DNA-Encoded Library-Derived DDR1 Inhibitor Prevents Fibrosis and Renal Function Loss in a Genetic Mouse Model of Alport Syndrome von Richter, Hans, Satz, Alexander L, Bedoucha, Marc, Buettelmann, Bernd, Petersen, Ann C, Harmeier, Anja, Hermosilla, Ricardo, Hochstrasser, Remo, Burger, Dominique, Gsell, Bernard, Gasser, Rodolfo, Huber, Sylwia, Hug, Melanie N, Kocer, Buelent, Kuhn, Bernd, Ritter, Martin, Rudolph, Markus G, Weibel, Franziska, Molina-David, Judith, Kim, Jin-Ju, Santos, Javier Varona, Stihle, Martine, Georges, Guy J, Bonfil, R. Daniel, Fridman, Rafael, Uhles, Sabine, Moll, Solange, Faul, Christian, Fornoni, Alessia, Prunotto, Marco

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Assessment of AI-Based Protein Structure Prediction for the NLRP3 Target von Yin, Jian, Lei, Junkun, Yu, Jialin, Cui, Weiren, Satz, Alexander L, Zhou, Yifan, Feng, Hua, Deng, Jason, Su, Wenji, Kuai, Letian

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What Do You Get from DNA-Encoded Libraries? von Satz, Alexander L

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Simulated Screens of DNA Encoded Libraries: The Potential Influence of Chemical Synthesis Fidelity on Interpretation of Structure–Activity Relationships von Satz, Alexander L.

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DNA Encoded Library Selections and Insights Provided by Computational Simulations von Satz, Alexander L

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Selections and screenings of DNA-encoded chemical libraries against enzyme and cellular targets von Satz, Alexander L., Kuai, Letian, Peng, Xuanjia

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Discovery of SARS-CoV-2 main protease covalent inhibitors from a DNA-encoded library selection von Ge, Rui, Shen, Zuyuan, Yin, Jian, Chen, Wenhua, Zhang, Qi, An, Yulong, Tang, Dewei, Satz, Alexander L., Su, Wenji, Kuai, Letian

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Discovery and Characterization of a Class of Pyrazole Inhibitors of Bacterial Undecaprenyl Pyrophosphate Synthase von Concha, Nestor, Huang, Jianzhong, Bai, Xiaopeng, Benowitz, Andrew, Brady, Pat, Grady, LaShadric C, Kryn, Luz Helena, Holmes, David, Ingraham, Karen, Jin, Qi, Pothier Kaushansky, Laura, McCloskey, Lynn, Messer, Jeffrey A, O’Keefe, Heather, Patel, Amish, Satz, Alexander L, Sinnamon, Robert H, Schneck, Jessica, Skinner, Steve R, Summerfield, Jennifer, Taylor, Amy, Taylor, J. David, Evindar, Ghotas, Stavenger, Robert A

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Development of DNA-Compatible Van Leusen Three-Component Imidazole Synthesis von Geigle, Stefanie N, Petersen, Ann C, Satz, Alexander L

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Analysis of Current DNA Encoded Library Screening Data Indicates Higher False Negative Rates for Numerically Larger Libraries von Satz, Alexander L, Hochstrasser, Remo, Petersen, Ann C

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High-Throughput Solid-Phase Building Block Synthesis for DNA-Encoded Libraries von Zambaldo, Claudio, Geigle, Stefanie N, Satz, Alexander L

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Solution-Phase DNA-Compatible Pictet-Spengler Reaction Aided by Machine Learning Building Block Filtering von Li, Ke, Liu, Xiaohong, Liu, Sixiu, An, Yulong, Shen, Yanfang, Sun, Qingxia, Shi, Xiaodong, Su, Wenji, Cui, Weiren, Duan, Zhiqiang, Kuai, Letian, Yang, Hongfang, Satz, Alexander L., Chen, Kaixian, Jiang, Hualiang, Zheng, Mingyue, Peng, Xuanjia, Lu, Xiaojie

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DNA-Compatible Cyclization Reaction to Access 1,3,4-Oxadiazoles and 1,2,4-Triazoles von Wang, Gaonan, Tan, Yu, Zou, Hanzhi, Sui, Xihang, Wang, Zhanlong, Satz, Alexander L., Kuai, Letian, Su, Wenji, Zhang, Qi

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Analysis of the productivity of DNA encoded libraries von Eidam, Oliv, Satz, Alexander L.

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Synthesis of 1,2-Amino Alcohols by Photoredox-Mediated Decarboxylative Coupling of α‑Amino Acids and DNA-Conjugated Carbonyls von Wen, Huanan, Ge, Rui, Qu, Yi, Sun, Jialin, Shi, Xiaodong, Cui, Weiren, Yan, Hao, Zhang, Qi, An, Yulong, Su, Wenji, Yang, Hongfang, Kuai, Letian, Satz, Alexander L, Peng, Xuanjia

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Activity-Based DNA-Encoded Library Screening von Cochrane, Wesley G, Malone, Marie L, Dang, Vuong Q, Cavett, Valerie, Satz, Alexander L, Paegel, Brian M

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Triaging of DNA-Encoded Library Selection Results by High-Throughput Resynthesis of DNA–Conjugate and Affinity Selection Mass Spectrometry von Su, Wenji, Ge, Rui, Ding, Duanchen, Chen, Wenhua, Wang, Wenqing, Yan, Hao, Wang, Weikun, Yuan, Youlang, Liu, Huan, Zhang, Meng, Zhang, Jiyuan, Shu, Qisheng, Satz, Alexander L, Kuai, Letian

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Palladium-mediated Suzuki-Miyaura Cross-Coupling Reaction of Potassium Boc-protected aminomethyltrifluoroborate with DNA-Conjugated aryl bromides for DNA-Encoded chemical library s... von Qu, Yi, Liu, Sixiu, Wen, Huanan, Xu, Yanfen, An, Yulong, Li, Ke, Ni, Mengyuan, Shen, Yanfang, Shi, Xiaodong, Su, Wenji, Cui, Weiren, Kuai, Letian, Satz, Alexander L., Yang, Hongfang, Lu, Xiaojie, Peng, Xuanjia

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Discovery of a Highly Selective BET BD2 Inhibitor from a DNA-Encoded Library Technology Screening Hit von Rianjongdee, Francesco, Atkinson, Stephen J, Chung, Chun-wa, Grandi, Paola, Gray, James R. J, Kaushansky, Laura J, Medeiros, Patricia, Messenger, Cassie, Phillipou, Alex, Preston, Alex, Prinjha, Rab K, Rioja, Inmaculada, Satz, Alexander L, Taylor, Simon, Wall, Ian D, Watson, Robert J, Yao, Gang, Demont, Emmanuel H

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Copper-Mediated DNA-Compatible One-Pot Click Reactions of Alkynes with Aryl Borates and TMS-N-3 von Qu, Yi, Wen, Huanan, Ge, Rui, Xu, Yanfen, Gao, Hong, Shi, Xiaodong, Wang, Jiangong, Cui, Weiren, Su, Wenji, Yang, Hongfang, Kuai, Letian, Satz, Alexander L., Peng, Xuanjia

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