Allostery at G protein-coupled receptor homo- and heteromers: uncharted pharmacological landscapes von Smith, Nicola J, Milligan, Graeme

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Drug Discovery Opportunities at the Endothelin B Receptor-Related Orphan G Protein-Coupled Receptors, GPR37 and GPR37L1 von Smith, Nicola J

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Allosteric modulation of heterodimeric G-protein-coupled receptors von Milligan, Graeme, Smith, Nicola J

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Identifying ligands at orphan GPCRs: current status using structure‐based approaches von Ngo, Tony, Kufareva, Irina, Coleman, James LJ, Graham, Robert M, Abagyan, Ruben, Smith, Nicola J

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Structural basis of promiscuous substrate transport by Organic Cation Transporter 1 von Zeng, Yi C., Sobti, Meghna, Quinn, Ada, Smith, Nicola J., Brown, Simon H. J., Vandenberg, Jamie I., Ryan, Renae M., O’Mara, Megan L., Stewart, Alastair G.

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Regulation of mitochondrial metabolism in murine skeletal muscle by the medium‐chain fatty acid receptor Gpr84 von Montgomery, Magdalene K., Osborne, Brenna, Brandon, Amanda E., O'Reilly, Liam, Fiveash, Corrine E., Brown, Simon H. J., Wilkins, Brendan P., Samsudeen, Azrah, Yu, Josephine, Devanapalli, Beena, Hertzog, Ashley, Tolun, Adviye A., Kavanagh, Tomas, Cooper, Antony A., Mitchell, Todd W., Biden, Trevor J., Smith, Nicola J., Cooney, Gregory J., Turner, Nigel

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Biogeochemical cycling in the anthropocene: Quantifying global environment-economy exchanges von Smith, Nicola J, McDonald, Garry W, Patterson, Murray G

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Critically evaluating sweet taste receptor expression and signaling through a molecular pharmacology lens von Smith, Nicola J., Grant, Jennifer N., Moon, Justin I., So, Sean S., Finch, Angela M.

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Deconvolution of complex G protein-coupled receptor signaling in live cells using dynamic mass redistribution measurements von Mohr, Klaus, Kostenis, Evi, Schröder, Ralf, Janssen, Nicole, Schmidt, Johannes, Kebig, Anna, Merten, Nicole, Hennen, Stephanie, Müller, Anke, Blättermann, Stefanie, Mohr-Andrä, Marion, Zahn, Sabine, Wenzel, Jörg, Smith, Nicola J, Gomeza, Jesús, Drewke, Christel, Milligan, Graeme

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Cryo-EM reveals distinct conformations of E. coli ATP synthase on exposure to ATP von Sobti, Meghna, Ishmukhametov, Robert, Bouwer, James C, Ayer, Anita, Suarna, Cacang, Smith, Nicola J, Christie, Mary, Stocker, Roland, Duncan, Thomas M, Stewart, Alastair G

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A Molecular Mechanism for Sequential Activation of a G Protein-Coupled Receptor von Grundmann, Manuel, Tikhonova, Irina G., Hudson, Brian D., Smith, Nicola J., Mohr, Klaus, Ulven, Trond, Milligan, Graeme, Kenakin, Terry, Kostenis, Evi

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Type 2 diabetes influences intraepithelial corneal nerve parameters and corneal stromal‐epithelial nerve penetration sites von Machet, Joshua, Park, Mijeong, Richardson, Alexander, Carnell, Michael, Mouat, Margaret A, Smith, Nicola J, Turner, Nigel, Cochran, Blake J, Rye, Kerry‐Anne, Di Girolamo, Nick

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Primary cilia, A‐kinase anchoring proteins and constitutive activity at the orphan G protein‐coupled receptor GPR161: A tale about a tail von Patel, Kinjal, Smith, Nicola J.

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The Action and Mode of Binding of Thiazolidinedione Ligands at Free Fatty Acid Receptor 1 von Smith, Nicola J., Stoddart, Leigh A., Devine, Nicola M., Jenkins, Laura, Milligan, Graeme

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Identification of novel species-selective agonists of the G-protein-coupled receptor GPR35 that promote recruitment of β-arrestin-2 and activate Gα13 von Jenkins, Laura, Brea, Jose, Smith, Nicola J, Hudson, Brian D, Reilly, Graeme, Bryant, Nia J, Castro, Marian, Loza, María-Isabel, Milligan, Graeme

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Shifting our perspective on orphan G protein-coupled receptors von Smith, Nicola J., Murray, Fiona

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Conserved Polar Residues in Transmembrane Domains V, VI, and VII of Free Fatty Acid Receptor 2 and Free Fatty Acid Receptor 3 Are Required for the Binding and Function of Short Cha... von Stoddart, Leigh A., Smith, Nicola J., Jenkins, Laura, Brown, Andrew J., Milligan, Graeme

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Metalloprotease cleavage of the N terminus of the orphan G protein-coupled receptor GPR37L1 reduces its constitutive activity von Coleman, James L J, Ngo, Tony, Schmidt, Johannes, Mrad, Nadine, Liew, Chu Kong, Jones, Nicole M, Graham, Robert M, Smith, Nicola J

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Retraction Note: Orphan receptor ligand discovery by pickpocketing pharmacological neighbors von Ngo, Tony, Ilatovskiy, Andrey V., Stewart, Alastair G., Coleman, James L. J., McRobb, Fiona M., Riek, R. Peter, Graham, Robert M., Abagyan, Ruben, Kufareva, Irina, Smith, Nicola J.

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Niclosamide blocks glucagon phosphorylation of Ser552 on β-catenin in primary rat hepatocytes via PKA signalling von Chowdhury, Md Kamrul H, Wu, Lindsay E, Coleman, James L J, Smith, Nicola J, Morris, Margaret J, Shepherd, Peter R, Smith, Greg C

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