Design of N‑Benzoxaborole Benzofuran GSK8175Optimization of Human Pharmacokinetics Inspired by Metabolites of a Failed Clinical HCV Inhibitor von Chong, Pek Y, Shotwell, J. Brad, Miller, John, Price, Daniel J, Maynard, Andy, Voitenleitner, Christian, Mathis, Amanda, Williams, Shawn, Pouliot, Jeffrey J, Creech, Katrina, Wang, Feng, Fang, Jing, Zhang, Huichang, Tai, Vincent W.-F, Turner, Elizabeth, Kahler, Kirsten M, Crosby, Renae, Peat, Andrew J

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Hepatitis C Replication Inhibitors That Target the Viral NS4B Protein von Miller, John F., Chong, Pek Y., Shotwell, J. Brad, Catalano, John G., Tai, Vincent W.-F., Fang, Jing, Banka, Anna L., Roberts, Christopher D., Youngman, Michael, Zhang, Huichang, Xiong, Zhiping, Mathis, Amanda, Pouliot, Jeffery J., Hamatake, Robert K., Price, Daniel J., Seal, John W., Stroup, Lisa L., Creech, Katrina L., Carballo, Luz H., Todd, Dan, Spaltenstein, Andrew, Furst, Sylvia, Hong, Zhi, Peat, Andrew J.

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Design and synthesis of spirocyclic compounds as HCV replication inhibitors by targeting viral NS4B protein von Tai, Vincent W.-F., Garrido, Dulce, Price, Daniel J., Maynard, Andrew, Pouliot, Jeffrey J., Xiong, Zhiping, Seal, John W., Creech, Katrina L., Kryn, Luz H., Baughman, Todd M., Peat, Andrew J.

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Imidazo[1,2-a]pyridines That Directly Interact with Hepatitis C NS4B: Initial Preclinical Characterization von Shotwell, J. Brad, Baskaran, Subramanian, Chong, Pek, Creech, Katrina L, Crosby, Renae M, Dickson, Hamilton, Fang, Jing, Garrido, Dulce, Mathis, Amanda, Maung, Jack, Parks, Derek J, Pouliot, Jeffrey J, Price, Daniel J, Rai, Roopa, Seal, John W, Schmitz, Uli, Tai, Vincent W. F, Thomson, Michael, Xie, Mi, Xiong, Zhiping Z, Peat, Andrew J

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Discovery and structure–activity relationship of 2-phenyl-oxazole-4-carboxamide derivatives as potent apoptosis inducers von Tai, Vincent W.-F., Sperandio, David, Shelton, Emma J., Litvak, Joane, Pararajasingham, Keith, Cebon, Ben, Lohman, Julia, Eksterowicz, John, Kantak, Seema, Sabbatini, Peter, Brown, Cindy, Zeitz, Jennifer, Reed, Chris, Maske, Bill, Graupe, Doris, Estevez, Alberto, Oeh, Jason, Wong, Darren, Ni, Yong, Sprengeler, Paul, Yee, Robert, Magill, Catherine, Neri, Anthony, Cai, Sui Xiong, Drewe, John, Qiu, Ling, Herich, John, Tseng, Ben, Kasibhatla, Shailaja, Spencer, Jeffrey R.

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Ruthenium-Catalyzed cis-Dihydroxylation of Alkenes: Scope and Limitations von Shing, Tony K. M., Tam, Eric K. W., Tai, Vincent W.-F., Chung, Ivan H. F., Jiang, Qin

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Novel, potent, selective, and orally bioavailable human βII-tryptase inhibitors von Sperandio, David, Tai, Vincent W.-F., Lohman, Julia, Hirschbein, Bernie, Mendonca, Rohan, Lee, Chang-Sun, Spencer, Jeffrey R., Janc, James, Nguyen, Margaret, Beltman, Jerlyn, Sprengeler, Paul, Scheerens, Heleen, Lin, Tong, Liu, Liang, Gadre, Ashwini, Kellogg, Alisha, Green, Michael J., McGrath, Mary E.

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Elaborate Manifold of Short Hydrogen Bond Arrays Mediating Binding of Active Site-directed Serine Protease Inhibitors von Katz, Bradley A., Elrod, Kyle, Verner, Erik, Mackman, Richard L., Luong, Christine, Shrader, William D., Sendzik, Martin, Spencer, Jeffrey R., Sprengeler, Paul A., Kolesnikov, Aleks, Tai, Vincent W.-F., Hui, Hon C., Guy Breitenbucher, J., Allen, Darin, Janc, James W.

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Stereoselective synthesis of β-linked TBDMS-protected chitobiose-asparagine: a versatile building block for amyloidogenic glycopeptides von Bosques, Carlos J, Tai, Vincent W.-F, Imperiali, Barbara

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Substrate specificity of N-acetylglucosaminyl(diphosphodolichol) N-acetylglucosaminyl transferase, a key enzyme in the dolichol pathway von Tai, Vincent W.-F, O'Reilly, Mary K, Imperiali, Barbara

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Model study for the incorporation of the ( syn, anti)-2-amino-1,3-diol functionality in carbocycles von Tai, Vincent W.-F., Imperiali, Barbara

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Enantiospecific Syntheses of Penta-N,O,O,O,O-acetylvalidamine and Penta-N,O,O,O,O-acetyl-2-epi-validamine von Shing, Tony K. M, Tai, Vincent W.-F

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Facile and Enantiospecific Syntheses of Goniotriol Analogues von Shing, Tony K. M, Tai, Vincent W.-F

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INDOLE DERIVATIVES AS INHIBITORS OF HISTONE DEACETYLASE von TAI VINCENT W.F, LEE CHANG-SUN, VERNER ERIK, BUGGY JOSEPH J, BALASUBRAMANIAN SRIRAM

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INDOLE DERIVATIVES AS INHIBITORS OF HISTONE DEACETYLASE von TAI VINCENT W.F, LEE CHANG-SUN, VERNER ERIK, BUGGY JOSEPH J, BALASUBRAMANIAN SRIRAM

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(–)-Quinic acid in organic synthesis. Part 4. Syntheses of cyclophellitol and its (1R, 6S)-, (2S)-, (1R, 2S, 6S)-diastereoisomers von Shing, Tony K. M., Tai, Vincent W.-F.

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Certain Nitrogen Containing Bicyclic Chemical Entities For Treating Viral Infections von TAI VINCENT W.F, BASKARAN SUBRAMANIAN, ABADI ALI DEHGHANI MOHAMMAD, RAL ROOPA, SCHMITZ FRANZ ULRICH, SLOBODOV IRINA, MAUNG JACK, ROBERTS CHRISTOPHER DON, NEITZEL MARTIN LEON

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Facile syntheses of cyclopnellitol and its (1R,6S)-, (1R,2S,6S)-, (2S)-diastereoisomers from (–)-quinic acid von Shing, Tony K. M., Tai, Vincent W.-F.

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Substrate Specificity of the Glycosyl Donor for Oligosaccharyl Transferase von Tai, Vincent W.-F, Imperiali, Barbara

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