Design, Synthesis and Biological Evaluation of N-phenylindole Derivatives as Pks13 Inhibitors againstMycobacterium tuberculosis von Cai, Yanpeng, Zhang, Wei, Lun, Shichun, Zhu, Tongtong, Xu, Weijun, Yang, Fan, Tang, Jie, Bishai, William R., Yu, Lifang

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Preliminary Structure–Activity Relationships and Biological Evaluation of Novel Antitubercular Indolecarboxamide Derivatives Against Drug-Susceptible and Drug-Resistant Mycobacteri... von Onajole, Oluseye K, Pieroni, Marco, Tipparaju, Suresh K, Lun, Shichun, Stec, Jozef, Chen, Gang, Gunosewoyo, Hendra, Guo, Haidan, Ammerman, Nicole C, Bishai, William R, Kozikowski, Alan P

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Risk of Tuberculosis Reactivation With Tofacitinib (CP-690550) von Maiga, Mamoudou, Lun, Shichun, Guo, Haidan, Winglee, Kathryn, Ammerman, Nicole C., Bishai, William R.

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Evaluation of gyrase B as a drug target in Mycobacterium tuberculosis von CHOPRA, Sidharth, MATSUYAMA, Karen, MADRID, Peter B, TRAN, Tran, MALERICH, Jeremiah P, BAOJIE WAN, FRANZBLAU, Scott G, SHICHUN LUN, HAIDAN GUO, MAIGA, Mariama C, BISHAI, William R

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Characterization of a Novel Cell Wall-anchored Protein with Carboxylesterase Activity Required for Virulence in Mycobacterium tuberculosis von Lun, Shichun, Bishai, William R.

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Adjunctive Integrated Stress Response Inhibition Accelerates Tuberculosis Clearance in Mice von Krug, Stefanie, Prasad, Pankaj, Xiao, Shiqi, Lun, Shichun, Ruiz-Bedoya, Camilo A, Klunk, Mariah, Ordonez, Alvaro A, Jain, Sanjay K, Srikrishna, Geetha, Kramnik, Igor, Bishai, William R

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Successful shortening of tuberculosis treatment using adjuvant host-directed therapy with FDA-approved phosphodiesterase inhibitors in the mouse model von Maiga, Mamoudou, Agarwal, Nisheeth, Ammerman, Nicole C, Gupta, Radhika, Guo, Haidan, Maiga, Marama C, Lun, Shichun, Bishai, William R

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MDA5 RNA-sensing pathway activation by Mycobacterium tuberculosis promotes innate immune subversion and pathogen survival von Bullen, C Korin, Singh, Alok K, Krug, Stefanie, Lun, Shichun, Thakur, Preeti, Srikrishna, Geetha, Bishai, William R

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Pharmacokinetic and In Vivo Efficacy Studies of the Mycobactin Biosynthesis Inhibitor Salicyl-AMS in Mice von Lun, Shichun, Guo, Haidan, Adamson, John, Cisar, Justin S, Davis, Tony D, Chavadi, Sivagami Sundaram, Warren, J David, Quadri, Luis E N, Tan, Derek S, Bishai, William R

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The two-domain LysX protein of Mycobacterium tuberculosis is required for production of lysinylated phosphatidylglycerol and resistance to cationic antimicrobial peptides von Maloney, Erin, Stankowska, Dorota, Zhang, Jian, Fol, Marek, Cheng, Qi-Jian, Lun, Shichun, Bishai, William R, Rajagopalan, Malini, Chatterjee, Delphi, Madiraju, Murty V

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Indoleamides are active against drug-resistant Mycobacterium tuberculosis von Lun, Shichun, Guo, Haidan, Onajole, Oluseye K., Pieroni, Marco, Gunosewoyo, Hendra, Chen, Gang, Tipparaju, Suresh K., Ammerman, Nicole C., Kozikowski, Alan P., Bishai, William R.

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Isoniazid resistance without a loss of fitness in Mycobacterium tuberculosis von Lee, Jong-Hee, Ammerman, Nicole C., Nolan, Scott, Geiman, Deborah E., Lun, Shichun, Guo, Haidan, Bishai, William R.

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Rv2190c, an NlpC/P60 family protein, is required for full virulence of Mycobacterium tuberculosis von Parthasarathy, Geetha, Lun, Shichun, Guo, Haidan, Ammerman, Nicole C, Geiman, Deborah E, Bishai, William R

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Extrapulmonary Dissemination of Mycobacterium bovis but Not Mycobacterium tuberculosis in a Bronchoscopic Rabbit Model of Cavitary Tuberculosis von Nedeltchev, Gueno G, Raghunand, Tirumalai R, Jassal, Mandeep S, Lun, Shichun, Cheng, Qi-Jian, Bishai, William R

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Synthetic lethality reveals mechanisms of Mycobacterium tuberculosis resistance to β-lactams von Lun, Shichun, Miranda, David, Kubler, Andre, Guo, Haidan, Maiga, Mariama C, Winglee, Kathryn, Pelly, Shaaretha, Bishai, William R

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Pyrido[1,2-a]benzimidazole-Based Agents Active Against Tuberculosis (TB), Multidrug-Resistant (MDR) TB and Extensively Drug-Resistant (XDR) TB von Pieroni, Marco, Tipparaju, Suresh K., Lun, Shichun, Song, Yang, Sturm, A. Willem, Bishai, William R., Kozikowski, Alan P.

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Targeting the chromosome partitioning protein ParA in tuberculosis drug discovery von Nisa, Shahista, Blokpoel, Marian C. J., Robertson, Brian D., Tyndall, Joel D. A., Lun, Shichun, Bishai, William R., O'Toole, Ronan

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Efficacy of Adjunctive Tofacitinib Therapy in Mouse Models of Tuberculosis von Maiga, Mamoudou, Ahidjo, Bintou Ahmadou, Maiga, Mariama C., Cheung, Laurene, Pelly, Shaaretha, Lun, Shichun, Bougoudogo, Flabou, Bishai, William R.

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Indole-2-carboxamide-based MmpL3 Inhibitors Show Exceptional Antitubercular Activity in an Animal Model of Tuberculosis Infection von Stec, Jozef, Onajole, Oluseye K, Lun, Shichun, Guo, Haidan, Merenbloom, Benjamin, Vistoli, Giulio, Bishai, William R, Kozikowski, Alan P

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