Photoredox-catalyzed deuteration and tritiation of pharmaceutical compounds von Loh, Yong Yao, Nagao, Kazunori, Hoover, Andrew J., Hesk, David, Rivera, Nelo R., Colletti, Steven L., Davies, Ian W., MacMillan, David W. C.

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Cheminformatic analysis of natural product-based drugs and chemical probes von Stone, Samantha, Newman, David J, Colletti, Steven L, Tan, Derek S

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International Union of Basic and Clinical Pharmacology. LXXXII: Nomenclature and Classification of Hydroxy-carboxylic Acid Receptors (GPR81, GPR109A, and GPR109B) von Offermanns, Stefan, Colletti, Steven L, Lovenberg, Timothy W, Semple, Graeme, Wise, Alan, IJzerman, Adriaan P

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Discovery of platencin, a dual FabF and FabH inhibitor with in vivo antibiotic properties von Wang, Jun, Kodali, Srinivas, Lee, Sang Ho, Galgoci, Andrew, Painter, Ronald, Dorso, Karen, Racine, Fred, Motyl, Mary, Hernandez, Lorraine, Tinney, Elizabeth, Colletti, Steven L, Herath, Kithsiri, Cummings, Richard, Salazar, Oscar, González, Ignacio, Basilio, Angela, Vicente, Francisca, Genilloud, Olga, Pelaez, Fernando, Jayasuriya, Hiranthi, Young, Katherine, Cully, Doris F, Singh, Sheo B

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GPR40 reduces food intake and body weight through GLP-1 von Gorski, Judith N, Pachanski, Michele J, Mane, Joel, Plummer, Christopher W, Souza, Sarah, Thomas-Fowlkes, Brande S, Ogawa, Aimie M, Weinglass, Adam B, Di Salvo, Jerry, Cheewatrakoolpong, Boonlert, Howard, Andrew D, Colletti, Steven L, Trujillo, Maria E

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GPR40 partial agonists and AgoPAMs: Differentiating effects on glucose and hormonal secretions in the rodent von Pachanski, Michele J, Kirkland, Melissa E, Kosinski, Daniel T, Mane, Joel, Cheewatrakoolpong, Boonlert, Xue, Jiyan, Szeto, Daphne, Forrest, Gail, Miller, Corin, Bunzel, Michelle, Plummer, Christopher W, Chobanian, Harry R, Miller, Michael W, Souza, Sarah, Thomas-Fowlkes, Brande S, Ogawa, Aimie M, Weinglass, Adam B, Di Salvo, Jerry, Li, Xiaoyan, Feng, Yue, Tatosian, Daniel A, Howard, Andrew D, Colletti, Steven L, Trujillo, Maria E

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Chemoselective Peptide Modification via Photocatalytic Tryptophan β‑Position Conjugation von Yu, Younong, Zhang, Li-Kang, Buevich, Alexei V, Li, Guoqing, Tang, Haiqun, Vachal, Petr, Colletti, Steven L, Shi, Zhi-Cai

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Profiling and Application of Photoredox C(sp3)–C(sp2) Cross-Coupling in Medicinal Chemistry von Zhang, Rui, Li, Guoqing, Wismer, Michael, Vachal, Petr, Colletti, Steven L., Shi, Zhi-Cai

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Systematic chemical modifications of single stranded siRNAs significantly improved CTNNB1 mRNA silencing von Chang, Wonsuk, Pei, Yi, Guidry, Erin N., Zewge, Daniel, Parish, Craig A., Sherer, Edward C., DiMuzio, Jillian, Zhang, Hangchun, South, Victoria J., Strapps, Walter R., Sepp-Lorenzino, Laura, Colletti, Steven L., Stanton, Matthew G.

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Structure–Activity Relationship of Novel and Selective Biaryl-Chroman GPR40 AgoPAMs von Chen, Helen Y., Plummer, Christopher W., Xiao, Dong, Chobanian, Harry R., DeMong, Duane, Miller, Michael, Trujillo, Maria E., Kirkland, Melissa, Kosinski, Daniel, Mane, Joel, Pachanski, Michele, Cheewatrakoolpong, Boonlert, Di Salvo, Jerry, Thomas-Fowlkes, Brande, Souza, Sarah, Tatosian, Daniel A., Chen, Qing, Hafey, Michael J., Houle, Robert, Nolting, Andrew F., Orr, Robert, Ehrhart, Juliann, Weinglass, Adam B., Tschirret-Guth, Richard, Howard, Andrew D., Colletti, Steven L.

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Structural basis for the cooperative allosteric activation of the free fatty acid receptor GPR40 von Lu, Jun, Byrne, Noel, Wang, John, Bricogne, Gerard, Brown, Frank K, Chobanian, Harry R, Colletti, Steven L, Di Salvo, Jerry, Thomas-Fowlkes, Brande, Guo, Yan, Hall, Dawn L, Hadix, Jennifer, Hastings, Nicholas B, Hermes, Jeffrey D, Ho, Thu, Howard, Andrew D, Josien, Hubert, Kornienko, Maria, Lumb, Kevin J, Miller, Michael W, Patel, Sangita B, Pio, Barbara, Plummer, Christopher W, Sherborne, Bradley S, Sheth, Payal, Souza, Sarah, Tummala, Srivanya, Vonrhein, Clemens, Webb, Maria, Allen, Samantha J, Johnston, Jennifer M, Weinglass, Adam B, Sharma, Sujata, Soisson, Stephen M

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Synthesis and biological evaluation of platensimycin analogs von SHEN, Hong C, DING, Fa-Xiang, TATA, James R, HAMMOND, Milton L, MACCOSS, Malcolm, COLLETTI, Steven L, SINGH, Sheo B, PARTHASARATHY, Gopalakrishnan, SOISSON, Stephen M, HA, Sookhee N, XUN CHEN, KODALI, Srinivas, JUN WANG, DORSO, Karen

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Discovery of spirocyclic secondary amine-derived tertiary ureas as highly potent, selective and bioavailable soluble epoxide hydrolase inhibitors von Shen, Hong C., Ding, Fa-Xiang, Wang, Siyi, Xu, Suoyu, Chen, Hsuan-shen, Tong, Xinchun, Tong, Vincent, Mitra, Kaushik, Kumar, Sanjeev, Zhang, Xiaoping, Chen, Yuli, Zhou, Gaochao, Pai, Lee-Yuh, Alonso-Galicia, Magdalena, Chen, Xiaoli, Zhang, Bei, Tata, James R., Berger, Joel P., Colletti, Steven L.

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Apicidin: A Novel Antiprotozoal Agent that Inhibits Parasite Histone Deacetylase von Darkin-Rattray, Sandra J., Gurnett, Anne M., Myers, Robert W., Dulski, Paula M., Crumley, Tami M., Allocco, John J., Cannova, Christine, Meinke, Peter T., Colletti, Steven L., Bednarek, Maria A., Singh, Sheo B., Goetz, Michael A., Dombrowski, Anne W., Polishook, Jon D., Schmatz, Dennis M.

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Medicinal Chemistry of siRNA Delivery von Stanton, Matthew G, Colletti, Steven L

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Palladium-Catalyzed Suzuki−Miyaura Coupling of Pyridyl-2-boronic Esters with Aryl Halides Using Highly Active and Air-Stable Phosphine Chloride and Oxide Ligands von Yang, David X, Colletti, Steven L, Wu, Kevin, Song, Maoying, Li, George Y, Shen, Hong C

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Discovery of the Development Candidate N-tert-Butyl Nodulisporamide: A Safe and Efficacious Once Monthly Oral Agent for the Control of Fleas and Ticks on Companion Animals von Meinke, Peter T, Colletti, Steven L, Fisher, Michael H, Wyvratt, Matthew J, Shih, Thomas L, Ayer, Michelle B, Li, Chunshi, Lim, Julie, Ok, Dong, Salva, Steve, Warmke, Lynn M, Zakson, Michelle, Michael, Bruce F, deMontigny, Pierre, Ostlind, Dan A, Fink, David, Drag, Marlene, Schmatz, Dennis M, Shoop, Wesley L

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The discovery of non-benzimidazole and brain-penetrant prolylcarboxypeptidase inhibitors von Graham, Thomas H., Shen, Hong C., Liu, Wensheng, Xiong, Yusheng, Verras, Andreas, Bleasby, Kelly, Bhatt, Urmi R., Chabin, Renee M., Chen, Dunlu, Chen, Qing, Garcia-Calvo, Margarita, Geissler, Wayne M., He, Huaibing, Lassman, Michael E., Shen, Zhu, Tong, Xinchun, Tung, Elaine C., Xie, Dan, Xu, Suoyu, Colletti, Steven L., Tata, James R., Hale, Jeffrey J., Pinto, Shirly, Shen, Dong-Ming

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Discovery of Biaryl Anthranilides as Full Agonists for the High Affinity Niacin Receptor von Shen, Hong C, Ding, Fa-Xiang, Luell, Silvi, Forrest, Michael J, Carballo-Jane, Ester, Wu, Kenneth K, Wu, Tsuei-Ju, Cheng, Kang, Wilsie, Larissa C, Krsmanovic, Mihajlo L, Taggart, Andrew K, Ren, Ning, Cai, Tian-Quan, Deng, Qiaolin, Chen, Qing, Wang, Junying, Wolff, Michael S, Tong, Xinchun, Holt, Tom G, Waters, M. Gerard, Hammond, Milton L, Tata, James R, Colletti, Steven L

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Design, synthesis and biological evaluation of indane derived GPR40 agoPAMs von Pio, Barbara, Chobanian, Harry R., Guo, Yan, Josien, Hubert, Hagmann, William K., Miller, Michael, Trujillo, Maria E., Kirkland, Melissa, Kosinski, Daniel, Mane, Joel, Pachanski, Michele, Cheewatrakoolpong, Boonlert, Ashley, Eric, Orr, Robert, Wright, Michael J., Bugianesi, Randal, Souza, Sarah, Zhang, Xiaoping, Di Salvo, Jerry, Weinglass, Adam B., Tschirret-Guth, Richard, Samuel, Koppara, Chen, Qing, Shang, Jackie, Lamca, James, Ehrhart, Juliann, Nargund, Ravi, Howard, Andrew D., Colletti, Steven L.

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