The cGAS–STING pathway as a therapeutic target in inflammatory diseases von Decout, Alexiane, Katz, Jason D., Venkatraman, Shankar, Ablasser, Andrea

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The Behavioral and Neurochemical Effects of a Novel d-Amino Acid Oxidase Inhibitor Compound 8 [4 H-Thieno [3,2-b]pyrrole-5-carboxylic Acid] and d-Serine von Smith, Sean M., Uslaner, Jason M., Yao, Lihang, Mullins, Chadwick M., Surles, Nathan O., Huszar, Sarah L., McNaughton, Caitlyn H., Pascarella, Danette M., Kandebo, Monika, Hinchliffe, Richard M., Sparey, Tim, Brandon, Nicholas J., Jones, Brian, Venkatraman, Shankar, Young, Mary Beth, Sachs, Nancy, Jacobson, Marlene A., Hutson, Peter H.

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The discovery of fused pyrrole carboxylic acids as novel, potent d-amino acid oxidase (DAO) inhibitors von Sparey, Tim, Abeywickrema, Pravien, Almond, Sarah, Brandon, Nick, Byrne, Noel, Campbell, Alister, Hutson, Pete H., Jacobson, Marlene, Jones, Brian, Munshi, Sanjeev, Pascarella, Danette, Pike, Andrew, Prasad, G. Sridhar, Sachs, Nancy, Sakatis, Melanie, Sardana, Vinod, Venkatraman, Shankar, Young, Mary Beth

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Structure-Based Design of β‑Site APP Cleaving Enzyme 1 (BACE1) Inhibitors for the Treatment of Alzheimer’s Disease von Yuan, Jing, Venkatraman, Shankar, Zheng, Yajun, McKeever, Brian M, Dillard, Lawrence W, Singh, Suresh B

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Process Development of the BACE Inhibitors BI 1147560 BS and BI 1181181 MZ von Li, Guisheng, Tan, Zhulin, Xu, Yibo, Sidhu, Kanwar P. S., Qu, Bo, Herbage, Melissa A., Eriksson, Magnus C., Zeng, Xingzhong, Busacca, Carl A., Desrosiers, Jean-Nicolas, Hampel, Thomas, Niemeier, Oliver, Reichel, Carsten, Quynh Dang, Mai Thi, Schoerer, Marvin, Kemmer, Dirk, Eick, Melanie, Werle, Holger, Kim, Soojin, Li, Zhibin, Venkatraman, Shankar, Jia, Lanqi, Claremon, David A., Fuchs, Klaus, Heine, Niklas, Byrne, Denis, Narayanan, Bikshandarkoil, Sarvestani, Max, Johnson, Joe, Premasiri, Ajith, Nummy, Larry J., Lorenz, Jon C., Haddad, Nizar, Gonnella, Nina C., Pennino, Scott, Krawiec, Mariusz, Senanayake, Chris H., Buono, Frederic, Lee, Heewon, Hossain, Azad, Song, Jinhua J., Reeves, Jonathan T.

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Potent and selective HIV-1 ribonuclease H inhibitors based on a 1-hydroxy-1,8-naphthyridin-2(1H)-one scaffold von Williams, Peter D., Staas, Donnette D., Venkatraman, Shankar, Loughran, H. Marie, Ruzek, Rowena D., Booth, Theresa M., Lyle, Terry A., Wai, John S., Vacca, Joseph P., Feuston, Bradley P., Ecto, Linda T., Flynn, Jessica A., DiStefano, Daniel J., Hazuda, Daria J., Bahnck, Carolyn M., Himmelberger, Amy L., Dornadula, Geetha, Hrin, Renee C., Stillmock, Kara A., Witmer, Marc V., Miller, Michael D., Grobler, Jay A.

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Design and Synthesis of Tri-Ring P 3 Benzamide-Containing Aminonitriles as Potent, Selective, Orally Effective Inhibitors of Cathepsin K von Palmer, James T., Bryant, Clifford, Wang, Dan-Xiong, Davis, Dana E., Setti, Eduardo L., Rydzewski, Robert M., Venkatraman, Shankar, Tian, Zong-Qiang, Burrill, Leland C., Mendonca, Rohan V., Springman, Eric, McCarter, John, Chung, Tobee, Cheung, Harry, Janc, James W., McGrath, Mary, Somoza, John R., Enriquez, Philip, Yu, Z. Walter, Strickley, Robert M., Liu, Liang, Venuti, Michael C., Percival, M. David, Falgueyret, Jean-Pierre, Prasit, Peppi, Oballa, Renata, Riendeau, Denis, Young, Robert N., Wesolowski, Gregg, Rodan, Sevgi B., Johnson, Colena, Kimmel, Donald B., Rodan, Gideon

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Pharmacological characterization of the new bace1 inhibitor bi 1181181 von Dorner-Ciossek, Cornelia, Hobson, Scott, Fuchs, Klaus, Sauer, Achim, Bauer, Margit, Morales-Ramos, Angel, Venkatraman, Shankar, Dillard, Lawrence W, Kruk, Barbara, Howard, Lamont, Bukhtiyarov, Yuri, Zhao, Yi, Lala, Deepak S

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P1‐314: Pharmacological characterization of the new bace1 inhibitor bi 1181181 von Dorner-Ciossek, Cornelia, Hobson, Scott, Fuchs, Klaus, Sauer, Achim, Bauer, Margit, Morales-Ramos, Angel, Venkatraman, Shankar, Dillard, Lawrence W., Kruk, Barbara, Howard, Lamont, Bukhtiyarov, Yuri, Zhao, Yi, Lala, Deepak S.

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A Novel Class of Nonpeptidic Biaryl Inhibitors of Human Cathepsin K von Robichaud, Joël, Oballa, Renata, Prasit, Peppi, Falgueyret, Jean-Pierre, Percival, M. David, Wesolowski, Gregg, Rodan, Sevgi B, Kimmel, Donald, Johnson, Colena, Bryant, Cliff, Venkatraman, Shankar, Setti, Eduardo, Mendonca, Rohan, Palmer, James T

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Peptidyl Diazomethyl Ketones Inhibit the Human Rhinovirus 3C Protease: Effect on Virus Yield by Partial Block of P3 Polyprotein Processing von Murray, Michael A, Janc, James W, Venkatraman, Shankar, Babé, Lilia M

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An activity-based probe for the determination of cysteine cathepsin protease activities in whole cells von Falgueyret, Jean-Pierre, Black, W. Cameron, Cromlish, Wanda, Desmarais, Sylvie, Lamontagne, Sonia, Mellon, Christophe, Riendeau, Denis, Rodan, Sevgi, Tawa, Paul, Wesolowski, Gregg, Bass, Kathryn E., Venkatraman, Shankar, Percival, M. David

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Identification and synthesis of [1,2,4]triazolo[3,4-a]phthalazine derivatives as high-affinity ligands to the α2δ-1 subunit of voltage gated calcium channel von LEBSACK, Alec D, GUNZNER, Janet, VENKATRAMAN, Shankar, BOWEI WANG, PRACITTO, Richard, SCHAFFHAUSER, Hervé, SANTINI, Angelina, AIYAR, Jayashree, BEZVERKOV, Robert, MUNOZ, Benito, WENSHENG LIU

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Synthesis of Oxadiazolidinedione Derivatives as Quisqualic Acid Analogs and Their Evaluation at a Quisqualate-Sensitized Site in the Rat Hippocampus von Venkatraman, Shankar, Roon, Robert J., Schulte, Marvin K., Koerner, James F., Johnson, Rodney L.

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Discovery of N-{ N-[(3-cyanobenzene) sulfonyl]-4( R)-(3,3-difluoropiperidin-1-yl)-( l)-prolyl}-4-[(3′,5′-dichloro-isonicotinoyl) amino]-( l)-phenylalanine (MK-0617), a highly poten... von Venkatraman, Shankar, Lebsack, Alec D., Alves, Kenneth, Gardner, Michael F., James, Joyce, Lingham, Russell B., Maniar, Salony, Mumford, Richard A., Si, Qian, Stock, Nicholas, Treonze, Kelly M., Wang, Bowei, Zunic, Jasmine, Munoz, Benito

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Compounds and compositions for treating conditions associated with STING activity von Venkatraman, Shankar, Seidel, Hans Martin, Katz, Jason, Roush, William R

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COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH STING ACTIVITY von KATZ, Jason, VENKATRAMAN, Shankar, SEIDEL, Hans Martin, ROUSH, William R

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COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH STING ACTIVITY von KATZ, Jason, VENKATRAMAN, Shankar, SEIDEL, Hans Martin, ROUSH, William R

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COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH STING ACTIVITY von Venkatraman, Shankar, Katz, Jason, Roush, William R

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Data for: 3487540 von Fish, Alexander

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