Selectivity of Hydroxamate- and Difluoromethyloxadiazole-Based Inhibitors of Histone Deacetylase 6 In Vitro and in Cells von Ptacek, Jakub, Snajdr, Ivan, Schimer, Jiri, Kutil, Zsofia, Mikesova, Jana, Baranova, Petra, Havlinova, Barbora, Tueckmantel, Werner, Majer, Pavel, Kozikowski, Alan, Barinka, Cyril

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Highly enantioselective organocatalytic synthesis of piperidines. Formal synthesis of (−)-Paroxetine von Valero, Guillem, Schimer, Jiri, Cisarova, Ivana, Vesely, Jan, Moyano, Albert, Rios, Ramon

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iBodies: Modular Synthetic Antibody Mimetics Based on Hydrophilic Polymers Decorated with Functional Moieties von Šácha, Pavel, Knedlík, Tomáš, Schimer, Jiří, Tykvart, Jan, Parolek, Jan, Navrátil, Václav, Dvořáková, Petra, Sedlák, František, Ulbrich, Karel, Strohalm, Jiří, Majer, Pavel, Šubr, Vladimír, Konvalinka, Jan

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Stimulated Emission Depletion Nanoscopy Reveals Time-Course of Human Immunodeficiency Virus Proteolytic Maturation von Hanne, Janina, Göttfert, Fabian, Schimer, Jiří, Anders-Össwein, Maria, Konvalinka, Jan, Engelhardt, Johann, Müller, Barbara, Hell, Stefan W, Kräusslich, Hans-Georg

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Comparison of human glutamate carboxypeptidases II and III reveals their divergent substrate specificities von Navrátil, Michal, Tykvart, Jan, Schimer, Jiří, Pachl, Petr, Navrátil, Václav, Rokob, Tibor András, Hlouchová, Klára, Rulíšek, Lubomír, Konvalinka, Jan

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Structure-Aided Design of Novel Inhibitors of HIV Protease Based on a Benzodiazepine Scaffold von Schimer, Jiří, Cígler, Petr, Veselý, Jan, Grantz Šašková, Klára, Lepšík, Martin, Brynda, Jiří, Řezáčová, Pavlína, Kožíšek, Milan, Císařová, Ivana, Oberwinkler, Heike, Kraeusslich, Hans-Georg, Konvalinka, Jan

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Inhibitor-Decorated Polymer Conjugates Targeting Fibroblast Activation Protein von Dvořáková, Petra, Bušek, Petr, Knedlík, Tomáš, Schimer, Jiří, Etrych, Tomáš, Kostka, Libor, Stollinová Šromová, Lucie, Šubr, Vladimír, Šácha, Pavel, Šedo, Aleksi, Konvalinka, Jan

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Triggering HIV polyprotein processing by light using rapid photodegradation of a tight-binding protease inhibitor von Schimer, Jiří, Pávová, Marcela, Anders, Maria, Pachl, Petr, Šácha, Pavel, Cígler, Petr, Weber, Jan, Majer, Pavel, Řezáčová, Pavlína, Kräusslich, Hans-Georg, Müller, Barbara, Konvalinka, Jan

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Visualization of Sentinel Lymph Nodes with Mannosylated Fluorescent Nanodiamonds von Kvakova, Klaudia, Ondra, Martin, Schimer, Jiri, Petrik, Milos, Novy, Zbynek, Raabova, Helena, Hajduch, Marian, Cigler, Petr

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Design of Highly Potent Urea-Based, Exosite-Binding Inhibitors Selective for Glutamate Carboxypeptidase II von Tykvart, Jan, Schimer, Jiří, Jančařík, Andrej, Bařinková, Jitka, Navrátil, Václav, Starková, Jana, Šrámková, Karolína, Konvalinka, Jan, Majer, Pavel, Šácha, Pavel

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Nanoscale Dynamic Readout of a Chemical Redox Process Using Radicals Coupled with Nitrogen-Vacancy Centers in Nanodiamonds von Barton, Jan, Gulka, Michal, Tarabek, Jan, Mindarava, Yuliya, Wang, Zhenyu, Schimer, Jiri, Raabova, Helena, Bednar, Jan, Plenio, Martin B, Jelezko, Fedor, Nesladek, Milos, Cigler, Petr

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Rational design of urea-based glutamate carboxypeptidase II (GCPII) inhibitors as versatile tools for specific drug targeting and delivery von Tykvart, Jan, Schimer, Jiří, Bařinková, Jitka, Pachl, Petr, Poštová-Slavětínská, Lenka, Majer, Pavel, Konvalinka, Jan, Šácha, Pavel

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Inhibitor–Polymer Conjugates as a Versatile Tool for Detection and Visualization of Cancer-Associated Carbonic Anhydrase Isoforms von Pospíšilová, Klára, Knedlík, Tomáš, Šácha, Pavel, Kostka, Libor, Schimer, Jiří, Brynda, Jiří, Král, Vlastimil, Cígler, Petr, Navrátil, Václav, Etrych, Tomáš, Šubr, Vladimír, Kugler, Michael, Fábry, Milan, Řezáčová, Pavlína, Konvalinka, Jan

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DNA-linked Inhibitor Antibody Assay (DIANA) for sensitive and selective enzyme detection and inhibitor screening von Navrátil, Václav, Schimer, Jiří, Tykvart, Jan, Knedlík, Tomáš, Vik, Viktor, Majer, Pavel, Konvalinka, Jan, Šácha, Pavel

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Highly enantioselective organocatalytic cascade reaction for the synthesis of piperidines and oxazolidines von Číhalová, Sylva, Valero, Guillem, Schimer, Jiří, Humpl, Marek, Dračínský, Martin, Moyano, Albert, Rios, Ramon, Vesely, Jan

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Nanodiamonds as traps for fibroblast growth factors: Parameters influencing the interaction von Mikesova, Jana, Miliaieva, Daria, Stenclova, Pavla, Kindermann, Marek, Vuckova, Tereza, Madlikova, Marcela, Fabry, Milan, Veverka, Vaclav, Schimer, Jiri, Krejci, Pavel, Stehlik, Stepan, Cigler, Petr

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Glycan-Modified Virus-like Particles Evoke T Helper Type 1‑like Immune Responses von Alam, Mohammad Murshid, Jarvis, Cassie M, Hincapie, Robert, McKay, Craig S, Schimer, Jiri, Sanhueza, Carlos A, Xu, Ke, Diehl, Roger C, Finn, M. G, Kiessling, Laura L

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Lung Tissue Delivery of Virus-Like Particles Mediated by Macrolide Antibiotics von Crooke, Stephen N, Schimer, Jiri, Raji, Idris, Wu, Bocheng, Oyelere, Adegboyega K, Finn, M. G

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Identification of Novel Carbonic Anhydrase IX Inhibitors Using High-Throughput Screening of Pooled Compound Libraries by DNA-Linked Inhibitor Antibody Assay (DIANA) von Tykvart, Jan, Navrátil, Václav, Kugler, Michael, Šácha, Pavel, Schimer, Jiří, Hlaváčková, Anna, Tenora, Lukáš, Zemanová, Jitka, Dejmek, Milan, Král, Vlastimil, Potáček, Milan, Majer, Pavel, Jahn, Ullrich, Brynda, Jiří, Řezáčová, Pavlína, Konvalinka, Jan

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iBodies: Modular Synthetic Antibody Mimetics Based on Hydrophilic Polymers Decorated with Functional Moieties von Šácha, Pavel, Knedlík, Tomáš, Schimer, Jiří, Tykvart, Jan, Parolek, Jan, Navrátil, Václav, Dvořáková, Petra, Sedlák, František, Ulbrich, Karel, Strohalm, Jiří, Majer, Pavel, Šubr, Vladimír, Konvalinka, Jan

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