Nanomolar Inhibitors of Glycogen Phosphorylase Based on β‑d‑Glucosaminyl Heterocycles: A Combined Synthetic, Enzyme Kinetic, and Protein Crystallography Study von Bokor, Éva, Kyriakis, Efthimios, Solovou, Theodora G.A, Koppány, Csenge, Kantsadi, Anastassia L, Szabó, Katalin E, Szakács, Andrea, Stravodimos, George A, Docsa, Tibor, Skamnaki, Vassiliki T, Zographos, Spyros E, Gergely, Pál, Leonidas, Demetres D, Somsák, László

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Mutagenesis of a Lotus japonicus GSK3β/Shaggy-like kinase reveals functionally conserved regulatory residues von Solovou, Theodora G.A., Garagounis, Constantine, Kyriakis, Efthimios, Bobas, Charalambos, Papadopoulos, Georgios E., Skamnaki, Vassiliki T., Papadopoulou, Kalliope K., Leonidas, Demetres D.

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van der Waals interactions govern C-β-d-glucopyranosyl triazoles’ nM inhibitory potency in human liver glycogen phosphorylase von Kantsadi, Anastassia L., Stravodimos, George A., Kyriakis, Efthimios, Chatzileontiadou, Demetra S.M., Solovou, Theodora G.A., Kun, Sándor, Bokor, Éva, Somsák, László, Leonidas, Demetres D.

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Probing the β-pocket of the active site of human liver glycogen phosphorylase with 3-(C-β-d-glucopyranosyl)-5-(4-substituted-phenyl)-1, 2, 4-triazole inhibitors von Kyriakis, Efthimios, Solovou, Theodora G.A., Kun, Sándor, Czifrák, Katalin, Szőcs, Béla, Juhász, László, Bokor, Éva, Stravodimos, George A., Kantsadi, Anastassia L., Chatzileontiadou, Demetra S.M., Skamnaki, Vassiliki T., Somsák, László, Leonidas, Demetres D.

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Fig. 5 in Mutagenesis of a Lotus japonicus GSK3β/Shaggy-like kinase reveals functionally conserved regulatory residues von Solovou, Theodora G.A., Garagounis, Constantine, Kyriakis, Efthimios, Bobas, Charalambos, Papadopoulos, Georgios E., Skamnaki, Vassiliki T., Papadopoulou, Kalliope K., Leonidas, Demetres D.

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Fig. 7 in Mutagenesis of a Lotus japonicus GSK3β/Shaggy-like kinase reveals functionally conserved regulatory residues von Solovou, Theodora G.A., Garagounis, Constantine, Kyriakis, Efthimios, Bobas, Charalambos, Papadopoulos, Georgios E., Skamnaki, Vassiliki T., Papadopoulou, Kalliope K., Leonidas, Demetres D.

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Fig. 4 in Mutagenesis of a Lotus japonicus GSK3β/Shaggy-like kinase reveals functionally conserved regulatory residues von Solovou, Theodora G.A., Garagounis, Constantine, Kyriakis, Efthimios, Bobas, Charalambos, Papadopoulos, Georgios E., Skamnaki, Vassiliki T., Papadopoulou, Kalliope K., Leonidas, Demetres D.

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Fig. 3 in Mutagenesis of a Lotus japonicus GSK3β/Shaggy-like kinase reveals functionally conserved regulatory residues von Solovou, Theodora G.A., Garagounis, Constantine, Kyriakis, Efthimios, Bobas, Charalambos, Papadopoulos, Georgios E., Skamnaki, Vassiliki T., Papadopoulou, Kalliope K., Leonidas, Demetres D.

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