Discovery of a Potent and Orally Efficacious TGR5 Receptor Agonist von Agarwal, Sameer, Patil, Amit, Aware, Umesh, Deshmukh, Prashant, Darji, Brijesh, Sasane, Santosh, Sairam, Kalapatapu V. V. M, Priyadarsiny, Priyanka, Giri, Poonam, Patel, Harilal, Giri, Suresh, Jain, Mukul, Desai, Ranjit C

Volltext

Discovery of potent, selective and orally bioavailable triaryl-sulfonamide based PTP1B inhibitors von Patel, Dipam, Jain, Mukul, Shah, Shailesh R., Bahekar, Rajesh, Jadav, Pradip, Joharapurkar, Amit, Dhanesha, Nirav, Shaikh, Mubeen, Sairam, Kalapatapu V.V.M., Kapadnis, Prashant

Volltext

Long-acting peptidomimetics based DPP-IV inhibitors von Jadav, Pradip, Bahekar, Rajesh, Shah, Shailesh R., Patel, Dipam, Joharapurkar, Amit, Kshirsagar, Samadhan, Jain, Mukul, Shaikh, Mubeen, Sairam, Kalapatapu V.V.M.

Volltext

Synthesis and structure–activity relationship of potent, selective and orally active anthranilamide-based factor Xa inhibitors: Application of weakly basic sulfoximine group as nov... von Pandya, Vrajesh, Jain, Mukul, Chakrabarti, Ganes, Soni, Hitesh, Parmar, Bhavesh, Chaugule, Balaji, Patel, Jigar, Jarag, Tushar, Joshi, Jignesh, Joshi, Nirav, Rath, Akshyaya, Unadkat, Vishal, Sharma, Bhavesh, Ajani, Haresh, Kumar, Jeevan, Sairam, Kalapatapu V.V.M., Patel, Harilal, Patel, Pankaj

Volltext

Discovery of liver selective non-steroidal glucocorticoid receptor antagonist as novel antidiabetic agents von Shah, Kiran, Patel, Dipam, Jadav, Pradip, Sheikh, Mubeen, Sairam, Kalapatapu V.V.M., Joharapurkar, Amit, Jain, Mukul R., Bahekar, Rajesh

Volltext

Discovery of inhibitors of plasminogen activator inhibitor-1: Structure–activity study of 5-nitro-2-phenoxybenzoic acid derivatives von Pandya, Vrajesh, Jain, Mukul, Chakrabarti, Ganes, Soni, Hitesh, Parmar, Bhavesh, Chaugule, Balaji, Patel, Jigar, Joshi, Jignesh, Joshi, Nirav, Rath, Akshyaya, Raviya, Mehul, Shaikh, Mubeen, Sairam, Kalapatapu V.V.M., Patel, Harilal, Patel, Pankaj

Volltext

Discovery of Orally Active, Potent, and Selective Benzotriazole-Based PTP1B Inhibitors von Patel, Dipam, Jain, Mukul, Shah, Shailesh R., Bahekar, Rajesh, Jadav, Pradip, Darji, Brijesh, Siriki, Yernaidu, Bandyopadhyay, Debdutta, Joharapurkar, Amit, Kshirsagar, Samadhan, Patel, Harilal, Shaikh, Mubeen, Sairam, Kalapatapu V. V. M., Patel, Pankaj

Volltext

In the Quest for Potent and Selective Malic Enzyme 3 Inhibitors for the Treatment of Pancreatic Ductal Adenocarcinoma von Sheth, Gaurav, Shah, Shailesh R., Sengupta, Prabal, Jarag, Tushar, Chimanwala, Sabbirhusen, Sairam, Kalapatapu V. V. M., Jain, Vaibhav, Talwar, Rashmi, Dhanave, Avinash, Raviya, Mehul, Menon, Soumya, Trivedi, Shivangi, Chitturi, Trinadha Rao

Volltext

Modulation of PPAR receptor subtype selectivity of the ligands: Aliphatic chain vs aromatic ring as a spacer between pharmacophore and the lipophilic moiety von Pingali, Harikishore, Jain, Mukul, Shah, Shailesh, Patil, Pravin, Makadia, Pankaj, Zaware, Pandurang, Sairam, Kalapatapu V.V.M., Jamili, Jeevankumar, Goel, Ashish, Patel, Megha, Patel, Pankaj

Volltext

Design, synthesis and biological evaluation of novel aminomethyl-piperidones based DPP-IV inhibitors von Jadav, Pradip, Bahekar, Rajesh, Shah, Shailesh R, Patel, Dipam, Joharapurkar, Amit, Jain, Mukul, Sairam, Kalapatapu V V M, Singh, Praveen Kumar

Volltext

Modulation of PPAR subtype selectivity. Part 2: Transforming PPAR α/ γ dual agonist into α selective PPAR agonist through bioisosteric modification von Zaware, Pandurang, Shah, Shailesh R., Pingali, Harikishore, Makadia, Pankaj, Thube, Baban, Pola, Suresh, Patel, Darshit, Priyadarshini, Priyanka, Suthar, Dinesh, Shah, Maanan, Jamili, Jeevankumar, Sairam, Kalapatapu V.V.M., Giri, Suresh, Patel, Lala, Patel, Harilal, Sudani, Hareshkumar, Patel, Hiren, Jain, Mukul, Patel, Pankaj, Bahekar, Rajesh

Volltext

Facile synthesis, ex-vivo and in vitro screening of 3-sulfonamide derivative of 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxylic acid piperidin-1-ylamide... von Kumar Srivastava, Brijesh, Soni, Rina, Patel, Jayendra Z, Jha, Satadru, Shedage, Sandeep A, Gandhi, Neha, Sairam, Kalapatapu V V M, Pawar, Vishwanath, Sadhwani, Nisha, Mitra, Prasenjit, Jain, Mukul R, Patel, Pankaj R

Volltext

Bioisosteric replacement of dihydropyrazole of 4S-(-)-3-(4-chlorophenyl)-N-methyl-N'-[(4-chlorophenyl)-sulfonyl]-4-phenyl-4,5-dihydro-1H-pyrazole-1-caboxamidine (SLV-319) a potent... von Srivastava, Brijesh Kumar, Soni, Rina, Joharapurkar, Amit, Sairam, Kalapatapu V V M, Patel, Jayendra Z, Goswami, Amitgiri, Shedage, Sandeep A, Kar, Sidhartha S, Salunke, Rahul P, Gugale, Shivaji B, Dhawas, Amol, Kadam, Pravin, Mishra, Bhupendra, Sadhwani, Nisha, Unadkat, Vishal B, Mitra, Prasenjit, Jain, Mukul R, Patel, Pankaj R

Volltext

Three Dimensional Pharmacophore Modelling of Monoamine oxidase-A (MAO-A) inhibitors von Sairam, Kalapatapu V.V.M., Khar, Roop K., Mukherjee, Rama, Jain, Swatantra K.

Volltext

Design, synthesis and biological evaluation of γ-lactam hydroxamate based TACE inhibitors von Argade, Anil, Bahekar, Rajesh, Desai, Jigar, Thombare, Pravin, Shah, Kiran, Gite, Sanjay, Sunder, Rajesh, Ranvir, Ramchandra, Bandyopadhyay, Debdutta, Chakrabarti, Ganes, Joharapurkar, Amit, Mahapatra, Jogeswar, Chatterjee, Abhijit, Patel, Harilal, Shaikh, Mubeen, Sairam, Kalapatapu V. V. M., Jain, Mukul, Patel, Pankaj

Volltext

3D-QSAR studies of some [[1-aryl(or benzyl)-1-(benzenesulphonamido)methyl] phenyl] alkanoic acid derivatives as thromboxane A2 receptor antagonists von SAIRAM, Kalapatapu V. V. M, SARMA, Jagarlapudi A. R. P, DESIRAJU, Gautam R

Volltext

ChemInform Abstract: Discovery of Liver Selective Non-Steroidal Glucocorticoid Receptor Antagonist as Novel Antidiabetic Agents von Shah, Kiran, Patel, Dipam, Jadav, Pradip, Sheikh, Mubeen, Sairam, Kalapatapu V. V. M., Joharapurkar, Amit, Jain, Mukul R., Bahekar, Rajesh

Volltext

Facile synthesis, ex-vivo and in vitro screening of 3-sulfonamide derivative of 5-(4-chlorophenyl)-l-(2.4-dichlorophenyl)-4-methyl-lH-pyrazole-3-carboxylic acid piperidin-1-ylamide... von BRIJESH KUMAR SRIVASTAVA, SONI, Rina, JAIN, Mukul R, PATEL, Pankaj R, PATEL, Jayendra Z, JHA, Satadru, SHEDAGE, Sandeep A, GANDHI, Neha, SAIRAM, Kalapatapu V. V. M, PAWAR, Vishwanath, SADHWANI, Nisha, MITRA, Prasenjit

Volltext

Bioisosteric replacement of dihydropyrazole of 4S-(-)-3-(4-chlorophenyl)-N-methyl-N'-[(4-chlorophenyl)-sulfonyl]-4-phenyl-4,5-dihydro-lH-pyrazole-1-caboxamidine (SLV-319) a potent... von BRIJESH KUMAR SRIVASTAVA, SONI, Rina, DHAWAS, Amol, KADAM, Pravin, MISHRA, Bhupendra, SADHWANI, Nisha, UNADKAT, Vishal B, MITRA, Prasenjit, JAIN, Mukul R, PATEL, Pankaj R, JOHARAPURKAR, Amit, SAIRAM, Kalapatapu V. V. M, PATEL, Jayendra Z, GOSWAMI, Amitgiri, SHEDAGE, Sandeep A, KAR, Sidhartha S, SALUNKE, Rahul P, GUGALE, Shivaji B

Volltext

Malic enzyme inhibitors von Kalapatapu, Sairam V V M, Chitturi, Trinadha Rao, Venkat, Raj Gopal, Sengupta, Prabal, Sheth, Gaurav Sanjivkumar, Hampiholi, Aishwarya, Maity, Saikat, Jarag, Tushar Mukund, Chimanwala, Sabbirhusen Yusufbhai, Kadiyala, V. S. N. Murty, Jain, Vaibhav, Qureshi, Gulamnizami Abdulsattar, Chaudhari, Umesh Vishnu

Volltext bestellen