Functional characterization of agonists at recombinant human 5‐HT2A, 5‐HT2B and 5‐HT2C receptors in CHO‐K1 cells von Porter, R H P, Benwell, K R, Lamb, H, Malcolm, C S, Allen, N H, Revell, D F, Adams, D R, Sheardown, M J

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2,3-Dihydroxy-6-nitro-7-sulfamoyl-benzo(F)quinoxaline: A Neuroprotectant for Cerebral Ischemia von Sheardown, Malcolm J., Nielsen, Elsebet Ø., Hansen, Anker J., Jacobsen, Poul, Honoré, Tage

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Xanomeline, an M 1/M 4 preferring muscarinic cholinergic receptor agonist, produces antipsychotic-like activity in rats and mice von Shannon, Harlan E., Rasmussen, Kurt, Bymaster, Frank P., Hart, John C., Peters, Steven C., Swedberg, Michael D.B., Jeppesen, Lone, Sheardown, Malcolm J., Sauerberg, Per, Fink-Jensen, Anders

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AMPA, but not NMDA, receptor antagonism is neuroprotective in gerbil global ischaemia, even when delayed 24 h von Sheardown, Malcolm J., Suzdak, Peter D., Nordholm, Lars

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A potent antagonist of the strychnine insensitive glycine receptor has anticonvulsant properties von Sheardown, Malcolm J., Drejer, Jørgen, Helth Jensen, Leif, Stidsen, Carsten E., Honoré, Tage

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Muscarinic M 1 receptor agonists and M 2 receptor antagonists as therapeutic targets in Alzheimer’s disease von Sheardown, Malcolm J

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N-substituted adenosines as novel neuroprotective A(1) agonists with diminished hypotensive effects von Knutsen, L J, Lau, J, Petersen, H, Thomsen, C, Weis, J U, Shalmi, M, Judge, M E, Hansen, A J, Sheardown, M J

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The triggering of spreading depression in the chicken retina: a pharmacological study von Sheardown, Malcolm J.

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Novel functional M1 selective muscarinic agonists. Synthesis and structure-activity relationships of 3-(1,2,5-thiadiazolyl)-1,2,5,6-tetrahydro-1-methylpyridines von Sauerberg, Per, Olesen, Preben H, Nielsen, Susanne, Treppendahl, Svend, Sheardown, Malcolm J, Honore, Tage, Mitch, Charles H, Ward, John S, Pike, Andrew J

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The muscarinic receptor agonist BuTAC, a novel potential antipsychotic, does not impair learning and memory in mouse passive avoidance von Rasmussen, Thøger, Fink-Jensen, Anders, Sauerberg, Per, Swedberg, Michael D.B., Thomsen, Christian, Sheardown, Malcolm J., Jeppesen, Lone, Calligaro, David O., DeLapp, Neil W., Whitesitt, Celia, Ward, John S., Shannon, Harlan E., Bymaster, Frank P.

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Muscarinic receptor agonists decrease cocaine self-administration rates in drug-naive mice von Rasmussen, Thøger, Sauerberg, Per, Nielsen, Erik B, Swedberg, Michael D.B, Thomsen, Christian, Sheardown, Malcolm J, Jeppesen, Lone, Calligaro, David O, DeLapp, Neil W, Whitesitt, Celia, Ward, John S, Shannon, Harlan E, Bymaster, Frank P, Fink-Jensen, Anders

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Agonist-induced functional desensitization of recombinant human 5-HT2 receptors expressed in CHO-K1 cells von Porter, Richard H.P., Malcolm, Craig S., Allen, Nicola H., Lamb, Helen, Revell, Dean F., Sheardown, Malcolm J.

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Xanomeline compared to other muscarinic agents on stimulation of phosphoinositide hydrolysis in vivo and other cholinomimetic effects von Bymaster, Frank P., Carter, Petra A., Peters, Steven C., Zhang, Wei, Ward, John S., Mitch, Charles H., Calligaro, David O., Whitesitt, Celia A., DeLapp, Neil, Shannon, Harlan E., Rimvall, Karin, Jeppesen, Lone, Sheardown, Malcolm J., Fink-Jensen, Anders, Sauerberg, Per

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Unexpected antipsychotic-like activity with the muscarinic receptor ligand (5 R,6 R)6-(3-propylthio-1,2,5-thiadiazol-4-yl)-1-azabicyclo[3.2.1]octane von Bymaster, Frank P, Shannon, Harlan E, Rasmussen, Kurt, Delapp, Neil W, Mitch, Charles H, Ward, John S, Calligaro, David O, Ludvigsen, Thomas S, Sheardown, Malcolm J, Olesen, Preben H, Swedberg, Michael D.B, Sauerberg, Per, Fink-Jensen, Anders

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The triggering of spreading depression in the chick retina by nicotinic receptor agonists von Sheardown, Malcolm J

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Muscarinic Agonists with Antipsychotic-like Activity:  Structure−Activity Relationships of 1,2,5-Thiadiazole Analogues with Functional Dopamine Antagonist Activity von Sauerberg, Per, Jeppesen, Lone, Olesen, Preben H, Rasmussen, Thøger, Swedberg, Michael D. B, Sheardown, Malcolm J, Fink-Jensen, Anders, Thomsen, Christian, Thøgersen, Henning, Rimvall, Karin, Ward, John S, Calligaro, David O, DeLapp, Neil W, Bymaster, Frank P, Shannon, Harlan E

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Metabotropic glutamate receptor agonists reduce epileptiform activity in the rat cortex von Sheardown, Malcolm J

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Chlormethiazole inhibits epileptiform activity by potentiating GABA A receptor function von Empson, Ruth M., Gee, Veronica J., Sheardown, Malcolm J., Newberry, Nigel R.

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The pharmacology of AMPA receptors and their antagonists von Sheardown, M J

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Muscarinic agonists exhibit functional dopamine antagonism in unilaterally 6-OHDA lesioned rats von Fink-Jensen, Anders, Kristensen, Peter, Shannon, Harlan E, Calligaro, David O, Delapp, Neil W, Whitesitt, Cilia, Ward, John S, Thomsen, Christian, Rasmusseen, Thøger, Sheardown, Malcolm J, Jeppesen, Lone, Sauerberg, Per, Bymaster, Frank P

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