Bicyclo((aryl)methyl)benzamides as inhibitors of GlyT1 von Varnes, Jeffrey G., Xiong, Hui, Forst, Janet M., Holmquist, Christopher R., Ernst, Glen E., Frietze, William, Dembofsky, Bruce, Andisik, Don W., Palmer, William E., Hinkley, Lindsay, Steelman, Gary B., Wilkins, Deidre E., Tian, Gaochao, Jonak, Gerald, Potts, William M., Wang, Xia, Brugel, Todd A., Alhambra, Cristóbal, Wood, Michael W., Veale, Chris A., Albert, Jeffrey S.

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Potent Reversible Inhibitors of the Protein Tyrosine Phosphatase CD45 von Urbanek, Rebecca A, Suchard, Suzanne J, Steelman, Gary B, Knappenberger, Katharine S, Sygowski, Linda A, Veale, Chris A, Chapdelaine, Marc J

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Azepines and Piperidines with Dual Norepinephrine Dopamine Uptake Inhibition and Antidepressant Activity von Brown, Dean G, Bernstein, Peter R, Wu, Ye, Urbanek, Rebecca A, Becker, Christopher W, Throner, Scott R, Dembofsky, Bruce T, Steelman, Gary B, Lazor, Lois A, Scott, Clay W, Wood, Michael W, Wesolowski, Steven S, Nugiel, David A, Koch, Stephanie, Yu, Jian, Pivonka, Donald E, Li, Shuang, Thompson, Carol, Zacco, Anna, Elmore, Charles S, Schroeder, Patricia, Liu, JianWei, Hurley, Christopher A, Ward, Stuart, Hunt, Hazel J, Williams, Karen, McLaughlin, Joseph, Hoesch, Valerie, Sydserff, Simon, Maier, Donna, Aharony, David

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Pyridazinoquinolinetriones as NMDA Glycine-Site Antagonists with Oral Antinociceptive Activity in a Model of Neuropathic Pain von Bare, Thomas M, Brown, Dean G, Horchler, Carey L, Murphy, Megan, Urbanek, Rebecca A, Alford, Vernon, Barlaam, Christine, Dyroff, Martin C, Empfield, James B, Forst, Janet M, Herzog, Keith J, Keith, Richard A, Kirschner, Alan S, Lee, Chi-Ming C, Lewis, Joseph, McLaren, Frances M, Neilson, Kathy L, Steelman, Gary B, Trivedi, Shephali, Vacek, Edward P, Xiao, Wenhua

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Orally Active Trifluoromethyl Ketone Inhibitors of Human Leukocyte Elastase von Veale, Chris A, Bernstein, Peter R, Bohnert, Claudia M, Brown, Frederick J, Bryant, Craig, Damewood, James R, Earley, Roger, Feeney, Scott W, Edwards, Philip D, Gomes, Bruce, Hulsizer, James M, Kosmider, Ben J, Krell, Robert D, Moore, Gary, Salcedo, Theodora W, Shaw, Andrew, Silberstein, David S, Steelman, Gary B, Stein, Mark, Strimpler, Anne, Thomas, Roy M, Vacek, Edward P, Williams, Joseph C, Wolanin, Donald J, Woolson, Sheila

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Synthesis of 7-chloro-2,3-dihydro-2-[1-(pyridinyl)alkyl]-pyridazino[4,5-b]quinoline-1,4,10(5h )-triones as NMDA glycine-site antagonists von BROWN, Dean G, URBANEK, Rebecca A, XIAO, Wenhua, DYROFF, Martin C, LEE, Chi-Ming C, TRIVEDI, Shephali, NEILSON, Kathy L, KEITH, Richard A, BARE, Thomas M, MCLAREN, Frances M, HORCHLER, Carey L, MURPHY, Megan, STEELMAN, Gary B, EMPFIELD, James R, FORST, Janet M, HERZOG, Keith J

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The discovery of non-basic atrial natriuretic peptide clearance receptor antagonists. part 1 von Veale, Chris A, Alford, Vernon C, Aharony, David, Banville, Debra L, Bialecki, Russell A, Brown, Frederick J, Damewood, James R, Dantzman, Cathy L, Edwards, Philip D, Jacobs, Robert T, Mauger, Russell C, Murphy, Megan M, Palmer, Willam E, Pine, Kara K, Rumsey, William L, Garcia-Davenport, Laura E, Shaw, Andrew, Steelman, Gary B, Surian, Jean M, Vacek, Edward P

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Non-peptidic inhibitors of human leukocyte elastase. 4. Design, synthesis, and in vitro and in vivo activity of a series of .beta.-carbolinone-containing trifluoromethyl ketones von Veale, Chris A, Damewood, James R. Jr, Steelman, Gary B, Bryant, Craig, Gomes, Bruce, Williams, Joseph

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Efficient and scalable synthesis of thiazole fused benzazepine as a D2 partial agonist von Xiong, Hui, Wu, Ye, Lehr, Scott G., Blackwell, William, Steelman, Gary, Hulsizer, Jim, Urbanek, Rebecca A.

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Synthesis and SAR of aminothiazole fused benzazepines as selective dopamine D₂ partial agonists von Urbanek, Rebecca A, Xiong, Hui, Wu, Ye, Blackwell, William, Steelman, Gary, Rosamond, Jim, Wesolowski, Steven S, Campbell, James B, Zhang, Minli, Brockel, Becky, Widzowski, Daniel V

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BigBird: Big Data Storage and Analytics at Scale in Hybrid Cloud von Deochake, Saurabh, Channapattan, Vrushali, Steelman, Gary

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Efficient method for the synthesis of 1,4-disubstituted 5-carbomethoxypyrimidin-6-ones von Veale, Chris A, Steelman, Gary B, Chow, Margaret M

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BigBird: Big Data Storage and Analytics at Scale in Hybrid Cloud von Deochake, Saurabh, Channapattan, Vrushali, Steelman, Gary

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Nonpeptidic Inhibitors of Human Leukocyte Elastase. 2. Design, Synthesis, and in vitro Activity of a Series of 3-Amino-6-aryl-2-oxopyridyl Trifluoromethyl Ketones von Damewood, James R, Edwards, Philip D, Feeney, Scott, Gomes, Bruce C, Steelman, Gary B, Tuthill, Paul A, Williams, Joseph C, Warner, Peter, Woolson, Sheila A

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Nonpeptidic inhibitors of human leukocyte elastase. 5. Design, synthesis, and x-ray crystallography of a series of orally active 5-aminopyrimidin-6-one-containing trifluoromethyl k... von Veale, Chris A, Bernstein, Peter R, Bryant, Craig, Ceccarelli, Christopher, Damewood, James R. Jr, Earley, Roger, Feeney, Scott W, Gomes, Bruce, Kosmider, Ben J

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Discovery and Biological Activity of Orally Active Peptidyl Trifluoromethyl Ketone Inhibitors of Human Neutrophil Elastase von Edwards, Philip D, Andisik, Donald W, Bryant, Craig A, Ewing, Barbara, Gomes, Bruce, Lewis, Joseph J, Rakiewicz, Donna, Steelman, Gary, Strimpler, Ann, Trainor, Diane A, Tuthill, Paul A, Mauger, Russell C, Veale, Chris A, Wildonger, Richard A, Williams, Joseph C, Wolanin, Donald J, Zottola, Mark

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Design of Orally Active, Non-Peptidic Inhibitors of Human Leukocyte Elastase von Brown, Frederick J, Andisik, Donald W, Bernstein, Peter R, Bryant, Craig B, Ceccarelli, Chris, Damewood, James R. Jr, Edwards, Philip D, Earley, Roger A, Feeney, Scott

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Nonpeptidic inhibitors of human leukocyte elastase. 3. Design, synthesis, X-ray crystallographic analysis, and structure-activity relationships for a series of orally active 3-amin... von Bernstein, P R, Andisik, D, Bradley, P K, Bryant, C B, Ceccarelli, C, Damewood, Jr, J R, Earley, R, Edwards, P D, Feeney, S, Gomes, B C

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Nonpeptidic inhibitors of human leukocyte elastase. 2. Design, synthesis, and in vitro activity of a series of 3-amino-6-arylopyridin-2-one trifluoromethyl ketones von Damewood, Jr, J R, Edwards, P D, Feeney, S, Gomes, B C, Steelman, G B, Tuthill, P A, Williams, J C, Warner, P, Woolson, S A, Wolanin, D J

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Composto, composição, uso de um composto ou sal, e, métodos para tratar um distúrbio do sistema nervoso central e para preparar o composto oou sal von III, YE WU, JIAN WEI LIU, WILLIAM C. BLACKWELL, REBECCA URBANEK, GARY STEELMAN, JAMES HULSIZER, DAN WIDZOWSKI

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