Organocatalytic enantioselective synthesis of 2,5,5-trisubstituted piperidines bearing a quaternary stereocenter. Vinyl sulfonamide as a new amine protecting group von Escolano, Marcos, Guerola, Marta, Torres, Javier, Gaviña, Daniel, Alzuet-Piña, Gloria, Sánchez-Rosello, María, del Pozo, Carlos

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A Versatile Approach to CF3-Containing 2-Pyrrolidones by Tandem Michael Addition-Cyclization: Exemplification in the Synthesis of Amidine Class BACE1 Inhibitors von Mateu, Natalia, Ciordia, Myriam, Delgado, Oscar, Sánchez-Roselló, María, Trabanco, Andrés A., Van Gool, Michiel, Tresadern, Gary, Pérez-Benito, Laura, Fustero, Santos

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N-Sulfinyl Amines as a Nitrogen Source in the Asymmetric Intramolecular Aza-Michael Reaction: Total Synthesis of (−)-Pinidinol von Fustero, Santos, Monteagudo, Silvia, Sánchez-Roselló, María, Flores, Sonia, Barrio, Pablo, del Pozo, Carlos

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Organocatalytic Enantioselective Synthesis of Trifluoromethyl‐Containing Tetralin Derivatives by Sequential (Hetero)Michael Reaction–Intramolecular Nitrone Cycloaddition von Rabasa‐Alcañiz, Fernando, Torres, Javier, Sánchez‐Roselló, María, Tejero, Tomás, Merino, Pedro, Fustero, Santos, del Pozo, Carlos

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A Versatile Approach to CF3-Containing 2-Pyrrolidones by Tandem Michael Addition-Cyclization: Exemplification in the Synthesis of Amidine Class BACE1 Inhibitors von Mateu, Natalia, Ciordia, Myriam, Delgado, Oscar, Sánchez-Roselló, María, Trabanco, Andrés A., Van Gool, Michiel, Tresadern, Gary, Pérez-Benito, Laura, Fustero, Santos

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New Cathepsin Inhibitors to Explore the Fluorophilic Properties of the S2 Pocket of Cathepsin B: Design, Synthesis, and Biological Evaluation von Fustero, Santos, Rodrigo, Vanessa, Sánchez-Roselló, María, del Pozo, Carlos, Timoneda, Joaquín, Frizler, Maxim, Sisay, Mihiret T., Bajorath, Jürgen, Calle, Luis P., Cañada, F. Javier, Jiménez-Barbero, Jesús, Gütschow, Michael

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Synthesis and enzymatic evaluation of novel partially fluorinated thiol dual ACE/NEP inhibitors von Olimpieri, Francesca, Tambaro, Simone, Fustero, Santos, Lazzari, Paolo, Sanchez-Roselló, Maria, Pani, Luca, Volonterio, Alessandro, Zanda, Matteo

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Microwave-Assisted Tandem Cross Metathesis Intramolecular Aza-Michael Reaction:  An Easy Entry to Cyclic β-Amino Carbonyl Derivatives von Fustero, Santos, Jiménez, Diego, Sánchez-Roselló, María, del Pozo, Carlos

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Tandem Gold Self-Relay Catalysis for the Synthesis of 2,3-Dihydropyridin-4(1H)-ones: Combination of [sigma] and [pi] Lewis Acid Properties of Gold Salts von Fustero, Santos, Miro, Javier, Sanchez-Rosello, María, delPozo, Carlos

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Fluorine in Pharmaceutical Industry: Fluorine-Containing Drugs Introduced to the Market in the Last Decade (2001–2011) von Wang, Jiang, Sánchez-Roselló, María, Aceña, José Luis, del Pozo, Carlos, Sorochinsky, Alexander E, Fustero, Santos, Soloshonok, Vadim A, Liu, Hong

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From 2000 to Mid-2010: A Fruitful Decade for the Synthesis of Pyrazoles von Fustero, Santos, Sánchez-Roselló, María, Barrio, Pablo, Simón-Fuentes, Antonio

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Recent Strategies in the Nucleophilic Dearomatization of Pyridines, Quinolines, and Isoquinolines von Escolano, Marcos, Gaviña, Daniel, Alzuet-Piña, Gloria, Díaz-Oltra, Santiago, Sánchez-Roselló, María, Pozo, Carlos del

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Role of the gem-Difluoro Moiety in the Tandem Ring-Closing Metathesis−Olefin Isomerization:  Regioselective Preparation of Unsaturated Lactams von FUSTERO, Santos, SáNCHEZ-ROSELLó, María, JIMéNEZ, Diego, SANZ-CERVERA, Juan F., DEL POZO, Carlos, ACEñA, José Luis

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A general overview of the organocatalytic intramolecular aza-Michael reaction von Sánchez-Roselló, María, Aceña, José Luis, Simón-Fuentes, Antonio, del Pozo, Carlos

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Organocatalytic Enantioselective Friedel‐Crafts Alkylation Reactions of Pyrroles von Gaviña, Daniel, Escolano, Marcos, Torres, Javier, Alzuet‐Piña, Gloria, Sánchez‐Roselló, María, Pozo, Carlos

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Site-Selective Catalysis of Phenyl Thionoformate Transfer as a Tool for Regioselective Deoxygenation of Polyols von Sánchez-Roselló, María, Puchlopek, Angela L. A, Morgan, Adam J, Miller, Scott J

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Two Decades of Progress in the Asymmetric Intramolecular aza‐Michael Reaction von Sánchez‐Roselló, María, Escolano, Marcos, Gaviña, Daniel, Pozo, Carlos

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Asymmetric Synthesis of New β,β-Difluorinated Cyclic Quaternary α-Amino Acid Derivatives von Fustero, Santos, Sánchez-Roselló, Maria, Rodrigo, Vanessa, del Pozo, Carlos, Sanz-Cervera, Juan F, Simón, Antonio, Ramírez de Arellano, Carmen

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Cover Picture: A Versatile Approach to CF3-Containing 2-Pyrrolidones by Tandem Michael Addition-Cyclization: Exemplification in the Synthesis of Amidine Class BACE1 Inhibitors (Che... von Mateu, Natalia, Ciordia, Myriam, Delgado, Oscar, Sánchez-Roselló, María, Trabanco, Andrés A., Van Gool, Michiel, Tresadern, Gary, Pérez-Benito, Laura, Fustero, Santos

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Tandem Organocatalytic Cycloaromatization/Intramolecular Friedel–Crafts Alkylation Sequence for the Synthesis of Indolizinones and Pyrrolo-azepinone Derivatives von Rabasa-Alcañiz, Fernando, Sánchez-Roselló, María, Fustero, Santos, del Pozo, Carlos

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