Pathophysiological Role and Medicinal Chemistry of A2A Adenosine Receptor Antagonists in Alzheimer’s Disease von Merighi, Stefania, Borea, Pier Andrea, Varani, Katia, Vincenzi, Fabrizio, Travagli, Alessia, Nigro, Manuela, Pasquini, Silvia, Suresh, R. Rama, Kim, Sung Won, Volkow, Nora D., Jacobson, Kenneth A., Gessi, Stefania

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Ligand design by targeting a binding site water von Matricon, Pierre, Suresh, R. Rama, Gao, Zhan-Guo, Panel, Nicolas, Jacobson, Kenneth A, Carlsson, Jens

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Pharmacological characterization of DPTN and other selective A3 adenosine receptor antagonists von Gao, Zhan-Guo, Suresh, R. Rama, Jacobson, Kenneth A.

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Expanding the repertoire of methanocarba nucleosides from purinergic signaling to diverse targets von Jacobson, Kenneth A, Salmaso, Veronica, Suresh, R. Rama, Tosh, Dilip K

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Design and in vivo activity of A3 adenosine receptor agonist prodrugs von Suresh, R. Rama, Jain, Shanu, Chen, Zhoumou, Tosh, Dilip K., Ma, Yanling, Podszun, Maren C., Rotman, Yaron, Salvemini, Daniela, Jacobson, Kenneth A.

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Fluorescent A2A and A3 adenosine receptor antagonists as flow cytometry probes von Toti, Kiran S., Campbell, Ryan G., Lee, Hobin, Salmaso, Veronica, Suresh, R. Rama, Gao, Zhan-Guo, Jacobson, Kenneth A.

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Convergent synthesis of 2-thioether-substituted ()-methanocarba-adenosines as purine receptor agonists von Suresh, R. Rama, Poe, Russell B, Lin, Baorui, Lv, Kexin, Campbell, Ryan G, Gao, Zhan-Guo, Liston, Theodore E, Toti, Kiran S, Jacobson, Kenneth A

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Nucleotide P2Y1 receptor agonists are in vitro and in vivo prodrugs of A1/A3 adenosine receptor agonists: implications for roles of P2Y1 and A1/A3 receptors in physiology and patho... von Liston, Theodore E., Hinz, Sonja, Müller, Christa E., Holstein, Deborah M., Wendling, Jay, Melton, Roger J., Campbell, Mary, Korinek, William S., Suresh, R. Rama, Sethre-Hofstad, Dane A., Gao, Zhan-Guo, Tosh, Dilip K., Jacobson, Kenneth A., Lechleiter, James D.

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Activation of adenosine A2A or A2B receptors causes hypothermia in mice von Carlin, Jesse Lea, Jain, Shalini, Duroux, Romain, Suresh, R. Rama, Xiao, Cuiying, Auchampach, John A., Jacobson, Kenneth A., Gavrilova, Oksana, Reitman, Marc L.

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Allosteric Antagonism of the A2A Adenosine Receptor by a Series of Bitopic Ligands von Gao, Zhan-Guo, Toti, Kiran S., Campbell, Ryan, Suresh, R. Rama, Yang, Huijun, Jacobson, Kenneth A.

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Lipid Trolling to Optimize A3 Adenosine Receptor-Positive Allosteric Modulators (PAMs) von Pradhan, Balaram, Pavan, Matteo, Fisher, Courtney L., Salmaso, Veronica, Wan, Tina C., Keyes, Robert F., Rollison, Noah, Suresh, R. Rama, Kumar, T. Santhosh, Gao, Zhan-Guo, Smith, Brian C., Auchampach, John A., Jacobson, Kenneth A.

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Palladium-Catalyzed Annulation of Allenes with Indole-2-carboxylic Acid Derivatives: Synthesis of Indolo[2,3‑c]pyrane-1-ones via Ar–I Reactivity or C–H Functionalization von Suresh, R. Rama, Swamy, K. C. Kumara

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Lipid Trolling to Optimize A 3 Adenosine Receptor-Positive Allosteric Modulators (PAMs) von Pradhan, Balaram, Pavan, Matteo, Fisher, Courtney L, Salmaso, Veronica, Wan, Tina C, Keyes, Robert F, Rollison, Noah, Suresh, R Rama, Kumar, T Santhosh, Gao, Zhan-Guo, Smith, Brian C, Auchampach, John A, Jacobson, Kenneth A

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Structure–Activity Studies of 1H‑Imidazo[4,5‑c]quinolin-4-amine Derivatives as A3 Adenosine Receptor Positive Allosteric Modulators von Fallot, Lucas B., Suresh, R. Rama, Fisher, Courtney L., Salmaso, Veronica, O’Connor, Robert D., Kaufman, Noy, Gao, Zhan-Guo, Auchampach, John A., Jacobson, Kenneth A.

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Structure-Activity Studies of 1 H -Imidazo[4,5- c ]quinolin-4-amine Derivatives as A 3 Adenosine Receptor Positive Allosteric Modulators von Fallot, Lucas B, Suresh, R Rama, Fisher, Courtney L, Salmaso, Veronica, O'Connor, Robert D, Kaufman, Noy, Gao, Zhan-Guo, Auchampach, John A, Jacobson, Kenneth A

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Activation of adenosine A 2A or A 2B receptors causes hypothermia in mice von Carlin, Jesse Lea, Jain, Shalini, Duroux, Romain, Suresh, R Rama, Xiao, Cuiying, Auchampach, John A, Jacobson, Kenneth A, Gavrilova, Oksana, Reitman, Marc L

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Molecularly Nonstoichiometric Crystals in Phosphorus Compounds von Chakravarty, Manab, Rama Suresh, R, Kumara Swamy, K. C

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2-Amino-5-arylethynyl-thiophen-3-yl-(phenyl)methanones as A 1 Adenosine Receptor Positive Allosteric Modulators von Oliva, Paola, Suresh, R Rama, Pasquini, Silvia, Salmaso, Veronica, Will, Edward J, Tosh, Dilip K, Gao, Zhan-Guo, Liu, Naili, Gavrilova, Oksana, Vincenzi, Fabrizio, Varani, Katia, Jacobson, Kenneth A

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Assay-Dependent Inverse Agonism at the A3 Adenosine Receptor: When Neutral Is Not Neutral von Pottie, Eline, Suresh, R. Rama, Jacobson, Kenneth A., Stove, Christophe P.

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Assay-Dependent Inverse Agonism at the A 3 Adenosine Receptor: When Neutral Is Not Neutral von Pottie, Eline, Suresh, R Rama, Jacobson, Kenneth A, Stove, Christophe P

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