Discovery of a Potent Analgesic NOP and Opioid Receptor Agonist: Cebranopadol von Schunk, Stefan, Linz, Klaus, Hinze, Claudia, Frormann, Sven, Oberbörsch, Stefan, Sundermann, Bernd, Zemolka, Saskia, Englberger, Werner, Germann, Tieno, Christoph, Thomas, Kögel, Babette-Y, Schröder, Wolfgang, Harlfinger, Stephanie, Saunders, Derek, Kless, Achim, Schick, Hans, Sonnenschein, Helmut

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Design and synthesis of spirocyclic ligands of glucocorticoid receptors von Badarau, Eduard, Robert, Frédéric, Massip, Stéphane, Jakob, Florian, Lucas, Simon, Frormann, Sven, Ghosez, Léon

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Discovery of a subnanomolar and selective spirocyclic agonist of the glucocorticoid receptor von Badarau, Eduard, Robert, Frédéric, Massip, Stéphane, Jakob, Florian, Lucas, Simon, Friebe, Daniela, Hennen, Stephanie, Frormann, Sven, Ghosez, Léon

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Crystal Structure of an Inhibitor Complex of the 3C Proteinase from Hepatitis A Virus (HAV) and Implications for the Polyprotein Processing in HAV von Bergmann, Ernst M., Cherney, Maia M., Mckendrick, John, Frormann, Sven, Luo, Colin, Malcolm, Bruce A., Vederas, John C., James, Michael N.G.

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Discovery of Spiro[cyclohexane-dihydropyrano[3,4‑b]indole]-amines as Potent NOP and Opioid Receptor Agonists von Schunk, Stefan, Linz, Klaus, Frormann, Sven, Hinze, Claudia, Oberbörsch, Stefan, Sundermann, Bernd, Zemolka, Saskia, Englberger, Werner, Germann, Tieno, Christoph, Thomas, Kögel, Babette-Y, Schröder, Wolfgang, Harlfinger, Stephanie, Saunders, Derek, Kless, Achim, Schick, Hans, Sonnenschein, Helmut

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Pyridine C-region analogs of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as potent TRPV1 antagonists von Ryu, HyungChul, Seo, Sejin, Lee, Jee-Young, Ha, Tae-Hwan, Lee, Sunho, Jung, Aeran, Ann, Jihyae, Kim, Sung-Eun, Yoon, Suyoung, Hong, Mannkyu, Blumberg, Peter M., Frank-Foltyn, Robert, Bahrenberg, Gregor, Schiene, Klaus, Stockhausen, Hannelore, Christoph, Thomas, Frormann, Sven, Lee, Jeewoo

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2-Alkyl/alkenyl substituted pyridine C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as highly potent TRPV1 antagonists von Ryu, HyungChul, Seo, Sejin, Cho, Seong-Hee, Kim, Ho Shin, Jung, Aeran, Kang, Dong Wook, Son, Karam, Cui, Minghua, Hong, Sun-hye, Sharma, Pankaz Kumar, Choi, Sun, Blumberg, Peter M., Frank-Foltyn, Robert, Bahrenberg, Gregor, Stockhausen, Hannelore, Schiene, Klaus, Christoph, Thomas, Frormann, Sven, Lee, Jeewoo

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2-Aryl substituted pyridine C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as highly potent TRPV1 antagonists von Ryu, HyungChul, Seo, Sejin, Kim, Myeong Seop, Kim, Mi-Yeon, Kim, Ho Shin, Ann, Jihyae, Tran, Phuong-Thao, Hoang, Van-Hai, Byun, Jieun, Cui, Minghua, Son, Karam, Sharma, Pankaz Kumar, Choi, Sun, Blumberg, Peter M., Frank-Foltyn, Robert, Bahrenberg, Gregor, Koegel, Babette-Yvonne, Christoph, Thomas, Frormann, Sven, Lee, Jeewoo

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6,6-Fused heterocyclic ureas as highly potent TRPV1 antagonists von Sun, Wei, Kim, Hyo-Shin, Lee, Sunho, Jung, Aeran, Kim, Sung-Eun, Ann, Jihyae, Yoon, Suyoung, Choi, Sun, Lee, Jin Hee, Blumberg, Peter M., Frank-Foltyn, Robert, Bahrenberg, Gregor, Schiene, Klaus, Stockhausen, Hannelore, Christoph, Thomas, Frormann, Sven, Lee, Jeewoo

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TRPV1 antagonist with high analgesic efficacy: 2-Thio pyridine C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides von Ha, Tae-Hwan, Ryu, HyungChul, Kim, Sung-Eun, Kim, Ho Shin, Ann, Jihyae, Tran, Phuong-Thao, Hoang, Van-Hai, Son, Karam, Cui, Minghua, Choi, Sun, Blumberg, Peter M., Frank, Robert, Bahrenberg, Gregor, Schiene, Klaus, Christoph, Thomas, Frormann, Sven, Lee, Jeewoo

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In vitro and ex vivo inhibition of hepatitis A virus 3C proteinase by a peptidyl monofluoromethyl ketone von Morris, Tina S, Frormann, Sven, Shechosky, Shirley, Lowe, Christopher, Lall, Manjinder S, Gauss-Müller, Verena, Purcell, Robert H, Emerson, Suzanne U, Vederas, John C, Malcolm, Bruce A

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Rapid mass spectrometric determination of preferred irreversible proteinase inhibitors in combinatorial libraries von Mckendrick, John E., Frormann, Sven, Luo, Colin, Semchuck, Paul, Vederas, John C., Malcolm, Bruce A.

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AROMATIC AZA COMPOUNDS AS VR1/TRPV1 LIGANDS von Frank-Foltyn, Robert, Dr, Sven, Frormann, Dr, Chistoph, Thomas, Dr

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SUBSTITUTED BICYCLIC CARBOXAMIDE AND UREA DERIVATIVES AS VANILLOID RECEPTOR LIGANDS von FRORMANN, SVEN, FRANK, ROBERT, CHRISTOPH, THOMAS

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Substituted bicyclic carboxamide and urea derivatives as vanilloid receptor ligands von FRORMANN, SVEN, FRANK, ROBERT, CHRISTOPH, THOMAS

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Carboxamida substituída à base de tiazol e oxazol e derivados de ureia como ligantes de receptor vanilóide ii von SAUNDERS DEREK, HABERMANN CHRISTOPHER, STOCKHAUSEN HANNELORE, DAMANN NILS, LESCH BERNHARD, FRANK-FOLTYN ROBERT, FRORMANN SVEN, LEE JEEWOO, CHRISTOPH THOMAS, BAHRENBERG GREGOR, SCHIENE KLAUS

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SUBSTITUTED OXAZOLE- AND THIAZOLE-BASED CARBOXAMIDE AND UREA DERIVATIVES AS VANILLOID RECEPTOR LIGANDS II von LEE, Jeewoo, DAMANN, Nils, CHRISTOPH, Thomas, FRORMANN, Sven, SAUNDERS, Derek, LESCH, Bernhard, BAHRENBERG, Gregor, SCHIENE, Klaus, STOCKHAUSEN, Hannelore, HABERMANN, Christopher, FRANK-FOLTYN, Robert

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HYDROXYMETHYLCYCLOHEXYLAMINES von LINZ, KLAUS, FRORMANN, SVEN, THEIL, FRITZ, ZEMOLKA, SASKIA, ENGLBERGER, WERNER

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HYDROXYMETHYLCYCLOHEXYLAMINES von LINZ, KLAUS, FRORMANN, SVEN, THEIL, FRITZ, ZEMOLKA, SASKIA, ENGLBERGER, WERNER

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HYDROXYMETHYLCYCLOHEXYLAMINES von THEIL FRITZ, FRORMANN SVEN, LINZ KLAUS, ENGLBERGER WERNER, ZEMOLKA SASKIA

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