Quinazolinone Derivatives as Orally Available Ghrelin Receptor Antagonists for the Treatment of Diabetes and Obesity von Rudolph, Joachim, Esler, William P, O'Connor, Stephen, Coish, Philip D. G, Wickens, Philip L, Brands, Michael, Bierer, Donald E, Bloomquist, Brian T, Bondar, Georgiy, Chen, Libing, Chuang, Chih-Yuan, Claus, Thomas H, Fathi, Zahra, Fu, Wenlang, Khire, Uday R, Kristie, James A, Liu, Xiao-Gao, Lowe, Derek B, McClure, Andrea C, Michels, Martin, Ortiz, Astrid A, Ramsden, Philip D, Schoenleber, Robert W, Shelekhin, Tatiana E, Vakalopoulos, Alexandros, Tang, Weifeng, Wang, Lei, Yi, Lin, Gardell, Stephen J, Livingston, James N, Sweet, Laurel J, Bullock, William H

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Indanylacetic Acid Derivatives Carrying 4-Thiazolyl-phenoxy Tail Groups, a New Class of Potent PPAR α/γ/δ Pan Agonists:  Synthesis, Structure−Activity Relationship, and In Vivo Eff... von Rudolph, Joachim, Chen, Libing, Majumdar, Dyuti, Bullock, William H, Burns, Michael, Claus, Thomas, Dela Cruz, Fernando E, Daly, Michelle, Ehrgott, Frederick J, Johnson, Jeffrey S, Livingston, James N, Schoenleber, Robert W, Shapiro, Jeffrey, Yang, Ling, Tsutsumi, Manami, Ma, Xin

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PDE-10A inhibitors as insulin secretagogues von Cantin, Louis-David, Magnuson, Steven, Gunn, David, Barucci, Nicole, Breuhaus, Marina, Bullock, William H., Burke, Jennifer, Claus, Thomas H., Daly, Michelle, DeCarr, Lynn, Gore-Willse, Ann, Hoover-Litty, Helana, Kumarasinghe, Ellalahewage S., Li, Yaxin, Liang, Sidney X., Livingston, James N., Lowinger, Timothy, MacDougall, Margit, Ogutu, Herbert O., Olague, Alan, Ott-Morgan, Ronda, Schoenleber, Robert W., Tersteegen, Adrian, Wickens, Philip, Zhang, Zhonghua, Zhu, Jian, Zhu, Lei, Sweet, Laurel J.

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Indanylacetic acids as PPAR-δ activator insulin sensitizers von Wickens, Philip, Zhang, Chengzhi, Ma, Xin, Zhao, Qian, Amatruda, John, Bullock, William, Burns, Michael, Cantin, Louis-David, Chuang, Chih-Yuan, Claus, Thomas, Dai, Miao, Dela Cruz, Fernando, Dickson, David, Ehrgott, Frederick J., Fan, Dongping, Heald, Sarah, Hentemann, Martin, Iwuagwu, Christiana I., Johnson, Jeffrey S., Kumarasinghe, Ellalahewage, Ladner, David, Lavoie, Rico, Liang, Sidney, Livingston, James N., Lowe, Derek, Magnuson, Steve, Mannelly, Gretchen, Mugge, Ingo, Ogutu, Herbert, Pleasic-Williams, Susan, Schoenleber, Robert W., Shapiro, Jeff, Shelekhin, Tatiana, Sweet, Laurel, Town, Christopher, Tsutsumi, Manami

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Indanylacetic acid derivatives carrying aryl-pyridyl and aryl-pyrimidinyl tail groups—new classes of PPAR γ/δ and PPAR α/γ/δ agonists von Cantin, Louis-David, Liang, Sidney, Ogutu, Herbert, Iwuagwu, Christiana I., Boakye, Ken, Bullock, William H., Burns, Michael, Clark, Roger, Claus, Thomas, delaCruz, Fernando E., Daly, Michelle, Ehrgott, Frederick J., Johnson, Jeffrey S., Keiper, Christine, Livingston, James N., Schoenleber, Robert W., Shapiro, Jeffrey, Town, Christopher, Yang, Ling, Tsutsumi, Manami, Ma, Xin

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Novel Inhibitors of Cytokine-induced IκBα Phosphorylation and Endothelial Cell Adhesion Molecule Expression Show Anti-inflammatory Effects in Vivo von Pierce, Jacqueline W., Schoenleber, Robert, Jesmok, Gary, Best, Jennifer, Moore, Sarah A., Collins, Tucker, Gerritsen, Mary E.

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Synthesis and dopaminergic activity of 3-substituted 1-(aminomethyl)-3,4-dihydro-5,6-dihydroxy-1H-2-benzopyrans: characterization of an auxiliary binding region in the D1 receptor von DeNinno, Michael P, Schoenleber, Robert, Perner, Richard J, Lijewski, Linda, Asin, Karen E, Britton, Donald R, MacKenzie, Robert, Kebabian, John W

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A novel estrogen receptor ligand template von Sibley, Robert, Hatoum-Mokdad, Holia, Schoenleber, Robert, Musza, Laszlo, Stirtan, William, Marrero, Diana, Carley, William, Xiao, Hong, Dumas, Jacques

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1-Phenyl-5-pyrazolyl ureas: potent and selective p38 kinase inhibitors von Dumas, Jacques, Hatoum-Mokdad, Holia, Sibley, Robert, Riedl, Bernd, Scott, William J, Monahan, Mary Katherine, Lowinger, Timothy B, Brennan, Catherine, Natero, Reina, Turner, Tiffany, Johnson, Jeffrey S, Schoenleber, Robert, Bhargava, Ajay, Wilhelm, Scott M, Housley, Timothy J, Ranges, Gerald E, Shrikhande, Alka

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Discovery of a new class of p38 kinase inhibitors von Dumas, Jacques, Sibley, Robert, Riedl, Bernd, Monahan, Mary Katherine, Lee, Wendy, Lowinger, Timothy B, Redman, Anikó M, Johnson, Jeffrey S, Kingery-Wood, Jill, Scott, William J, Smith, Roger A, Bobko, Mark, Schoenleber, Robert, Ranges, Gerald E, Housley, Timothy J, Bhargava, Ajay, Wilhelm, Scott M, Shrikhande, Alka

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Relative stereochemistry of the A ring of plant bile pigments von Schoenleber, Robert W, Kim, Youseung, Rapoport, Henry

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Process for preparation of pegylated adrenomedullin, its intermediates and uses thereof von SCHOENLEBER ROBERT O, STELLMEIER ANDREAS

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SAR of a novel ‘Anthranilamide Like’ series of VEGFR-2, multi protein kinase inhibitors for the treatment of cancer von Wickens, Philip, Kluender, Harold, Dixon, Julie, Brennan, Catherine, Achebe, Furahi, Bacchiocchi, Antonella, Bankston, Don, Bierer, Donald, Brands, Michael, Braun, Debbie, Brown, Melissa S., Chuang, Chih-Yuan, Dumas, Jacques, Enyedy, Istvan, Hofilena, Gloria, Hong, Zhenqiu, Housley, Tim, Jones, Benjamin, Khire, Uday, Kreiman, Charles, Kumarasinghe, Ellalahewage, Lowinger, Timothy, Ott-Morgan, Ronda, Perkins, Louise, Phillips, Barton, Schoenleber, Robert, Scott, William J., Sheeler, Ryan, Redman, Anikó, Sun, Xiuying, Taylor, Ian, Wang, Lei, Wilhelm, Scott, Zhang, Xiaomei, Zhang, Mingbao, Sullivan, Elizabeth, Carter, Christopher, Miglarese, Mark, Levy, Joan

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A-77636 - A POTENT AND SELECTIVE DOPAMINE-D1 RECEPTOR AGONIST WITH ANTIPARKINSONIAN ACTIVITY IN MARMOSETS von KEBABIAN, JW, BRITTON, DR, DENINNO, MP, PERNER, R, SMITH, L, JENNER, P, SCHOENLEBER, R, WILLIAMS, M

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Synthesis and pharmacological characterization of a potent, orally active p38 kinase inhibitor von Dumas, Jacques, Hatoum-Mokdad, Holia, Sibley, Robert N, Smith, Roger A, Scott, William J, Khire, Uday, Lee, Wendy, Wood, Jill, Wolanin, Donald, Cooley, Jeffrey, Bankston, Donald, Redman, Aniko M, Schoenleber, Robert, Caringal, Yolanda, Gunn, David, Romero, Romulo, Osterhout, Martin, Paulsen, Holger, Housley, Timothy J, Wilhelm, Scott M, Pirro, John, Chien, Du-Shieng, Ranges, Gerald E, Shrikhande, Alka, Muzsi, Andrew, Bortolon, Elizabeth, Wakefield, Jean, Gianpaolo Ostravage, Cynthia, Bhargava, Ajay, Chau, Thuy

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Chromopeptides from phycoerythrins. Structure and linkage of a phycoerythrobilin tryptic tripeptide derived from a B-phycoerythrin von Schoenleber, Robert W, Leung, See Lap, Lundell, Daniel J, Glazer, Alexander N, Rapoport, Henry

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A68930: a potent agonist selective for the dopamine D1 receptor von DeNinno, M P, Schoenleber, R, MacKenzie, R, Britton, D R, Asin, K E, Briggs, C, Trugman, J M, Ackerman, M, Artman, L, Bednarz, L

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Novel Inhibitors of Cytokine-induced IκBα Phosphorylation and Endothelial Cell Adhesion Molecule Expression Show Anti-inflammatory Effects in Vivo von Jacqueline W. Pierce, Robert Schoenleber, Gary Jesmok, Jennifer Best, Sarah A. Moore, Tucker Collins, Mary E. Gerritsen

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(1R,3S)-1-(Aminomethyl)-3,4-dihydro-5,6-dihydroxy-3-phenyl-1H-2-benzopyran: a potent and selective D1 agonist von DeNinno, Michael P, Schoenleber, Robert, Asin, Karen E, MacKenzie, Robert, Kebabian, John W

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Synthesis and pharmacological evaluation of 1-(aminomethyl)-3,4-dihydro-5-hydroxy-1H-2-benzopyrans as dopamine D1 selective ligands von Michaelides, Michael R, Schoenleber, Robert, Thomas, Sheela, Yamamoto, Diane M, Britton, Donald R, MacKenzie, Robert, Kebabian, John W

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