Canonical PRC1 controls sequence-independent propagation of Polycomb-mediated gene silencing von Moussa, Hagar F., Bsteh, Daniel, Yelagandula, Ramesh, Pribitzer, Carina, Stecher, Karin, Bartalska, Katarina, Michetti, Luca, Wang, Jingkui, Zepeda-Martinez, Jorge A., Elling, Ulrich, Stuckey, Jacob I., James, Lindsey I., Frye, Stephen V., Bell, Oliver

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A cellular chemical probe targeting the chromodomains of Polycomb repressive complex 1 von Stuckey, Jacob I, Dickson, Bradley M, Cheng, Nancy, Liu, Yanli, Norris, Jacqueline L, Cholensky, Stephanie H, Tempel, Wolfram, Qin, Su, Huber, Katherine G, Sagum, Cari, Black, Karynne, Li, Fengling, Huang, Xi-Ping, Roth, Bryan L, Baughman, Brandi M, Senisterra, Guillermo, Pattenden, Samantha G, Vedadi, Masoud, Brown, Peter J, Bedford, Mark T, Min, Jinrong, Arrowsmith, Cheryl H, James, Lindsey I, Frye, Stephen V

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Discovery and Characterization of a Cellular Potent Positive Allosteric Modulator of the Polycomb Repressive Complex 1 Chromodomain, CBX7 von Lamb, Kelsey N., Bsteh, Daniel, Dishman, Sarah N., Moussa, Hagar F., Fan, Huitao, Stuckey, Jacob I., Norris, Jacqueline L., Cholensky, Stephanie H., Li, Dongxu, Wang, Jingkui, Sagum, Cari, Stanton, Benjamin Z., Bedford, Mark T., Pearce, Kenneth H., Kenakin, Terry P., Kireev, Dmitri B., Wang, Gang Greg, James, Lindsey I., Bell, Oliver, Frye, Stephen V.

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Structure–Activity Relationships and Kinetic Studies of Peptidic Antagonists of CBX Chromodomains von Stuckey, Jacob I, Simpson, Catherine, Norris-Drouin, Jacqueline L, Cholensky, Stephanie H, Lee, Junghyun, Pasca, Ryan, Cheng, Nancy, Dickson, Bradley M, Pearce, Kenneth H, Frye, Stephen V, James, Lindsey I

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Chromodomain Ligand Optimization via Target-Class Directed Combinatorial Repurposing von Barnash, Kimberly D, Lamb, Kelsey N, Stuckey, Jacob I, Norris, Jacqueline L, Cholensky, Stephanie H, Kireev, Dmitri B, Frye, Stephen V, James, Lindsey I

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Discovery of Peptidomimetic Ligands of EED as Allosteric Inhibitors of PRC2 von Barnash, Kimberly D, The, Juliana, Norris-Drouin, Jacqueline L, Cholensky, Stephanie H, Worley, Beau M, Li, Fengling, Stuckey, Jacob I, Brown, Peter J, Vedadi, Masoud, Arrowsmith, Cheryl H, Frye, Stephen V, James, Lindsey I

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Identification and characterization of second-generation EZH2 inhibitors with extended residence times and improved biological activity von Stuckey, Jacob I., Cantone, Nico R., Côté, Alexandre, Arora, Shilpi, Vivat, Valerie, Ramakrishnan, Ashwin, Mertz, Jennifer A., Khanna, Avinash, Brenneman, Jehrod, Gehling, Victor S., Moine, Ludivine, Sims, Robert J., Audia, James E., Trojer, Patrick, Levell, Julian R., Cummings, Richard T.

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Design, Synthesis, and Pharmacological Evaluation of Second Generation EZH2 Inhibitors with Long Residence Time von Khanna, Avinash, Côté, Alexandre, Arora, Shilpi, Moine, Ludivine, Gehling, Victor S., Brenneman, Jehrod, Cantone, Nico, Stuckey, Jacob I., Apte, Shruti, Ramakrishnan, Ashwin, Bruderek, Kamil, Bradley, William D., Audia, James E., Cummings, Richard T., Sims, Robert J., Trojer, Patrick, Levell, Julian R.

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Quantitative Characterization of Bivalent Probes for a Dual Bromodomain Protein, Transcription Initiation Factor TFIID Subunit 1 von Suh, Junghyun L, Watts, Brian, Stuckey, Jacob I, Norris-Drouin, Jacqueline L, Cholensky, Stephanie H, Dickson, Bradley M, An, Yi, Mathea, Sebastian, Salah, Eidarus, Knapp, Stefan, Khan, Abid, Adams, Alexander T, Strahl, Brian D, Sagum, Cari A, Bedford, Mark T, James, Lindsey I, Kireev, Dmitri B, Frye, Stephen V

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Correction to “Quantitative Characterization of Bivalent Probes for a Dual Bromodomain Protein, Transcription Initiation Factor TFIID subunit 1” von Suh, Junghyun L, Watts, Brian, Stuckey, Jacob I, Norris-Drouin, Jacqueline L, Cholensky, Stephanie H, Dickson, Bradley M, An, Yi, Mathea, Sebastian, Salah, Eidarus, Knapp, Stefan, Khan, Abid, Adams, Alexander T, Strahl, Brian D, Sagum, Cari A, Bedford, Mark T, James, Lindsey I, Kireev, Dmitri B, Frye, Stephen V

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Abstract ND08: Discovery of FX-909, a first-in-class inverse agonist of the peroxisome proliferator-activated receptor gamma (PPARG) lineage transcription factor, to potentially tr... von Sims, Robert, Mertz, Jennifer A., Wilson, Jonathan E., Audia, James E., Williamson, Kaylyn E., Li, Yong, Kuljanin, Miljan, Motely, Will W., DeLaBarre, Byron, Bowden, Michaela, Stuckey, Jacob I.

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Discovery and Characterization of a Cellularly Potent Positive Allosteric Modulator of the Polycomb Repressive Complex 1 Chromodomain, CBX7 von Lamb, Kelsey N., Bsteh, Daniel, Dishman, Sarah N., Moussa, Hagar F., Fan, Huitao, Stuckey, Jacob I., Norris, Jacqueline L., Cholensky, Stephanie H., Li, Dongxu, Wang, Jingkui, Sagum, Cari, Stanton, Benjamin Z., Bedford, Mark T., Pearce, Kenneth H., Kenakin, Terry P., Kireev, Dmitri B., Wang, Gang Greg, James, Lindsey I., Bell, Oliver, Frye, Stephen V.

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Addendum: A cellular chemical probe targeting the chromodomains of Polycomb repressive complex 1 von Stuckey, Jacob I, Dickson, Bradley M, Cheng, Nancy, Liu, Yanli, Norris, Jacqueline L, Cholensky, Stephanie H, Tempel, Wolfram, Qin, Su, Huber, Katherine G, Sagum, Cari, Black, Karynne, Li, Fengling, Huang, Xi-Ping, Roth, Bryan L, Baughman, Brandi M, Senisterra, Guillermo, Pattenden, Samantha G, Vedadi, Masoud, Brown, Peter J, TBedford, Mark, Min, Jinrong, Arrowsmith, Cheryl H, James, Lindsey I, Frye, Stephen V

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PPARG inverse agonists and uses thereof von Wilson, Jonathan E, Stuckey, Jacob I, Audia, James E

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PPARG INVERSE AGONISTS AND USES THEREOF von Wilson, Jonathan E, Stuckey, Jacob I, Audia, James E

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PPARG 역 효능제 및 그의 용도 von WANG FEI, AUDIA JAMES E, WADE PETER, MARK E. SCOTT, HUANG YAOHUI, WANG XIAOYANG, WILSON JONATHAN E, STUCKEY JACOB I, ZHENG BO, LI RUNYAN, MICHAEL J. GEIER, CONG LIQING, DAI DANMEI

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MODULATORS OF METHYL MODIFYING ENZYMES, COMPOSITIONS AND USES THEREOF von Gehling, Victor, S, Stuckey, Jacob, I, Côté, Alexandre, Moine, Ludivine, Khanna, Avinash

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MODULATORS OF METHYL MODIFYING ENZYMES, COMPOSITIONS AND USES THEREOF von COTE Alexandre, STUCKEY Jacob I, KHANNA Avinash, GEHLING Victor S, MOINE Ludivine

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MODULATORS OF METHYL MODIFYING ENZYMES, COMPOSITIONS AND USES THEREOF von GEHLING, Victor S, MOINE, Ludivine, STUCKEY, Jacob I, CÔTÉ, Alexandre, KHANNA, Avinash

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MODULATORS OF METHYL MODIFYING ENZYMES, COMPOSITIONS AND USES THEREOF von MOINE, LUDIVINE, KHANNA, AVINASH, STUCKEY, JACOB, I, CÔTÉ, ALEXANDRE, GEHLING, VICTOR, S

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