Preclinical selection of a novel poly(ADP-ribose) polymerase inhibitor for clinical trial von Thomas, Huw D, Calabrese, Christopher R, Batey, Michael A, Canan, Stacie, Hostomsky, Zdenek, Kyle, Suzanne, Maegley, Karen A, Newell, David R, Skalitzky, Donald, Wang, Lan-Zhen, Webber, Stephen E, Curtin, Nicola J

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Transcription inactivation through local refolding of the RNA polymerase structure von Belogurov, Georgiy A., Vassylyeva, Marina N., Sevostyanova, Anastasiya, Appleman, James R., Xiang, Alan X., Lira, Ricardo, Webber, Stephen E., Klyuyev, Sergiy, Nudler, Evgeny, Artsimovitch, Irina, Vassylyev, Dmitry G.

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Novel Poly(ADP-ribose) Polymerase-1 Inhibitor, AG14361, Restores Sensitivity to Temozolomide in Mismatch Repair-Deficient Cells von CURTIN, Nicola J, WANG, Lan-Zhen, NEWELL, David R, YIAKOUVAKI, Anthie, KYLE, Suzanne, ARRIS, Christine A, CANAN-KOCH, Stacie, WEBBER, Stephen E, DURKACZ, Barbara W, CALVERT, Hilary A, HOSTOMSKY, Zdenek

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Therapeutic Benefit of a Dissociated Glucocorticoid and the Relevance of In Vitro Separation of Transrepression from Transactivation Activity von Belvisi, Maria G, Wicks, Sharon L, Battram, Clifford H, Bottoms, Stephen E. W, Redford, Jane E, Woodman, Paul, Brown, Thomas J, Webber, Stephen E, Foster, Martyn L

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Structure-based Design of Pyridone–Aminal eFT508 Targeting Dysregulated Translation by Selective Mitogen-activated Protein Kinase Interacting Kinases 1 and 2 (MNK1/2) Inhibition von Reich, Siegfried H, Sprengeler, Paul A, Chiang, Gary G, Appleman, James R, Chen, Joan, Clarine, Jeff, Eam, Boreth, Ernst, Justin T, Han, Qing, Goel, Vikas K, Han, Edward Z. R, Huang, Vera, Hung, Ivy N. J, Jemison, Adrianna, Jessen, Katti A, Molter, Jolene, Murphy, Douglas, Neal, Melissa, Parker, Gregory S, Shaghafi, Michael, Sperry, Samuel, Staunton, Jocelyn, Stumpf, Craig R, Thompson, Peggy A, Tran, Chinh, Webber, Stephen E, Wegerski, Christopher J, Zheng, Hong, Webster, Kevin R

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Energy Transfer in Molecular Layer-by-Layer Films of Water-Soluble Perylene Diimides von Tang, Tingji, Herrmann, Andreas, Peneva, Kalina, Müllen, Klaus, Webber, Stephen E

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Anticancer chemosensitization and radiosensitization by the novel Poly(ADP-ribose) polymerase-1 inhibitor AG14361 von CALABRESE, Christopher R, ALMASSY, Robert, LI, Jianke, MAEGLEY, Karen, NEWELL, David R, NOTARIANNI, Elena, STRATFORD, Ian J, SKALITZKY, Donald, THOMAS, Huw D, WANG, Ian-Zhen, WEBBER, Stephen E, WILLIAMS, Kaye J, BARTON, Stephanie, CURTIN, Nicola J, BATEY, Michael A, CALVERT, A. Hilary, CANAN-KOCH, Stacie, DURKACZ, Barbara W, HOSTOMSKY, Zdenek, KUMPF, Robert A, KYLE, Suzanne

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Syntheses of novel myxopyronin B analogs as potential inhibitors of bacterial RNA polymerase von Lira, Ricardo, Xiang, Alan X., Doundoulakis, Thomas, Biller, William T., Agrios, Konstantinos A., Simonsen, Klaus B., Webber, Stephen E., Sisson, Wes, Aust, Robert M., Shah, Amit M., Showalter, Richard E., Banh, Virginia N., Steffy, Kevin R., Appleman, James R.

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Role of p38 MAP kinase in LPS‐induced airway inflammation in the rat von Haddad, El‐Bdaoui, Birrell, Mark, McCluskie, Kerryn, Ling, Andrea, Webber, Stephen E, Foster, Martyn L, Belvisi, Maria G

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Water-in-Carbon Dioxide Microemulsions with Methylated Branched Hydrocarbon Surfactants von Ryoo, Won, Webber, Stephen E, Johnston, Keith P

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Antibacterial activity in serum of the 3,5-diamino-piperidine translation inhibitors von Zhou, Yuefen, Chow, Chun, Murphy, Douglas E., Sun, Zhongxiang, Bertolini, Thomas, Froelich, Jamie M., Webber, Stephen E., Hermann, Thomas, Wall, Daniel

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Synthesis and SAR of 3,5-diamino-piperidine derivatives: Novel antibacterial translation inhibitors as aminoglycoside mimetics von Zhou, Yuefen, Gregor, Vlad E., Ayida, Benjamin K., Winters, Geoffrey C., Sun, Zhongxiang, Murphy, Douglas, Haley, Greg, Bailey, Dwight, Froelich, Jamie M., Fish, Sarah, Webber, Stephen E., Hermann, Thomas, Wall, Daniel

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Water-in-carbon dioxide emulsions stabilized with hydrophobic silica particles von Adkins, Stephanie S, Gohil, Dhiren, Dickson, Jasper L, Webber, Stephen E, Johnston, Keith P

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A Simple and Practical Synthesis of 2-Aminoimidazoles von Little, Thomas L, Webber, Stephen E

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Molecular Layer-by-Layer Self-Assembly of Water-Soluble Perylene Diimides through π−π and Electrostatic Interactions von Tang, Tingji, Qu, Jiangqiang, Müllen, Klaus, Webber, Stephen E

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Mediator involvement in antigen‐induced bronchospasm and microvascular leakage in the airways of ovalbumin sensitized Brown Norway rats von Hele, Dave J, Birrell, Mark A, Webber, Stephen E, Foster, Martyn L, Belvisi, Maria G

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Tricyclic Benzimidazoles as Potent Poly(ADP-ribose) Polymerase-1 Inhibitors von Skalitzky, Donald J, Marakovits, Joseph T, Maegley, Karen A, Ekker, Anne, Yu, Xiao-Hong, Hostomsky, Zdenek, Webber, Stephen E, Eastman, Brian W, Almassy, Robert, Li, Jianke, Curtin, Nicola J, Newell, David R, Calvert, A. Hilary, Griffin, Roger J, Golding, Bernard T

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Photophysics of Water Soluble Perylene Diimides in Surfactant Solutions von Tang, Tingji, Peneva, Kalina, Müllen, Klaus, Webber, Stephen E

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Abstract 582: Selection of a novel toll-like receptor 7 (TLR7) agonist PRX034 for immunotherapy of cancer von Appleman, James Richard, Webber, Stephen E.

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Discovery of tricyclic 5,6-dihydro-1H-pyridin-2-ones as novel, potent, and orally bioavailable inhibitors of HCV NS5B polymerase von RUEBSAM, Frank, MURPHY, Douglas E, BLAZEL, Julie K, SUN HEE KIM, YUEFEN ZHOU, QING HAN, KISSINGER, Charles R, WEBBER, Stephen E, SHOWALTER, Richard E, SHAH, Amit M, TSAN, Mei, PATEL, Rupal A, TRAN, Chinh V, THOMPSON, Peggy A, LEBRUN, Laurie A, HOU, Huiying J, KAMRAN, Ruhi, SERGEEVA, Maria V, BARTKOWSKI, Darian M, NOLAN, Thomas G, NORRIS, Daniel A, KHANDURINA, Julia, BROOKS, Jennifer, LI, Lian-Sheng, OKAMOTO, Ellen, KIRKOVSKY, Leo, JINGJING ZHAO, DRAGOVICH, Peter S, MCGUIRE, Helen M, XIANG, Alan X, ZHONGXIANG SUN, AYIDA, Benjamin K

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