The Lipid Kinase PIP5K1C Regulates Pain Signaling and Sensitization von Wright, Brittany D., Loo, Lipin, Street, Sarah E., Ma, Anqi, Taylor-Blake, Bonnie, Stashko, Michael A., Jin, Jian, Janzen, William P., Frye, Stephen V., Zylka, Mark J.

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The Synthesis and Initial Evaluation of MerTK Targeted PET Agents von Wang, Li, Zhou, Yubai, Wu, Xuedan, Ma, Xinrui, Li, Bing, Ding, Ransheng, Stashko, Michael A, Wu, Zhanhong, Wang, Xiaodong, Li, Zibo

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Pseudo-Cyclization through Intramolecular Hydrogen Bond Enables Discovery of Pyridine Substituted Pyrimidines as New Mer Kinase Inhibitors von Zhang, Weihe, Zhang, Dehui, Stashko, Michael A, DeRyckere, Deborah, Hunter, Debra, Kireev, Dmitri, Miley, Michael J, Cummings, Christopher, Lee, Minjung, Norris-Drouin, Jacqueline, Stewart, Wendy M, Sather, Susan, Zhou, Yingqiu, Kirkpatrick, Gregory, Machius, Mischa, Janzen, William P, Earp, H. Shelton, Graham, Douglas K, Frye, Stephen V, Wang, Xiaodong

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Discovery of Macrocyclic Pyrimidines as MerTK‐Specific Inhibitors von McIver, Andrew L., Zhang, Weihe, Liu, Qingyang, Jiang, Xinpeng, Stashko, Michael A., Nichols, James, Miley, Michael J., Norris‐Drouin, Jacqueline, Machius, Mischa, DeRyckere, Deborah, Wood, Edgar, Graham, Douglas K., Earp, H. Shelton, Kireev, Dmitri, Frye, Stephen V., Wang, Xiaodong

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Retraction: A High-Throughput Screening-Compatible Strategy for the Identification of Inositol Pyrophosphate Kinase Inhibitors von Baughman, Brandi M, Wang, Huanchen, An, Yi, Kireev, Dmitri, Stashko, Michael A, Jessen, Henning J, Pearce, Kenneth H, Frye, Stephen V, Shears, Stephen B

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Efficacy of a Mer and Flt3 tyrosine kinase small molecule inhibitor, UNC1666, in acute myeloid leukemia von Lee-Sherick, Alisa B, Zhang, Weihe, Menachof, Kelly K, Hill, Amanda A, Rinella, Sean, Kirkpatrick, Gregory, Page, Lauren S, Stashko, Michael A, Jordan, Craig T, Wei, Qi, Liu, Jing, Zhang, Dehui, DeRyckere, Deborah, Wang, Xiaodong, Frye, Stephen, Earp, H Shelton, Graham, Douglas K

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A High-Throughput Screening-Compatible Strategy for the Identification of Inositol Pyrophosphate Kinase Inhibitors von Baughman, Brandi M, Wang, Huanchen, An, Yi, Kireev, Dmitri, Stashko, Michael A, Jessen, Henning J, Pearce, Kenneth H, Frye, Stephen V, Shears, Stephen B

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Discovery of a Potent, Selective Protein Tyrosine Phosphatase 1B Inhibitor Using a Linked-Fragment Strategy von Szczepankiewicz, Bruce G, Liu, Gang, Hajduk, Philip J, Abad-Zapatero, Cele, Pei, Zhonghua, Xin, Zhili, Lubben, Thomas H, Trevillyan, James M, Stashko, Michael A, Ballaron, Stephen J, Liang, Heng, Huang, Flora, Hutchins, Charles W, Fesik, Stephen W, Jirousek, Michael R

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Development of Novel IP6K Inhibitors for the Treatment of Obesity and Obesity-Induced Metabolic Dysfunctions von Zhou, Yubai, Mukherjee, Sandip, Huang, Daowei, Chakraborty, Molee, Gu, Chunfang, Zong, Guangning, Stashko, Michael A., Pearce, Kenneth H., Shears, Stephen B., Chakraborty, Anutosh, Wang, Huanchen, Wang, Xiaodong

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Discovery of Novel Macrocyclic MERTK/AXL Dual Inhibitors von Kong, Deyu, Tian, Qiang, Chen, Zhilong, Zheng, Hongchao, Stashko, Michael A., Yan, Dan, Earp, H. Shelton, Frye, Stephen V., DeRyckere, Deborah, Kireev, Dmitri, Graham, Douglas K., Wang, Xiaodong

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UNC2025, a Potent and Orally Bioavailable MER/FLT3 Dual Inhibitor von Zhang, Weihe, DeRyckere, Deborah, Hunter, Debra, Liu, Jing, Stashko, Michael A, Minson, Katherine A, Cummings, Christopher T, Lee, Minjung, Glaros, Trevor G, Newton, Dianne L, Sather, Susan, Zhang, Dehui, Kireev, Dmitri, Janzen, William P, Earp, H. Shelton, Graham, Douglas K, Frye, Stephen V, Wang, Xiaodong

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Inhibition of Inositol Polyphosphate Kinases by Quercetin and Related Flavonoids: A Structure–Activity Analysis von Gu, Chunfang, Stashko, Michael A, Puhl-Rubio, Ana C, Chakraborty, Molee, Chakraborty, Anutosh, Frye, Stephen V, Pearce, Kenneth H, Wang, Xiaodong, Shears, Stephen B, Wang, Huanchen

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MerTK activity is not necessary for the proliferation of glioblastoma stem cells von Hoque, Monira, Wai Wong, Siu, Recasens, Ariadna, Abbassi, Ramzi, Nguyen, Nghi, Zhang, Dehui, Stashko, Michael A., Wang, Xiaodong, Frye, Stephen, Day, Bryan W., Baell, Jonathan, Munoz, Lenka

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Nonsteroidal Selective Glucocorticoid Modulators:  The Effect of C-10 Substitution on Receptor Selectivity and Functional Potency of 5-Allyl-2,5-dihydro-2,2,4-trimethyl-1H-[1]benzo... von Kym, Philip R, Kort, Michael E, Coghlan, Michael J, Moore, Jimmie L, Tang, Rui, Ratajczyk, James D, Larson, Daniel P, Elmore, Steven W, Pratt, John K, Stashko, Michael A, Falls, H. Douglass, Lin, Chun W, Nakane, Masake, Miller, Loan, Tyree, Curtis M, Miner, Jeffery N, Jacobson, Peer B, Wilcox, Denise M, Nguyen, Phong, Lane, Benjamin C

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Highly Selective MERTK Inhibitors Achieved by a Single Methyl Group von Zhao, Jichen, Zhang, Dehui, Zhang, Weihe, Stashko, Michael A, DeRyckere, Deborah, Vasileiadi, Eleana, Parker, Rebecca E, Hunter, Debra, Liu, Qingyang, Zhang, Yuewei, Norris-Drouin, Jacqueline, Li, Bing, Drewry, David H, Kireev, Dmitri, Graham, Douglas K, Earp, Henry Shelton, Frye, Stephen V, Wang, Xiaodong

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Identification of a cell-active chikungunya virus nsP2 protease inhibitor using a covalent fragment-based screening approach von Merten, Eric M, Sears, John D, Leisner, Tina M, Hardy, P Brian, Ghoshal, Anirban, Hossain, Mohammad Anwar, Asressu, Kesatebrhan Haile, Brown, Peter J, Tse, Edwin G, Stashko, Michael A, Li, Kelin, Norris-Drouin, Jacqueline L, Herring, Laura E, Mordant, Angie L, Webb, Thomas S, Mills, Christine A, Barker, Natalie K, Streblow, Zachary J, Perveen, Sumera, Arrowsmith, Cheryl H, Couñago, Rafael Miguez, Arnold, Jamie J, Cameron, Craig E, Streblow, Daniel N, Moorman, Nathaniel J, Heise, Mark T, Willson, Timothy M, Popov, Konstantin I, Pearce, Kenneth H

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Discovery, Structure−Activity Relationship, and Pharmacological Evaluation of (5-Substituted-pyrrolidinyl-2-carbonyl)-2-cyanopyrrolidines as Potent Dipeptidyl Peptidase IV Inhibito... von Pei, Zhonghua, Li, Xiaofeng, Longenecker, Kenton, von Geldern, Thomas W, Wiedeman, Paul E, Lubben, Thomas H, Zinker, Bradley A, Stewart, Kent, Ballaron, Stephen J, Stashko, Michael A, Mika, Amanda K, Beno, David W. A, Long, Michelle, Wells, Heidi, Kempf-Grote, Anita J, Madar, David J, McDermott, Todd S, Bhagavatula, Lakshmi, Fickes, Michael G, Pireh, Daisy, Solomon, Larry R, Lake, Marc R, Edalji, Rohinton, Fry, Elizabeth H, Sham, Hing L, Trevillyan, James M

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SETDB1 Triple Tudor Domain Ligand, (R,R)‑59, Promotes Methylation of Akt1 in Cells von Uguen, Mélanie, Deng, Yu, Li, Fengling, Shell, Devan J., Norris-Drouin, Jacqueline L., Stashko, Michael A., Ackloo, Suzanne, Arrowsmith, Cheryl H., James, Lindsey I., Liu, Pengda, Pearce, Kenneth H., Frye, Stephen V.

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UNC5293, a potent, orally available and highly MERTK-selective inhibitor von Zheng, Hongchao, Zhao, Jichen, Li, Bing, Zhang, Weihe, Stashko, Michael A., Minson, Katherine A., Huey, Madeline G., Zhou, Yubai, Earp, Henry Shelton, Kireev, Dmitri, Graham, Douglas K., DeRyckere, Deborah, Frye, Stephen V., Wang, Xiaodong

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Development of [18F]MIPS15692, a radiotracer with in vitro proof-of-concept for the imaging of MER tyrosine kinase (MERTK) in neuroinflammatory disease von Wong, Siu Wai, Vivash, Lucy, Mudududdla, Ramesh, Nguyen, Nghi, Hermans, Stefan J., Shackleford, David M., Field, Judith, Xue, Lian, Aprico, Andrea, Hancock, Nancy C., Haskali, Mohammad, Stashko, Michael A., Frye, Stephen V., Wang, Xiaodong, Binder, Michele D., Ackermann, Uwe, Parker, Michael W., Kilpatrick, Trevor J., Baell, Jonathan B.

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