery of the mGlu5 Negative Allosteric Modulator HTL14242 (3-Chloro-5-[6-(5-fluoropyridin-2-yl)pyrimidin-4-yl]be... von Christopher, John A, Aves, Sarah J, Bennett, Kirstie A, Doré, Andrew S, Errey, James C, Jazayeri, Ali, Marshall, Fiona H, Okrasa, Krzysztof, Serrano-Vega, Maria J, Tehan, Benjamin G, Wiggin, Giselle R, Congreve, Miles

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Author Correction: Acetylcholine prioritises direct synaptic inputs from entorhinal cortex to CA1 by differential modulation of feedforward inhibitory circuits von Palacios-Filardo, Jon, Udakis, Matt, Brown, Giles A., Tehan, Benjamin G., Congreve, Miles S., Nathan, Pradeep J., Brown, Alastair J. H., Mellor, Jack R.

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Selective Negative Allosteric Modulation Of Metabotropic Glutamate Receptors – A Structural Perspective of Ligands and Mutants von Harpsøe, Kasper, Isberg, Vignir, Tehan, Benjamin G., Weiss, Dahlia, Arsova, Angela, Marshall, Fiona H., Bräuner-Osborne, Hans, Gloriam, David E.

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Mutagenic Mapping Suggests a Novel Binding Mode for Selective Agonists of M1 Muscarinic Acetylcholine Receptors von Lebon, Guillaume, Langmead, Christopher J, Tehan, Ben G, Hulme, Edward C

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Comparisons of the HBV and HIV polymerase, and antiviral resistance mutations von BARTHOLOMEUSZ, Angeline, TEHAN, Benjamin G, CHALMERS, David K

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Water Network Perturbation in Ligand Binding: Adenosine A2A Antagonists as a Case Study von Bortolato, Andrea, Tehan, Ben G, Bodnarchuk, Michael S, Essex, Jonathan W, Mason, Jonathan S

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Water network perturbation in ligand binding: adenosine A(2A) antagonists as a case study von Bortolato, Andrea, Tehan, Ben G, Bodnarchuk, Michael S, Essex, Jonathan W, Mason, Jonathan S

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Characterisation of inverse agonism of the orphan-G protein-coupled receptor GPR52 by cannabinoid ligands Cannabidiol and O-1918 von Stott, Lisa A., Brighton, Cheryl A., Brown, Jason, Mould, Richard, Bennett, Kirstie A., Newman, Robert, Currinn, Heather, Autore, Flavia, Higueruelo, Alicia P., Tehan, Benjamin G., MacSweeney, Cliona, O'Brien, Michael A., Watson, Steve P.

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From structure to clinic: Design of a muscarinic M1 receptor agonist with potential to treatment of Alzheimer's disease von Brown, Alastair J H, Bradley, Sophie J, Marshall, Fiona H, Brown, Giles A, Bennett, Kirstie A, Brown, Jason, Cansfield, Julie E, Cross, David M, de Graaf, Chris, Hudson, Brian D, Dwomoh, Louis, Dias, João M, Errey, James C, Hurrell, Edward, Liptrot, Jan, Mattedi, Giulio, Molloy, Colin, Nathan, Pradeep J, Okrasa, Krzysztof, Osborne, Greg, Patel, Jayesh C, Pickworth, Mark, Robertson, Nathan, Shahabi, Shahram, Bundgaard, Christoffer, Phillips, Keith, Broad, Lisa M, Goonawardena, Anushka V, Morairty, Stephen R, Browning, Michael, Perini, Francesca, Dawson, Gerard R, Deakin, John F W, Smith, Robert T, Sexton, Patrick M, Warneck, Julie, Vinson, Mary, Tasker, Tim, Tehan, Benjamin G, Teobald, Barry, Christopoulos, Arthur, Langmead, Christopher J, Jazayeri, Ali, Cooke, Robert M, Rucktooa, Prakash, Congreve, Miles S, Weir, Malcolm, Tobin, Andrew B

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Roof and Floor of the Muscarinic Binding Pocket: Variations in the Binding Modes of Orthosteric Ligands von Goodwin, J Alex, Hulme, Edward C, Langmead, Christopher J, Tehan, Ben G

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The use of conformationally thermostabilised GPCRs in drug discovery: application to fragment, structure and biophysical techniques von Tehan, Benjamin G, Christopher, John A

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Methodologies for the Examination of Water in GPCRs von Bortolato, Andrea, Tehan, Benjamin G., Smith, Robert T., Mason, Jonathan S.

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Orthosteric and allosteric modes of interaction of novel selective agonists of the M1 muscarinic acetylcholine receptor von Avlani, Vimesh A, Langmead, Christopher J, Guida, Elizabeth, Wood, Martyn D, Tehan, Ben G, Herdon, Hugh J, Watson, Jeannette M, Sexton, Patrick M, Christopoulos, Arthur

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A Consensus Neural Network-Based Technique for Discriminating Soluble and Poorly Soluble Compounds von Manallack, David T, Tehan, Benjamin G, Gancia, Emanuela, Hudson, Brian D, Ford, Martyn G, Livingstone, David J, Whitley, David C, Pitt, Will R

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Backward recall and benchmark effects of working memory von Bireta, Tamra J., Fry, Sheena E., Jalbert, Annie, Neath, Ian, Surprenant, Aimée M., Tehan, Gerald, Tolan, Georgina Anne

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Target similarity effects : Support for the parallel distributed processing assumptions von HUMPHREYS, M. S, TEHAN, G, O'SHEA, A, BOLLAND, S. W

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