Drug repurposing and human parasitic protozoan diseases von Andrews, Katherine T., Fisher, Gillian, Skinner-Adams, Tina S.

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A Subset Screen of the Compounds Australia Scaffold Library Identifies 7-Acylaminodibenzoxazepinones as Potent and Selective Hits for Anti- Giardia Drug Discovery von Hart, Christopher J S, Riches, Andrew G, Tiash, Snigdha, Clapper, Erin, Ramu, Soumya, Zuegg, Johannes, Ryan, John H, Skinner-Adams, Tina S

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Effect of clinically approved HDAC inhibitors on Plasmodium, Leishmania and Schistosoma parasite growth von Chua, Ming Jang, Arnold, Megan S.J., Xu, Weijun, Lancelot, Julien, Lamotte, Suzanne, Späth, Gerald F., Prina, Eric, Pierce, Raymond J., Fairlie, David P., Skinner-Adams, Tina S., Andrews, Katherine T.

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Fingerprinting the substrate specificity of M1 and M17 aminopeptidases of human malaria, Plasmodium falciparum von Poreba, Marcin, McGowan, Sheena, Skinner-Adams, Tina S, Trenholme, Katharine R, Gardiner, Donald L, Whisstock, James C, To, Joyce, Salvesen, Guy S, Dalton, John P, Drag, Marcin

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Structural basis for the inhibition of the essential Plasmodium falciparum M1 neutral aminopeptidase von McGowan, Sheena, Porter, Corrine J, Lowther, Jonathan, Stack, Colin M, Golding, Sarah J, Skinner-Adams, Tina S, Trenholme, Katharine R, Teuscher, Franka, Donnelly, Sheila M, Grembecka, Jolanta, Mucha, Artur, Kafarski, Pawel, DeGori, Ross, Buckle, Ashley M, Gardiner, Donald L, Whisstock, James C, Dalton, John P

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Activity of bromodomain protein inhibitors/binders against asexual-stage Plasmodium falciparum parasites von Chua, Ming Jang, Robaa, Dina, Skinner-Adams, Tina S., Sippl, Wolfgang, Andrews, Katherine T.

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An ELISA method to assess HDAC inhibitor-induced alterations to P. falciparum histone lysine acetylation von Hesping, Eva, Skinner-Adams, Tina S., Fisher, Gillian M., Kurz, Thomas, Andrews, Katherine T.

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Thieno[3,2-b]pyrrole 5-carboxamides as potent and selective inhibitors of Giardia duodenalis von Hart, Christopher JS, Riches, Andrew G., Tiash, Snigdha, Abraham, Rebecca, Fayd’Herbe, Keely, Joch, Ellis, Zulfiqar, Bilal, Sykes, Melissa L., Avery, Vicky M., Šlapeta, Jan, Abraham, Sam, Ryan, John H., Skinner-Adams, Tina S.

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The Key Glycolytic Enzyme Phosphofructokinase Is Involved in Resistance to Antiplasmodial Glycosides von Fisher, Gillian M, Cobbold, Simon A, Jezewski, Andrew, Carpenter, Emma F, Arnold, Megan, Cowell, Annie N, Tjhin, Erick T, Saliba, Kevin J, Skinner-Adams, Tina S, Lee, Marcus C S, Odom John, Audrey, Winzeler, Elizabeth A, McConville, Malcolm J, Poulsen, Sally-Ann, Andrews, Katherine T

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Effect of Antimalarial Drugs on Plasmodium falciparum Gametocytes von Peatey, Christopher L., Skinner-Adams, Tina S., Dixon, Matthew W. A., McCarthy, James S., Gardiner, Donald L., Trenholme, Katharine R.

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The Aminopeptidase Inhibitor CHR-2863 Is an Orally Bioavailable Inhibitor of Murine Malaria von SKINNER-ADAMS, Tina S, PEATEY, Christopher L, DALTON, John P, GARDINER, Donald L, ANDERSON, Karen, TRENHOLME, Katharine R, KRIGE, David, BROWN, Christopher L, STACK, Colin, NSANGOU, Desire M. M, MATHEWS, Rency T, THIVIERGE, Karine

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Identification of Phosphinate Dipeptide Analog Inhibitors Directed against the Plasmodium falciparum M17 Leucine Aminopeptidase as Lead Antimalarial Compounds von Skinner-Adams, Tina S, Lowther, Jonathan, Teuscher, Franka, Stack, Colin M, Grembecka, Jolanta, Mucha, Artur, Kafarski, Pawel, Trenholme, Katharine R, Dalton, John P, Gardiner, Donald L

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An image-based Pathogen Box screen identifies new compounds with anti-Giardia activity and highlights the importance of assay choice in phenotypic drug discovery von Tiash, Snigdha, Saunders, Jake, Hart, Christopher J.S., Ryan, John H., Riches, Andrew G., Skinner-Adams, Tina S.

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Saquinavir Inhibits the Malaria Parasite's Chloroquine Resistance Transporter von Martin, Rowena E, Butterworth, Alice S, Gardiner, Donald L, Kirk, Kiaran, McCarthy, James S, Skinner-Adams, Tina S

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A novel in vitro image-based assay identifies new drug leads for giardiasis von Hart, Christopher J.S., Munro, Taylah, Andrews, Katherine T., Ryan, John H., Riches, Andrew G., Skinner-Adams, Tina S.

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Antimalarial Asexual Stage-Specific and Gametocytocidal Activities of HIV Protease Inhibitors von PEATEY, Christopher L, ANDREWS, Katherine T, EICKEL, Nina, MACDONALD, Timothy, BUTTERWORTH, Alice S, TRENHOLME, Katharine R, GARDINER, Donald L, MCCARTHY, James S, SKINNER-ADAMS, Tina S

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Synthesis and Antiplasmodial Evaluation of Analogues Based on the Tricyclic Core of Thiaplakortones A-D von Schwartz, Brett D, Coster, Mark J, Skinner-Adams, Tina S, Andrews, Katherine T, White, Jonathan M, Davis, Rohan A

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The frequency of malaria is similar among women receiving either lopinavir/ritonavir or nevirapine-based antiretroviral treatment von Skinner-Adams, Tina S, Butterworth, Alice S, Porter, Kimberly A, D'Amico, Ronald, Sawe, Fred, Shaffer, Doug, Siika, Abraham, Hosseinipour, Mina C, Stringer, Elizabeth, Currier, Judith S, Chipato, Tsungai, Salata, Robert, Lockman, Shahin, Eron, Joseph J, Meshnick, Steven R, McCarthy, James S

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The M18 Aspartyl Aminopeptidase of the Human Malaria Parasite Plasmodium falciparum von Teuscher, Franka, Lowther, Jonathan, Skinner-Adams, Tina S., Spielmann, Tobias, Dixon, Matthew W.A., Stack, Colin M., Donnelly, Sheila, Mucha, Artur, Kafarski, Paweł, Vassiliou, Stamatia, Gardiner, Donald L., Dalton, John P., Trenholme, Katharine R.

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Synthesis, Antimalarial Properties, and SAR Studies of Alkoxyurea-Based HDAC Inhibitors von Hansen, Finn K., Skinner-Adams, Tina S., Duffy, Sandra, Marek, Linda, Sumanadasa, Subathdrage D. M., Kuna, Krystina, Held, Jana, Avery, Vicky M., Andrews, Katherine T., Kurz, Thomas

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