Sensing transport: label-free in vitro assays as an atTRACTive alternative for solute carrier transporter drug discovery von Sijben, H.J.

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Targeting solute carriers to modulate receptor-ligand interactions von Sijben, H.J., Superti-Furga, G., IJzerman, A.P., Heitman, L.H.

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MPP+-induced changes in cellular impedance as a measure for organic cation transporter (SLC22A1-3) activity and inhibition von Mocking, T.A.M., Sijben, H.J., Vermeulen, Y., IJzerman, A.P., Heitman, L.H.

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Proteochemometric modeling identifies chemically diverse norepinephrine transporter inhibitors von Bongers, B.J., Sijben, H.J., Hartog, P.B.R., Tarnovskiy, A., IJzerman, A.P., Heitman, L.H., Westen, G.J.P. van

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Molecular insights into disease-associated glutamate transporter (EAAT1 / SLC1A3) variants using in silico and in vitro approaches von Gorostiola Gonzalez, M., Sijben, H.J., Dall' Acqua, L., Liu, R., IJzerman, A.P., Heitman, L.H., Westen, G.J.P. van

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Still in search for an EAAT activator: GT949 does not activate EAAT2, nor EAAT3 in impedance and radioligand uptake assays von Veggel, L. van, Mocking, T.A.M., Sijben, H.J., Liu, R., Gorostiola González, M., Dilweg, M.A., Royakkers, J., Li, A., Kumar, V., Dong, Y.Y., Bullock, A., Sauer, D.B., Diliën, H., Westen, G.J.P. van, Schreiber, R., Heitman, L.H., Vanmierlo, T.

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A study of the dopamine transporter using the TRACT assay, a novel in vitro tool for solute carrier drug discovery von Sijben, H.J., Berg, J.E. van den, Broekhuis, J.D., IJzerman, A.P., Heitman, L.H.

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Label-free high-throughput screening assay for the identification of norepinephrine transporter (NET/SLC6A2) inhibitors von Sijben, H.J., Oostveen, W.M. van, Hartog, P.B.R., Stucchi, L., Rossignoli, A., Maresca, G., IJzerman, A.P., Heitman, L.H.

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A novel selective inverse agonist of the CB2 receptor as a radiolabeled tool compound for kinetic binding studies von Martella, A., Sijben, H.J., Rufer, A.C., Grether, U., Fingerle, J., Ullmer, C., Hartung, T., IJzerman, A.P., Stelt, M. van der, Heitman, L.H.

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Impedance-based phenotypic readout of transporter function: a case for glutamate transporters von Sijben, H.J., Dall’ Acqua, L., Liu, R., Jarret, A., Christodoulaki, E., Onstein, S., Wolf, G., Verburgt, S.J., Le Dévédec, S.E., Wiedmer, T., Superti-Furga, G., IJzerman, A.P., Heitman, L.H.

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An overview of cell-based assay platforms for the solute carrier family of transporters von Wiedmer, T., Ingles-Prieto, A., Altermatt, P., Batoulis, H, Bärenz, F., Bender, E., Digles, D., Dürrenberger, F., Heitman, L.H., IJzerman, A.P., Kell, D.B., Kickinger, S., Körzö, D., Leippe, P., Licher, T., Manolova, V., Rizzetto, R., Sassone, F., Scarabottolo, L., Schlessinger, A., Schneider, V., Sijben, H.J., Steck, A.L., Sundström, H., Tremolada, S., Wilhelm, M., Wright Muelas, M., Zindel, D., Steppan, C.M., Superti-Furga, G.

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The RESOLUTE consortium: unlocking SLC transporters for drug discovery von Superti-Furga, G., Lackner, D., Wiedmer, T., Ingles-Prieto, A., Barbosa, B., Girardi, E., Goldmann, U., Gürtl, B., Klavins, K., Klimek, C., Lindinger, S., Liñeiro-Retes, E., Müller, A.C., Onstein, S., Redinger, G., Sedlyarov, V., Wolf, G., Crawford, M., Everley, R., Hepworth, D., Liu, S., Noell, S., Piotrowski, M., Stanton, R., Zhang, H., Corallino, S., Faedo, A., Insidioso, M., Maresca, G., Redaelli, L., Sassone, F., Scarabottolo, L., Stucchi, M., Tarroni, P., Tremolada, S., Batoulis, H., Becker, A., Bender, E., Chang, Y.N., Ehrmann, A., Müller-Fahrnow, A., Zindel, D., Hamilton, B., Lenter, M., Santacruz, D., Viollet, C., Whitehurst, C., Johnsson, K., Leippe, P., Chang, L., Ibig, Y., Pfeifer, M., Reinhardt, J., Schönbett, J., Selzer, P., Seuwen, K., Bettembourg, C., Biton, B., Czech, J., de Foucauld, H., Didier, M., Licher, T., Mikol, V., Pommereau, A., Puech, F., Yaligara, V., Edwards, A., Bongers, B.J., Heitman, L.H., IJzerman, A.P., Sijben, H.J., Westen, G.J.P. van, Grixti, J., Kell, D.B., Mughal, F., Swainston, N., Wright-Muelas, M., Bohstedt, T., Burgess-Brown, N., Carpenter, L., Dürr, K., Hansen, J., Scacioc, A., Banci, G., Colas, C., Digles, D., Ecker, G., Füzi, B., Gamsjäger, V., Grandits, M., Martini, R., Troger, F., Altermatt, P., Doucerain, C., Dürrenberger, F., Manolova, V., Steck, A.L., Sundström, H., Wilhelm, M., Steppan, C.M.

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A Qualitative Study of the Feasibility and Acceptability of Implementing 'Sit-To-Stand' Desks in Vocational Education and Training von Kirschner, Mara, Golsteijn, Rianne H. J., Sijben, Sanne M., Singh, Amika S., Savelberg, Hans H. C. M., de Groot, Renate H. M.

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