Enantioselective Organocatalytic Construction of Pyrroloindolines by a Cascade Addition-Cyclization Strategy: Synthesis of (-)-Flustramine B von Austin, Joel F., Kim, Sung-Gon, Sinz, Christopher J., Xiao, Wen-Jing, David W. C. Mac Millan, Halpern, Jack

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Selective N7 Alkylation of 7-Azaindazoles von Lei, Zhiyu, Bao, Jianming, Cheng, Chen, Yu, Wensheng, Hu, Bin, Jin, Weichen, Jabri, Salman, Yang, Song, Zhao, Lianyun, Sinz, Christopher J, Duffy, Joseph L

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Seven transmembrane G protein-coupled receptor repertoire of gastric ghrelin cells von Engelstoft, Maja S, Park, Won-mee, Sakata, Ichiro, Kristensen, Line V, Husted, Anna Sofie, Osborne-Lawrence, Sherri, Piper, Paul K, Walker, Angela K, Pedersen, Maria H, Nøhr, Mark K, Pan, Jie, Sinz, Christopher J, Carrington, Paul E, Akiyama, Taro E, Jones, Robert M, Tang, Cong, Ahmed, Kashan, Offermanns, Stefan, Egerod, Kristoffer L, Zigman, Jeffrey M, Schwartz, Thue W

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Total synthesis of diazonamide A von Knowles, Robert R, Carpenter, Joseph, Blakey, Simon B, Kayano, Akio, Mangion, Ian K, Sinz, Christopher J, Macmillan, David W C

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The Direct and Enantioselective Organocatalytic α-Oxidation of Aldehydes von Brown, Sean P, Brochu, Michael P, Sinz, Christopher J, MacMillan, David W. C

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Modeling a Crowdsourced Definition of Molecular Complexity von Sheridan, Robert P, Zorn, Nicolas, Sherer, Edward C, Campeau, Louis-Charles, Chang, Charlie (Zhenyu), Cumming, Jared, Maddess, Matthew L, Nantermet, Philippe G, Sinz, Christopher J, O’Shea, Paul D

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Discovery of benzofuran propanoic acid GPR120 agonists: From uHTS hit to mechanism-based pharmacodynamic effects von Lombardo, Matthew, Bender, Kate, London, Clare, Plotkin, Michael A., Kirkland, Melissa, Mane, Joel, Pachanski, Michele, Geissler, Wayne, Cummings, John, Habulihaz, Bahanu, Akiyama, Taro E., Di Salvo, Jerry, Madeira, Maria, Pols, Joanna, Powles, Mary Ann, Finley, Michael F., Johnson, Eric, Roussel, Thomas, Uebele, Victor N., Crespo, Alejandro, Leung, Dennis, Alleyne, Candice, Trusca, Dorina, Lei, Ying, Howard, Andrew D., Ujjainwalla, Feroze, Tata, James R., Sinz, Christopher J.

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Design, Synthesis, and Evaluation of Novel and Selective G‑protein Coupled Receptor 120 (GPR120) Spirocyclic Agonists von Cox, Jason M, Chu, Hong D, Chelliah, Mariappan V, Debenham, John S, Eagen, Keith, Lan, Ping, Lombardo, Matthew, London, Clare, Plotkin, Michael A, Shah, Unmesh, Sun, Zhongxiang, Vaccaro, Henry M, Venkatraman, Srikanth, Suzuki, Takao, Wang, Nengxue, Ashley, Eric R, Crespo, Alejandro, Madeira, Maria, Leung, Dennis H, Alleyne, Candice, Ogawa, Aimie M, Souza, Sarah, Thomas-Fowlkes, Brande, Di Salvo, Jerry, Weinglass, Adam, Kirkland, Melissa, Pachanski, Michele, Powles, Mary Ann, Tozzo, Effie, Akiyama, Taro E, Ujjainwalla, Feroze, Tata, James R, Sinz, Christopher J

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Discovery and development of benzo-[1,2,4]-triazolo-[1,4]-oxazepine GPR142 agonists for the treatment of diabetes von Wilson, Jonathan E., Kurukulasuriya, Ravi, Sinz, Christopher, Lombardo, Matthew, Bender, Kate, Parker, Dann, Sherer, Edward C., Costa, Melissa, Dingley, Karen, Li, Xiaofang, Mitelman, Stanley, Tong, Sharon, Bugianesi, Randal, Ehrhardt, Anka, Priest, Birgit, Ratliff, Kevin, Ujjainwalla, Feroze, Nargund, Ravi, Hagmann, William K., Edmondson, Scott

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Discovery of Orally Bioavailable and Liver-Targeted Hypoxia-Inducible Factor Prolyl Hydroxylase (HIF-PHD) Inhibitors for the Treatment of Anemia von Liu, Ping, Wang, Liping, DuBois, Byron G, Colandrea, Vincent J, Liu, Rongqiang, Cai, Jiaqiang, Du, Xiaoxing, Quan, Weiguo, Morris, William, Bai, Jianwu, Bishwokarma, Bimjhana, Cheng, Mangeng, Piesvaux, Jennifer, Ray, Kallol, Alpert, Carla, Chiu, Chi-Sung, Zielstorff, Mark, Metzger, Joseph M, Yang, Liming, Leung, Dennis, Alleyne, Candice, Vincent, Stella H, Pucci, Vincenzo, Li, Xiaofang, Crespo, Alejandro, Stickens, Dominique, Hale, Jeffrey J, Ujjainwalla, Feroze, Sinz, Christopher J

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Small molecule activation of lecithin cholesterol acyltransferase modulates lipoprotein metabolism in mice and hamsters von Chen, Zhu, Wang, Sheng-ping, Krsmanovic, Mihajlo L, Castro-Perez, Jose, Gagen, Karen, Mendoza, Vivienne, Rosa, Ray, Shah, Vinit, He, Timothy, Stout, Steve J, Geoghagen, Neil S, Lee, Sang H, McLaren, David G, Wang, Liangsu, Roddy, Thomas P, Plump, Andrew S, Hubbard, Brian K, Sinz, Christopher J, Johns, Douglas G

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Corrigendum to “Discovery of benzofuran propanoic acid GPR120 agonists: From uHTS hit to mechanism-based pharmacodynamic effects” [Bioorg. Med. Chem. Lett. 26 (2016) 5724–5728]... von Lombardo, Matthew, Bender, Kate, London, Clare, Plotkin, Michael A., Kirkland, Melissa, Mane, Joel, Pachanski, Michele, Geissler, Wayne, Cummings, John, Habulihaz, Bahanu, Akiyama, Taro E., Di Salvo, Jerry, Madeira, Maria, Pols, Joanna, Powles, Mary Ann, Finley, Michael F., Johnson, Eric, Roussel, Thomas, Uebele, Victor N., Crespo, Alejandro, Leung, Dennis, Alleyne, Candice, Trusca, Dorina, Lei, Ying, Howard, Andrew D., Ujjainwalla, Feroze, Tata, James R., Sinz, Christopher J.

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Discovery and Optimization of a Novel Triazole Series of GPR142 Agonists for the Treatment of Type 2 Diabetes von Guo, Liangqin, Parker, Dann L, Zang, Yi, Sweis, Ramzi F, Liu, Weiguo, Sherer, Edward C, Buist, Nicole, Terebetski, Jenna, Kelly, Terri, Bugianesi, Randal, Priest, Birgit T, Dingley, Karen H, Li, Xiaofang, Mitelman, Stan, Salituro, Gino, Trujillo, Maria E, Pachanski, Michele, Kirkland, Melissa, Powles, Mary Ann, Eiermann, George J, Feng, Yue, Shang, Jin, Howard, Andrew D, Ujjainwalla, Feroze, Sinz, Christopher J, Debenham, John S, Edmondson, Scott D, Nargund, Ravi P, Hagmann, William K, Li, Derun

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Total synthesis of the polyene macrolide dermostatin A von Sinz, Christopher J, Rychnovsky, Scott D

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Total Synthesis of Dermostatin A von Sinz, Christopher J., Rychnovsky, Scott D.

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MZ-301 Is a Small Molecule Inhibitor of APOL1 Pore Function That Attenuates Albuminuria in a Mouse Model of APOL1-Mediated Kidney Disease: FR-PO318 von Assimon, Victoria, Bronner, Sarah, Yu, Cecile, Zha, Weibin, Hoek, Maarten, Sinz, Christopher, Green, Eric, Morgans, David J.

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A Gpr120-selective agonist improves insulin resistance and chronic inflammation in obese mice von Oh, Da Young, Walenta, Evelyn, Akiyama, Taro E, Lagakos, William S, Lackey, Denise, Pessentheiner, Ariane R, Sasik, Roman, Hah, Nasun, Chi, Tyler J, Cox, Jason M, Powels, Mary Ann, Di Salvo, Jerry, Sinz, Christopher, Watkins, Steven M, Armando, Aaron M, Chung, Heekyung, Evans, Ronald M, Quehenberger, Oswald, McNelis, Joanne, Bogner-Strauss, Juliane G, Olefsky, Jerrold M

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Multimodal Imaging Reveals that Sustained Inhibition of HIF-Prolyl Hydroxylases Induces Opposing Effects on Right and Left Ventricular Function in Healthy Rats von Robinson, Gain, Zielstorff, Mark, Sevilla, Raquel, Vanko, Amy, Sinz, Christopher, Cicmil, Milenko, Zhang, Weisheng, Bettano, Kimberly

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Correction: Multimodal Imaging Reveals that Sustained Inhibition of HIF-Prolyl Hydroxylases Induces Opposing Effects on Right and Left Ventricular Function in Healthy Rats von Robinson, Gain, Zielstorff, Mark, Sevilla, Raquel, Vanko, Amy, Sinz, Christopher, Cicmil, Milenko, Zhang, Weisheng, Bettano, Kimberly

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Small Molecule Inhibition of APOL1 Reverses Albuminuria in a Chronic Mouse Model of APOL1-Mediated Kidney Disease: SA-PO788 von Assimon, Victoria, Bronner, Sarah, Yu, Cecile, Chan, Helen, Crasta, Sheela, Lee, Patrick S., Lin, Baiwei, Luo, Yunqi, Octaviani, Angela, Reid, Adam, Sanman, Laura, Shi, Licheng, Situ, Eva, Tep, Sam, Zhang, Birong, Beattie, David T., Sinz, Christopher, Hoek, Maarten, Bernstein, Harold S., Morgans, David J., Green, Eric

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