Oxalyl Boronates Enable Modular Synthesis of Bioactive Imidazoles von Lee, C. Frank, Holownia, Aleksandra, Bennett, James M., Elkins, Jonathan M., St. Denis, Jeffrey D., Adachi, Shinya, Yudin, Andrei K.

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Synthesis of Aminoboronic Acid Derivatives from Amines and Amphoteric Boryl Carbonyl Compounds von Diaz, Diego B., Scully, Conor C. G., Liew, Sean K., Adachi, Shinya, Trinchera, Piera, St. Denis, Jeffrey D., Yudin, Andrei K.

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Fragment-based drug discovery: opportunities for organic synthesis von St. Denis, Jeffrey D, Hall, Richard J, Murray, Christopher W, Heightman, Tom D, Rees, David C

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Boron-Containing Enamine and Enamide Linchpins in the Synthesis of Nitrogen Heterocycles von St. Denis, Jeffrey D, Zajdlik, Adam, Tan, Joanne, Trinchera, Piera, Lee, C. Frank, He, Zhi, Adachi, Shinya, Yudin, Andrei K

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Boroalkyl Group Migration Provides a Versatile Entry into α-Aminoboronic Acid Derivatives von He, Zhi, Zajdlik, Adam, St. Denis, Jeffrey D, Assem, Naila, Yudin, Andrei K

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Oxidative Geminal Functionalization of Organoboron Compounds von He, Zhi, Trinchera, Piera, Adachi, Shinya, St. Denis, Jeffrey D., Yudin, Andrei K.

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Access to Cyclic Amino Boronates via Rhodium-Catalyzed Functionalization of Alkyl MIDA Boronates von St. Denis, Jeffrey D, Lee, C. Frank, Yudin, Andrei K

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X‑ray Screening of an Electrophilic Fragment Library and Application toward the Development of a Novel ERK 1/2 Covalent Inhibitor von St. Denis, Jeffrey D., Chessari, Gianni, Cleasby, Anne, Cons, Benjamin D., Cowan, Suzanna, Dalton, Samuel E., East, Charlotte, Murray, Christopher W., O’Reilly, Marc, Peakman, Torren, Rapti, Magdalini, Stow, Jessie L.

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Evaluation of a chiral cubane-based Schiff base ligand in asymmetric catalysis reactions von Biegasiewicz, Kyle F, Ingalsbe, Michelle L, St Denis, Jeffrey D, Gleason, James L, Ho, Junming, Coote, Michelle L, Savage, G Paul, Priefer, Ronny

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Chemoselective palladium-catalyzed α-allylation of α-boryl aldehydes von St Denis, Jeffrey D, He, Zhi, Yudin, Andrei K

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Fragment-Based Discovery of Allosteric Inhibitors of SH2 Domain-Containing Protein Tyrosine Phosphatase‑2 (SHP2) von Day, James E. H., Berdini, Valerio, Castro, Joan, Chessari, Gianni, Davies, Thomas G., Day, Philip J., St. Denis, Jeffrey D., Fujiwara, Hideto, Fukaya, Satoshi, Hamlett, Christopher C. F., Hearn, Keisha, Hiscock, Steven D., Holvey, Rhian S., Ito, Satoru, Kandola, Navrohit, Kodama, Yasuo, Liebeschuetz, John W., Martins, Vanessa, Matsuo, Kenichi, Mortenson, Paul N., Muench, Sandra, Nakatsuru, Yoko, Ochiiwa, Hiroaki, Palmer, Nicholas, Peakman, Torren, Price, Amanda, Reader, Michael, Rees, David C., Rich, Sharna J., Shah, Alpesh, Shibata, Yoshihiro, Smyth, Tomoko, Twigg, David G., Wallis, Nicola G., Williams, Glyn, Wilsher, Nicola E., Woodhead, Andrew, Shimamura, Tadashi, Johnson, Christopher N.

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Fragment-Based Discovery of a Series of Allosteric-Binding Site Modulators of β‑Glucocerebrosidase von Palmer, Nick, Agnew, Christopher, Benn, Caroline, Buffham, William J., Castro, Joan N., Chessari, Gianni, Clark, Mellissa, Cons, Benjamin D., Coyle, Joseph E., Dawson, Lee A., Hamlett, Christopher C. F., Hodson, Charlotte, Holding, Finn, Johnson, Christopher N., Liebeschuetz, John W., Mahajan, Pravin, McCarthy, James M., Murray, Christopher W., O’Reilly, Marc, Peakman, Torren, Price, Amanda, Rapti, Magdalini, Reeks, Judith, Schöpf, Patrick, St-Denis, Jeffrey D., Valenzano, Chiara, Wallis, Nicola G., Walser, Reto, Weir, Heather, Wilsher, Nicola E., Woodhead, Andrew, Bento, Carla F., Tisi, Dominic

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Oxalyl Boronates Enable Modular Synthesis of Bioactive Imidazoles von Lee, C. Frank, Holownia, Aleksandra, Bennett, James M., Elkins, Jonathan M., St. Denis, Jeffrey D., Adachi, Shinya, Yudin, Andrei K.

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Chemoselective palladium-catalyzed α-allylation of α-boryl aldehydesElectronic supplementary information (ESI) available: 1H, 13C, 11B, HRMS. See DOI: 10.1039/c2ob26503f von St. Denis, Jeffrey D, He, Zhi, Yudin, Andrei K

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Facile synthesis of borofragments and their evaluation in activity-based protein profilingElectronic supplementary information (ESI) available. CCDC 1021097-1021099. For ESI and cr... von Adachi, Shinya, Cognetta 3rd, Armand B, Niphakis, Micah J, He, Zhi, Zajdlik, Adam, St. Denis, Jeffrey D, Scully, Conor C. G, Cravatt, Benjamin F, Yudin, Andrei K

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ChemInform Abstract: Access to Cyclic Amino Boronates via Rhodium‐Catalyzed Functionalization of Alkyl MIDA Boronates von St. Denis, Jeffrey D., Lee, C. Frank, Yudin, Andrei K.

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Development of a novel expression, ZIMAX/Kzi for determination of the counter-anion effect on the antimicrobial activity of tetrabutylammonium salts von INGALSBE, Michelle L, DENIS, Jeffrey D. St, MCGAHAN, Megan E, STEINER, Walter W, PRIEFER, Ronny

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ChemInform Abstract: Condensation‐Driven Assembly of Boron‐Containing Bis(Heteroaryl) Motifs Using a Linchpin Approach von Adachi, Shinya, Liew, Sean K., Lee, C. Frank, Lough, Alan, He, Zhi, Denis, Jeffrey D. St, Poda, Gennady, Yudin, Andrei K.

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ChemInform Abstract: Boron-Containing Enamine and Enamide Linchpins in the Synthesis of Nitrogen Heterocycles von St. Denis, Jeffrey D., Zajdlik, Adam, Tan, Joanne, Trinchera, Piera, Lee, C. Frank, He, Zhi, Adachi, Shinya, Yudin, Andrei K.

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ChemInform Abstract: Stereocontrolled Synthesis of 1,2- and 1,3-Diamine Building Blocks from Aziridine Aldehyde Dimers von Liew, Sean K., He, Zhi, St. Denis, Jeffrey D., Yudin, Andrei K.

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