Novel lead structures for antimalarial farnesyltransferase inhibitors von Kettler, K., Sakowski, J., Wiesner, J., Ortmann, R., Jomaa, H., Schlitzer, M.

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Synthesis of potential aldose reductase inhibitors based on minimal pharmacophore requirements von Schlitzer, Martin, Rodriguez, Labaniel, Kador, Peter F.

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2-(Aminoacylamino)benzophenones: farnesyltransferase inhibition and antimalarial activity von Kettler, K., Wiesner, J., Fucik, K., Sakowski, J., Ortmann, R., Dahse, H.-M., Jomaa, H., Schlitzer, M.

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Structure-activity relationships of novel anti-malarial agents part 8. Effect of different central aryls in biarylacryloylaminobenzophenones on antimalarial activity von Wiesner, J., Mitsch, A., Altenkämper, M., Ortmann, R., Jomaa, H., Schlitzer, M.

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Acyloxyalkyl ester prodrugs of FR900098 with improved in vivo anti-malarial activity von Ortmann, Regina, Wiesner, Jochen, Reichenberg, Armin, Henschker, Dajana, Beck, Ewald, Jomaa, Hassan, Schlitzer, Martin

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Inhibitors of farnesyltransferase: 5-arylacryloyl-aminobenzophenones show antimalarial activity von Wiesner, J., Wiesner, J., Ortmann, R., Mitsch, A., Wißner, P., Sattler, I., Jomaa, H., Schlitzer, M.

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Structure-activity relationships of novel anti-malarial agents : 1. arylacyl and cyclohexylacyl derivatives of 5-amino-2-tolylacetylaminobenzophenone von WIESNER, J, MITSCH, A, WISSNER, P, JOMAA, H, SCHLITZER, M

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Structure-activity relationships of novel anti-malarial agents. Part 2: Cinnamic acid derivatives von WIESNER, Jochen, MITSCH, Andreas, WISSNER, Pia, JOMAA, Hassan, SCHLITZER, Martin

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Structure activity relationship of antiproliferative N-acyl-aspartic acid dimethyl ester. 2. Variation of the aspartyl moiety von WISSNER, P, DAHSE, H.-M, SCHLITZER, M

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Non-thiol farnesyltransferase inhibitors: structure–activity relationships of benzophenone-based bisubstrate analogue farnesyltransferase inhibitors von Schlitzer, Martin, Böhm, Markus, Sattler, Isabel

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Non-thiol farnesyltransferase inhibitors: N-(4-tolylacetylamino-3-benzoylphenyl)-3-arylfurylacrylic acid amides von Mitsch, Andreas, Wißner, Pia, Silber, Katrin, Haebel, Peter, Sattler, Isabel, Klebe, Gerhard, Schlitzer, Martin

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Structure–Activity relationships of novel anti-Malarial agents: Part 5. N-(4-acylamino-3-benzoylphenyl)-[5-(4-nitrophenyl)-2-furyl]acrylic acid amides von Wiesner, Jochen, Kettler, Katja, Sakowski, Jacek, Ortmann, Regina, Jomaa, Hassan, Schlitzer, Martin

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Non-thiol farnesyltransferase inhibitors: the concept of benzophenone-based bisubstrate analogue farnesyltransferase inhibitors von Schlitzer, Martin, Sattler, Isabel

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Non-thiol farnesyltransferase inhibitors: N-(4-acylamino-3-benzoylphenyl)-3-[5-(4-nitrophenyl)-2-furyl]acrylic acid amides von KETTLER, Katja, SAKOWSKI, Jacek, SILBER, Katrin, SATTLER, Isabel, KLEBE, Gerhard, SCHLITZER, Martin

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Non-peptidic, non-prenylic inhibitors of the prenyl protein-specific protease Rce1 von Schlitzer, M, Winter-Vann, A, Casey, P J

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Non-thiol farnesyltransferase inhibitors: Utilization of an aryl binding site by 5-arylacryloylaminobenzophenones von MITSCH, Andreas, BÖHM, Markus, WISSNER, Pia, SATTLER, Isabel, SCHLITZER, Martin

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Non-Thiol Farnesyltransferase Inhibitors: Utilization of the Near Aryl Binding Site by 5-Arylacetylaminobenzophenones von Mitsch, Andreas, Böhm, Markus, Sattler, Isabel, Schlitzer, Martin

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Design, synthesis and early structure-activity relationship of farnesyltransferase inhibitors which mimic both the peptidic and the prenylic substrate von SCHLITZER, M, BÖHM, M, SATTLER, I, DAHSE, H.-M

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Non-thiol Farnesyltransferase Inhibitors: Utilization of the Far Aryl Binding Site by 5-Cinnamoylaminobenzophenones von Mitsch, Andreas, Wißner, Pia, Böhm, Markus, Silber, Katrin, Klebe, Gerhard, Sattler, Isabel, Schlitzer, Martin

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Non-Thiol Farnesyltransferase Inhibitors: Evaluation of Different AA(X)-Peptidomimetic Substructures in Combination with Arylic Cysteine Replacements von Sakowski, Jacek, Böhm, Markus, Sattler, Isabel, Schlitzer, Martin

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