A practical asymmetric synthesis of ( R)-fluoxetine and its major metabolite ( R)-norfluoxetine von Hilborn, James W, Lu, Zhi-Hui, Jurgens, Alex R, Fang, Q.Kevin, Byers, Paul, Wald, Stephen A, Senanayake, Chris H

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New General Sulfinylating Process for Asymmetric Synthesis of Enantiopure Sulfinates and Sulfoxides von Lu, Bruce Z, Jin, Fuqiang, Zhang, Yongda, Wu, Xinhe, Wald, Stephen A, Senanayake, Chris H

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A New Lithium Alkoxide Accelerated Diastereoselective Cyanation of Ketones von Wilkinson, H. Scott, Grover, Paul T, Vandenbossche, Charles P, Bakale, Roger P, Bhongle, Nandkumar N, Wald, Stephen A, Senanayake, Chris H

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Chiral Mandelic Acid Template Provides a Highly Practical Solution for (S)-Oxybutynin Synthesis von Grover, Paul T, Bhongle, Nandkumar N, Wald, Stephen A, Senanayake, Chris H

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Asymmetric synthesis of cetirizine dihydrochloride von Pflum, Derek A, Krishnamurthy, Dhileepkumar, Han, Zhengxu, Wald, Stephen A, Senanayake, Chris H

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Control of Diastereoselectivity by Solvent Effects in the Addition of Grignard Reagents to Enantiopure t-Butylsulfinimine:  Syntheses of the Stereoisomers of the Hydroxyl Derivativ... von Lu, Bruce Z, Senanayake, Chris, Li, Nansheng, Han, Zhengxu, Bakale, Roger P, Wald, Stephen A

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First Application of Tunable Alkyl or Aryl Sulfinamides to the Stereoselective Synthesis of a Chiral Amine:  Asymmetric Synthesis of (R)-Didesmethylsibutramine ((R)-DDMS) Using (R)... von Han, Zhengxu, Krishnamurthy, Dhileepkumar, Pflum, Derek, Grover, Paul, Wald, Stephen A, Senanayake, Chris H

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Rapid access to enantiopure bupropion and its major metabolite by stereospecific nucleophilic substitution on an α-ketotriflate von Fang, Qun K, Han, Zhengxu, Grover, Paul, Kessler, Donald, Senanayake, Chris H, Wald, Stephen A

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Remarkably selective palladium-catalyzed amination process: Rapid assembly of multiamino based structures von Hong, Yaping, Senanayake, Chris H., Xiang, Tingjian, Vandenbossche, Charles P., Tanoury, Gerald J., Bakale, Roger P., Wald, Stephen A.

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Chemoselective reductions of nitroarenes: bromoethanol-assisted phthalocyanatoiron/NaBH4 reductions von Wilkinson, H.Scott, Tanoury, Gerald J, Wald, Stephen A, Senanayake, Chris H

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Diethylanilineborane:  A Practical, Safe, and Consistent-Quality Borane Source for the Large-Scale Enantioselective Reduction of a Ketone Intermediate in the Synthesis of (R,R)-For... von Wilkinson, H. Scott, Tanoury, Gerald J, Wald, Stephen A, Senanayake, Chris H

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Palladium catalyzed amination of 2-chloro-1,3-azole derivatives: Mild entry to potent H1- antihistaminic norastemizole von Hong, Yaping, Tanoury, Gerald J., Wilkinson, H.Scott, Bakale, Roger P., Wald, Stephen A., Senanayake, Chris H.

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Large-Scale Synthesis of Enantio- and Diastereomerically Pure (R,R)-Formoterol von Hett, Robert, Fang, Qun K, Gao, Yun, Wald, Stephen A, Senanayake, Chris H

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A Large-Scale Synthesis of Enantiomerically Pure Cetirizine Dihydrochloride Using Preparative Chiral HPLC von Pflum, Derek A, Wilkinson, H. Scott, Tanoury, Gerald J, Kessler, Donald W, Kraus, Hali B, Senanayake, Chris H, Wald, Stephen A

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A large-scale asymmetric synthesis of ( S)-cyclohexylphenyl glycolic acid von Su, Xiping, Bhongle, Nandkumar N, Pflum, Derek, Butler, Hal, Wald, Stephen A, Bakale, Roger P, Senanayake, Chris H

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Taking Advantage of Polymorphism To Effect an Impurity Removal:  Development of a Thermodynamic Crystal Form of (R,R)-Formoterol Tartrate von Tanoury, Gerald J, Hett, Robert, Kessler, Donald W, Wald, Stephen A, Senanayake, Chris H

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Enantio- and diastereoselective synthesis of all four stereoisomers of formoterol von Hett, Robert, Fang, Qun Kevin, Gao, Yun, Hong, Yaping, Butler, Hal T, Nie, Xiaoyi, Wald, Stephen A

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Modulation of Catalyst Reactivity for the Chemoselective Hydrogenation of a Functionalized Nitroarene:  Preparation of a Key Intermediate in the Synthesis of (R,R)-Formoterol Tartr... von Wilkinson, H. Scott, Hett, Robert, Tanoury, Gerald J, Senanayake, Chris H, Wald, Stephen A

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First preparation of enantiomerically pure sibutramine and its major metabolite, and determination of their absolute configuration by single crystal X-ray analysis von Fang, Qun K, Senanayake, Chris H, Han, Zhengxu, Morency, Cynthia, Grover, Paul, Malone, Robert E, Bulter, Hal, Wald, Stephen A, Cameron, T.Stanley

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Rigid aminoalcohol backbone as a highly defined chiral template for the preparation of optically active tertiary α-hydroxyl acids von Senanayake, Chris H., Fang, Kevin, Grover, Paul, Bakale, Roger P., Vandenbossche, Charles P., Wald, Stephen A.

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