Greening the synthesis of peptide therapeutics: an industrial perspective von Martin, Vincent, Egelund, Peter H. G, Johansson, Henrik, Thordal Le Quement, Sebastian, Wojcik, Felix, Sejer Pedersen, Daniel

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Side Chain Cyclized Aromatic Amino Acids: Great Tools as Local Constraints in Peptide and Peptidomimetic Design von Van der Poorten, Olivier, Knuhtsen, Astrid, Sejer Pedersen, Daniel, Ballet, Steven, Tourwé, Dirk

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1,2,3-Triazoles in Peptidomimetic Chemistry von Pedersen, Daniel Sejer, Abell, Andrew

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Exploring endoperoxides as a new entry for the synthesis of branched azasugars von Domeyer, Svenja, Bjerregaard, Mark, Johansson, Henrik, Sejer Pedersen, Daniel

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Rational Design of Nanobody80 Loop Peptidomimetics: Towards Biased β2 Adrenergic Receptor Ligands von Martin, Charlotte, Moors, Samuel L. C., Danielsen, Mia, Betti, Cecilia, Fabris, Cecilia, Sejer Pedersen, Daniel, Pardon, Els, Peyressatre, Marion, Fehér, Krisztina, Martins, José C., Mosolff Mathiesen, Jesper, Morris, May C., Devoogdt, Nick, Caveliers, Vicky, De Proft, Frank, Steyaert, Jan, Ballet, Steven

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Bitopic Ligands and Metastable Binding Sites: Opportunities for G Protein-Coupled Receptor (GPCR) Medicinal Chemistry von Fronik, Philipp, Gaiser, Birgit I, Sejer Pedersen, Daniel

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Azide- and Alkyne-Derivatised α-Amino Acids von Johansson, Henrik, Pedersen, Daniel Sejer

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Dihydroxylation of 4-Substituted 1,2-Dioxines: A Concise Route to Branched Erythro Sugars von Robinson, Tony V, Pedersen, Daniel Sejer, Taylor, Dennis K, Tiekink, Edward R. T

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A Scalable Method for Regioselective 3‑Acylation of 2‑Substituted Indoles under Basic Conditions von Johansson, Henrik, Urruticoechea, Andoni, Larsen, Inna, Sejer Pedersen, Daniel

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Green Solid-Phase Peptide Synthesis: Oxyma-Triggered Spectrophotometric Monitoring of Residual Piperidine von Broman, So̷ren Lindbæk, Rosenberg, Martin, Wojcik, Felix, Holm Hansen, Anders, Egelund, Peter Hammer Guldager, Malmstro̷m, Joan, Sejer Pedersen, Daniel

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Process Mass Intensity (PMI): A Holistic Analysis of Current Peptide Manufacturing Processes Informs Sustainability in Peptide Synthesis von Kekessie, Ivy, Wegner, Katarzyna, Martinez, Isamir, Kopach, Michael E., White, Timothy D., Tom, Janine K., Kenworthy, Martin N., Gallou, Fabrice, Lopez, John, Koenig, Stefan G., Payne, Philippa R., Eissler, Stefan, Arumugam, Balasubramanian, Li, Changfeng, Mukherjee, Subha, Isidro-Llobet, Albert, Ludemann-Hombourger, Olivier, Richardson, Paul, Kittelmann, Jörg, Sejer Pedersen, Daniel, van den Bos, Leendert J.

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Bitopic Ligands Support the Presence of a Metastable Binding Site at the β2 Adrenergic Receptor von Gaiser, Birgit Isabel, Danielsen, Mia, Xu, Xinyu, Røpke Jørgensen, Kira, Fronik, Philipp, Märcher-Rørsted, Emil, Wróbel, Tomasz M., Liu, Xiangyu, Mosolff Mathiesen, Jesper, Sejer Pedersen, Daniel

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Fmoc-Removal with Pyrrolidine Expands the Available Solvent Space in Green Solid-Phase Peptide Synthesis von Egelund, Peter H. G, Jadhav, Sandip, Martin, Vincent, Johansson Castro, Henrik, Richner, Franziska, Le Quement, Sebastian Thordal, Dettner, Frank, Lechner, Carolin, Schoenleber, Ralph, Sejer Pedersen, Daniel

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Synthesis and stability study of a new major metabolite of γ-hydroxybutyric acid von Nymann Petersen, Ida, Langgaard Kristensen, Jesper, Tortzen, Christian, Breindahl, Torben, Sejer Pedersen, Daniel

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Identification of a new psychoactive substance in seized material: the synthetic opioid N‐phenyl‐N‐[1‐(2‐phenethyl)piperidin‐4‐yl]prop‐2‐enamide (Acrylfentanyl) von Breindahl, Torben, Kimergård, Andreas, Andreasen, Mette Findal, Pedersen, Daniel Sejer

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Synthesis of the calcilytic ligand NPS 2143 von Johansson, Henrik, Cailly, Thomas, Rojas Bie Thomsen, Alex, Bräuner-Osborne, Hans, Sejer Pedersen, Daniel

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Selective Allosteric Antagonists for the G Protein-Coupled Receptor GPRC6A Based on the 2‑Phenylindole Privileged Structure Scaffold von Johansson, Henrik, Boesgaard, Michael Worch, Nørskov-Lauritsen, Lenea, Larsen, Inna, Kuhne, Sebastiaan, Gloriam, David E, Bräuner-Osborne, Hans, Sejer Pedersen, Daniel

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Revisiting Bromohexitols as a Novel Class of Microenvironment‐Activated Prodrugs for Cancer Therapy von Johansson, Henrik, Hussain, Omar, Allison, Simon J., Robinson, Tony V., Phillips, Roger M., Sejer Pedersen, Daniel

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Rational Design of Nanobody80 Loop Peptidomimetics: Towards Biased β 2 Adrenergic Receptor Ligands von Martin, Charlotte, Moors, Samuel L C, Danielsen, Mia, Betti, Cecilia, Fabris, Cecilia, Sejer Pedersen, Daniel, Pardon, Els, Peyressatre, Marion, Fehér, Krisztina, Martins, José C, Mosolff Mathiesen, Jesper, Morris, May C, Devoogdt, Nick, Caveliers, Vicky, De Proft, Frank, Steyaert, Jan, Ballet, Steven

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Amino Triazolo Diazepines (Ata) as Constrained Histidine Mimics von Buysse, Koen, Farard, Julien, Nikolaou, Alexandros, Vanderheyden, Patrick, Vauquelin, Georges, Sejer Pedersen, Daniel, Tourwé, Dirk, Ballet, Steven

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