MPP + -Induced Changes in Cellular Impedance as a Measure for Organic Cation Transporter (SLC22A1-3) Activity and Inhibition von Mocking, Tamara A M, Sijben, Hubert J, Vermeulen, Yimé W, IJzerman, Adriaan P, Heitman, Laura H

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A study of the dopamine transporter using the TRACT assay, a novel in vitro tool for solute carrier drug discovery von Sijben, Hubert J., van den Berg, Julie J. E., Broekhuis, Jeremy D., IJzerman, Adriaan P., Heitman, Laura H.

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Label-free high-throughput screening assay for the identification of norepinephrine transporter (NET/SLC6A2) inhibitors von Sijben, Hubert J., van Oostveen, Wieke M., Hartog, Peter B. R., Stucchi, Laura, Rossignoli, Andrea, Maresca, Giovanna, Scarabottolo, Lia, IJzerman, Adriaan P., Heitman, Laura H.

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Impedance-Based Phenotypic Readout of Transporter Function: A Case for Glutamate Transporters von Sijben, Hubert J, Dall' Acqua, Laura, Liu, Rongfang, Jarret, Abigail, Christodoulaki, Eirini, Onstein, Svenja, Wolf, Gernot, Verburgt, Simone J, Le Dévédec, Sylvia E, Wiedmer, Tabea, Superti-Furga, Giulio, IJzerman, Adriaan P, Heitman, Laura H

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Molecular insights into disease-associated glutamate transporter (EAAT1 / SLC1A3 ) variants using in silico and in vitro approaches von Gorostiola González, Marina, Sijben, Hubert J, Dall' Acqua, Laura, Liu, Rongfang, IJzerman, Adriaan P, Heitman, Laura H, van Westen, Gerard J P

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Targeting solute carriers to modulate receptor–ligand interactions von Sijben, Hubert J., Superti-Furga, Giulio, IJzerman, Adriaan P., Heitman, Laura H.

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An Overview of Cell-Based Assay Platforms for the Solute Carrier Family of Transporters von Dvorak, Vojtech, Wiedmer, Tabea, Ingles-Prieto, Alvaro, Altermatt, Patrick, Batoulis, Helena, Baerenz, Felix, Bender, Eckhard, Digles, Daniela, Durrenberger, Franz, Heitman, Laura H., IJzerman, Adriaan P., Kell, Douglas B., Kickinger, Stefanie, Koerzoe, Daniel, Leippe, Philipp, Licher, Thomas, Manolova, Vania, Rizzetto, Riccardo, Sassone, Francesca, Scarabottolo, Lia, Schlessinger, Avner, Schneider, Vanessa, Sijben, Hubert J., Steck, Anna-Lena, Sundstrom, Hanna, Tremolada, Sara, Wilhelm, Maria, Wright Muelas, Marina, Zindel, Diana, Steppan, Claire M., Superti-Furga, Giulio

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Still in Search for an EAAT Activator: GT949 Does Not Activate EAAT2, nor EAAT3 in Impedance and Radioligand Uptake Assays von van Veggel, Lieve, Mocking, Tamara A.M., Sijben, Hubert J., Liu, Rongfang, Gorostiola González, Marina, Dilweg, Majlen A., Royakkers, Jeroen, Li, Anna, Kumar, Vijay, Dong, Yin Yao, Bullock, Alex, Sauer, David B., Diliën, Hanne, van Westen, Gerard J.P., Schreiber, Rudy, Heitman, Laura H., Vanmierlo, Tim

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Advancing drug discovery through assay development: a survey of tool compounds within the human solute carrier superfamily von Digles, Daniela, Ingles-Prieto, Alvaro, Dvorak, Vojtech, Mocking, Tamara A M, Goldmann, Ulrich, Garofoli, Andrea, Homan, Evert J, Di Silvio, Alberto, Azzollini, Lucia, Sassone, Francesca, Fogazza, Mario, Bärenz, Felix, Pommereau, Antje, Zuschlag, Yasmin, Ooms, Jasper F, Tranberg-Jensen, Jeppe, Hansen, Jesper S, Stanka, Josefina, Sijben, Hubert J, Batoulis, Helena, Bender, Eckhard, Martini, Riccardo, IJzerman, Adriaan P, Sauer, David B, Heitman, Laura H, Manolova, Vania, Reinhardt, Juergen, Ehrmann, Alexander, Leippe, Philipp, Ecker, Gerhard F, Huber, Kilian V M, Licher, Thomas, Scarabottolo, Lia, Wiedmer, Tabea, Superti-Furga, Giulio

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Proteochemometric modeling identifies chemically diverse norepinephrine transporter inhibitors - Protocol Files von Bongers, Brandon, Sijben, Hubert J., Hartog, Peter, Tarnovskiy, Andrey, Heitman, Laura, IJzerman, Adriaan P., van Westen, Gerard

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Proteochemometric modeling identifies chemically diverse norepinephrine transporter inhibitors - Protocol Files von Bongers, Brandon, Sijben, Hubert J., Hartog, Peter, Tarnovskiy, Andrey, Heitman, Laura, IJzerman, Adriaan P., van Westen, Gerard

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Proteochemometric modeling identifies chemically diverse norepinephrine transporter inhibitors - Protocol Files von Bongers, Brandon, Sijben, Hubert J., Hartog, Peter, Tarnovskiy, Andrey, Heitman, Laura, IJzerman, Adriaan P., van Westen, Gerard

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