Development of an Enantioselective [3 + 2] Cycloaddition To Synthesize the Pyrrolidine Core of ABBV-3221 on Multikilogram Scale von Hartung, John, Greszler, Stephen N, Klix, Russell C, Kallemeyn, Jeffrey M

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Diastereoselective Synthesis of Pentasubstituted γ-Butyrolactones from Silyl Glyoxylates and Ketones through a Double Reformatsky Reaction von Greszler, Stephen N, Johnson, Jeffrey S

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Asymmetric Synthesis of Dihydroindanes by Convergent Alkoxide-Directed Metallacycle-Mediated Bond Formation von Greszler, Stephen N, Reichard, Holly A, Micalizio, Glenn C

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Catalytic Redox-Initiated Glycolate Aldol Additions of Silyl Glyoxylates von Greszler, Stephen N, Johnson, Jeffrey S

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Synthesis of Substituted Cyclopropanecarboxylates via Room Temperature Palladium-Catalyzed α‑Arylation of Reformatsky Reagents von Greszler, Stephen N, Halvorsen, Geoff T, Voight, Eric A

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Synthesis of the Cortistatin Pentacyclic Core by Alkoxide-Directed Metallacycle-Mediated Annulative Cross-Coupling von Aquino, Claudio, Greszler, Stephen N, Micalizio, Glenn C

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Lithioarene Cycliacylation and Pd-Catalyzed Aminoethylation/Cyclization to Access Electronically Diverse Saturated Isoquinoline Derivatives von Buchman, Marek, Farney, Elliot P, Greszler, Stephen N, Altenbach, Robert J, Gfesser, Gregory A, Voight, Eric A

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Discovery of Small Molecule Interleukin 17A Inhibitors with Novel Binding Mode and Stoichiometry: Optimization of DNA-Encoded Chemical Library Hits to In Vivo Active Compounds von Ramos, Ashley L., Goedken, Eric R., Frank, Kristine E., Argiriadi, Maria A., Bazzaz, Sana, Bian, Zhiguo, Brown, Jesse T. C., Centrella, Paolo A., Chen, Hui-Ju, Disch, Jeremy S., Donner, Pamela L., Duignan, David B., Gikunju, Diana, Greszler, Stephen N., Guié, Marie-Aude, Habeshian, Sevan, Hartl, Hajnalka E., Hein, Christopher D., Hutchins, Charles W., Jetson, Rachael, Keefe, Anthony D., Khan, Hasan, Li, Huan-Qiu, Olszewski, Allison, Ortiz Cardona, Benjamin J., Osuma, Augustine, Panchal, Sanjay C., Phelan, Ryan, Qiu, Wei, Shotwell, J. Brad, Shrestha, Anurupa, Srikumaran, Myron, Su, Zhi, Sun, Chaohong, Upadhyay, Anup K., Wood, Michael D., Wu, Haihong, Zhang, Ruijie, Zhang, Ying, Zhao, Gang, Zhu, Haizhong, Webster, Matthew P.

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Remote Stereoinduction in the Acylation of Fully Substituted Enolates: Tandem Reformatsky/Quaternary Claisen Condensations of Silyl Glyoxylates and β-Lactones von Greszler, Stephen N, Malinowski, Justin T, Johnson, Jeffrey S

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Synthesis of ABBV-168, a 2′-Bromouridine for the Treatment of Hepatitis C von Voight, Eric A, Brown, Brian S, Greszler, Stephen N, Halvorsen, Geoff T, Zhao, Gang, Kruger, Albert W, Hartung, John, Lukin, Kirill A, Martinez, Steven R, Moschetta, Eric G, Tudesco, Michael T, Ide, Nathan D

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Synthesis of A‑9758, an Inverse Agonist of Retinoic Acid-Related Orphan Receptor γt von Marvin, Christopher C., Greszler, Stephen N., Shelat, Bhadra H., Voight, Eric A.

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Silyl Glyoxylates. Conception and Realization of Flexible Conjunctive Reagents for Multicomponent Coupling von Boyce, Gregory R, Greszler, Stephen N, Johnson, Jeffrey S, Linghu, Xin, Malinowski, Justin T, Nicewicz, David A, Satterfield, Andrew D, Schmitt, Daniel C, Steward, Kimberly M

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ChemInform Abstract: Asymmetric Synthesis of Dihydroindans by Convergent Alkoxide-Directed Metallacycle-Mediated Bond Formation von Greszler, Stephen N., Reichard, Holly A., Micalizio, Glenn C.

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Diastereoselective Synthesis of Pentasubstituted γ‐Butyrolactones from Silyl Glyoxylates and Ketones through a Double Reformatsky Reaction von Greszler, Stephen N., Johnson, Jeffrey S.

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Heteroaryl substituted pyridines and methods of use von COWART, Marlon D, WANG, Xueqing, COTI, Ghjuvanni Petru Diunisu, KYM, Philip R, KELGTERMANS, Hans, BOGDAN, Andrew, ALTENBACH, Robert J, VAN DER PLAS, Steven Emiel, GRESZLER, Stephen N

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Heteroaryl substituted pyridines and methods of use von COWART, Marlon D, WANG, Xueqing, COTI, Ghjuvanni Petru Diunisu, KYM, Philip R, KELGTERMANS, Hans, BOGDAN, Andrew, ALTENBACH, Robert J, VAN DER PLAS, Steven Emiel, GRESZLER, Stephen N

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Heteroaryl substituted pyridines and methods of use von KELGTERMANS Hans, GRESZLER Stephen N, ALTENBACH Robert J, BOGDAN Andrew, COTI Ghjuvanni Petru Diunisu, KYM Philip R, VAN DER PLAS Steven Emiel, WANG Xueqing, COWART Marlon D

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Heteroaryl substituted pyridines and methods of use von KELGTERMANS Hans, GRESZLER Stephen N, ALTENBACH Robert J, BOGDAN Andrew, COTI Ghjuvanni Petru Diunisu, KYM Philip R, VAN DER PLAS Steven Emiel, WANG Xueqing, COWART Marlon D

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Heteroaryl substituted pyridines and methods of use von KELGTERMANS Hans, GRESZLER Stephen N, ALTENBACH Robert J, BOGDAN Andrew, COTI Ghjuvanni Petru Diunisu, KYM Philip R, VAN DER PLAS Steven Emiel, WANG Xueqing, COWART Marlon D

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SUBSTITUTED CHROMANES AND METHOD OF USE von GRESZLER, STEPHEN N, SEARLE, XENIA B, KYM, PHILIP R, VOIGHT, ERIC, KOENIG, JOHN R, WANG, XUEQING, ALTENBACH, ROBERT J, LIU, BO, YEUNG, MING C, BOGDAN, ANDREW

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