Preclinical Profile of the HIV-1 Maturation Inhibitor VH3739937 von McAuliffe, Brian, Falk, Paul, Chen, Jie, Chen, Yan, Sit, Sing-Yuen, Swidorski, Jacob, Hartz, Richard A, Xu, Li, Venables, Brian, Sin, Ny, Meanwell, Nicholas A, Regueiro-Ren, Alicia, Wensel, David, Hanumegowda, Umesh, Krystal, Mark

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Epoxomicin, a Potent and Selective Proteasome Inhibitor, Exhibits in vivo Antiinflammatory Activity von Meng, Lihao, Mohan, Royce, Benjamin H. B. Kwok, Elofsson, Mikael, Sin, Ny, Crews, Craig M.

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Silver Benzoate Facilitates the Copper-Catalyzed C–N Coupling of Iodoazoles with Aromatic Nitrogen Heterocycles von Lozano, Cedric, Ramirez, Cristian, Sin, Ny, Viart, Hélène M.-F, Prusiner, Stanley B, Paras, Nick A, Conrad, Jay

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The Anti-Angiogenic Agent Fumagillin Covalently Binds and Inhibits the Methionine Aminopeptidase, MetAP-2 von Sin, Ny, Meng, Lihao, Margaret Q. W. Wang, Wen, James J., Bornmann, William G., Crews, Craig M.

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Orally Active Fusion Inhibitor of Respiratory Syncytial Virus von Cianci, Christopher, Yu, Kuo-Long, Combrink, Keith, Sin, Ny, Pearce, Bradley, Wang, Alan, Civiello, Rita, Voss, Stacey, Luo, Guangxiang, Kadow, Kathy, Genovesi, Eugene V, Venables, Brian, Gulgeze, Hatice, Trehan, Ashok, James, Jennifer, Lamb, Lucinda, Medina, Ivette, Roach, Julia, Yang, Zheng, Zadjura, Lisa, Colonno, Richard, Clark, Junius, Meanwell, Nicholas, Krystal, Mark

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Ernst Ralf Hintz u. Scott E. Pincikowski: The End-Times in Medieval German Literature. Sin, Evil, and the Apocalypse, Rochester/NY: Camden House 2020, X, 292 S., 2 Abb. (Studies in German Literature, Linguistics, and Culture) von Bowden, Sarah

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Oral Efficacy of a Respiratory Syncytial Virus Inhibitor in Rodent Models of Infection von CIANCI, Christopher, GENOVESI, Eugene V, COMBRINK, Keith, ZHUFANG LI, COLONNO, Richard, MEANWELL, Nicholas, CLARK, Junius, KRYSTAL, Mark, LAMB, Lucinda, MEDINA, Ivette, ZHENG YANG, ZADJURA, Lisa, HYEKYUNG YANG, D'ARIENZO, Celia, NY SIN, YU, Kuo-Long

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Total synthesis of the-potent proteasome inhibitor epoxomicin: a useful tool for understanding proteasome biology von Sin, Ny, Kim, Kyung Bo, Elofsson, Mikael, Meng, Lihao, Auth, Hak, Kwok, Benjamin H.B., Crews, Craig M.

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Metal Artefact Reduction by Dual-energy Computed Tomography Using Monoenergetic Extrapolation: In-vitro Determination of Optimal Monoenergetic Level with Different Metallic Implant... von Chan, WCS, Tsang, JPK, Wong, WY, Chu, PY, To, VYK, Lee, CY, Yeung, TW, Leung, OC, Sin, NY, Li, OC, Yuen, MK

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Eponemycin exerts its antitumor effect through the inhibition of proteasome function von LIHAO MENG, KWOK, B. H. B, NY SIN, CREWS, C. M

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Identification and Characterization of BMS-955176, a Second-Generation HIV-1 Maturation Inhibitor with Improved Potency, Antiviral Spectrum, and Gag Polymorphic Coverage von Nowicka-Sans, Beata, Protack, Tricia, Lin, Zeyu, Li, Zhufang, Zhang, Sharon, Sun, Yongnian, Samanta, Himadri, Terry, Brian, Liu, Zheng, Chen, Yan, Sin, Ny, Sit, Sing-Yuen, Swidorski, Jacob J, Chen, Jie, Venables, Brian L, Healy, Matthew, Meanwell, Nicholas A, Cockett, Mark, Hanumegowda, Umesh, Regueiro-Ren, Alicia, Krystal, Mark, Dicker, Ira B

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The Discovery of GSK3640254, a Next-Generation Inhibitor of HIV‑1 Maturation von Regueiro-Ren, Alicia, Sit, Sing-Yuen, Chen, Yan, Chen, Jie, Swidorski, Jacob J., Liu, Zheng, Venables, Brian L., Sin, Ny, Hartz, Richard A., Protack, Tricia, Lin, Zeyu, Zhang, Sharon, Li, Zhufang, Wu, Dauh-Rurng, Li, Peng, Kempson, James, Hou, Xiaoping, Gupta, Anuradha, Rampulla, Richard, Mathur, Arvind, Park, Hyunsoo, Sarjeant, Amy, Benitex, Yulia, Rahematpura, Sandhya, Parker, Dawn, Phillips, Thomas, Haskell, Roy, Jenkins, Susan, Santone, Kenneth S., Cockett, Mark, Hanumegowda, Umesh, Dicker, Ira, Meanwell, Nicholas A., Krystal, Mark

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Design, Synthesis, and SAR of C‑3 Benzoic Acid, C‑17 Triterpenoid Derivatives. Identification of the HIV‑1 Maturation Inhibitor 4‑((1R,3aS,5aR,5bR,7aR,11aS,11bR,13aR,13bR)‑3a-((2-(... von Regueiro-Ren, Alicia, Swidorski, Jacob J., Liu, Zheng, Chen, Yan, Sin, Ny, Sit, Sing-Yuen, Chen, Jie, Venables, Brian L., Zhu, Juliang, Nowicka-Sans, Beata, Protack, Tricia, Lin, Zeyu, Terry, Brian, Samanta, Himadri, Zhang, Sharon, Li, Zhufang, Easter, John, Beno, Brett R., Arora, Vinod, Huang, Xiaohua S., Rahematpura, Sandhya, Parker, Dawn D., Haskell, Roy, Santone, Kenneth S., Cockett, Mark I., Krystal, Mark, Meanwell, Nicholas A., Jenkins, Susan, Hanumegowda, Umesh, Dicker, Ira B.

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Discovery and Early Clinical Evaluation of BMS-605339, a Potent and Orally Efficacious Tripeptidic Acylsulfonamide NS3 Protease Inhibitor for the Treatment of Hepatitis C Virus Inf... von Scola, Paul M., Wang, Alan Xiangdong, Good, Andrew C., Sun, Li-Qiang, Combrink, Keith D., Campbell, Jeffrey A., Chen, Jie, Tu, Yong, Sin, Ny, Venables, Brian L., Sit, Sing-Yuen, Chen, Yan, Cocuzza, Anthony, Bilder, Donna M., D’Andrea, Stanley, Zheng, Barbara, Hewawasam, Piyasena, Ding, Min, Thuring, Jan, Li, Jianqing, Hernandez, Dennis, Yu, Fei, Falk, Paul, Zhai, Guangzhi, Sheaffer, Amy K., Chen, Chaoqun, Lee, Min S., Barry, Diana, Knipe, Jay O., Li, Wenying, Han, Yong-Hae, Jenkins, Susan, Gesenberg, Christoph, Gao, Qi, Sinz, Michael W., Santone, Kenneth S., Zvyaga, Tatyana, Rajamani, Ramkumar, Klei, Herbert E., Colonno, Richard J., Grasela, Dennis M., Hughes, Eric, Chien, Caly, Adams, Stephen, Levesque, Paul C., Li, Danshi, Zhu, Jialong, Meanwell, Nicholas A., McPhee, Fiona

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Invention of VH-937, a Potent HIV‑1 Maturation Inhibitor with the Potential for Infrequent Oral Dosing in Humans von Sit, Sing-Yuen, Chen, Yan, Chen, Jie, Venables, Brian L., Swidorski, Jacob J., Xu, Li, Sin, Ny, Hartz, Richard A., Lin, Zeyu, Zhang, Sharon, Li, Zhufang, Wu, Dauh-Rurng, Li, Peng, Kempson, James, Hou, Xiaoping, Shanmugam, Yoganand, Parker, Dawn, Jenkins, Susan, Simmermacher, Jean, Falk, Paul, McAuliffe, Brian, Cockett, Mark, Hanumegowda, Umesh, Dicker, Ira, Krystal, Mark, Meanwell, Nicholas A., Regueiro-Ren, Alicia

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Proteasome inhibition by the natural products epoxomicin and dihydroeponemycin: Insights into specificity and potency von Kim, Kyung Bo, Myung, Jayhyuk, Sin, Ny, Crews, Craig M.

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The design, synthesis and structure-activity relationships associated with C28 amine-based betulinic acid derivatives as inhibitors of HIV-1 maturation von Chen, Yan, Sit, Sing-Yuen, Chen, Jie, Swidorski, Jacob J., Liu, Zheng, Sin, Ny, Venables, Brian L., Parker, Dawn D., Nowicka-Sans, Beata, Lin, Zeyu, Li, Zhufang, Terry, Brian J., Protack, Tricia, Rahematpura, Sandhya, Hanumegowda, Umesh, Jenkins, Susan, Krystal, Mark, Dicker, Ira D., Meanwell, Nicholas A., Regueiro-Ren, Alicia

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Inhibitors of HIV-1 maturation: Development of structure–activity relationship for C-28 amides based on C-3 benzoic acid-modified triterpenoids von Swidorski, Jacob J., Liu, Zheng, Sit, Sing-Yuen, Chen, Jie, Chen, Yan, Sin, Ny, Venables, Brian L., Parker, Dawn D., Nowicka-Sans, Beata, Terry, Brian J., Protack, Tricia, Rahematpura, Sandhya, Hanumegowda, Umesh, Jenkins, Susan, Krystal, Mark, Dicker, Ira B., Meanwell, Nicholas A., Regueiro-Ren, Alicia

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Synthesis of (2S,3S,8S,9S)-Adda from D-glucose von Sin, Ny, Kallmerten, James

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P3-P4 ureas and reverse carbamates as potent HCV NS3 protease inhibitors: Effective transposition of the P4 hydrogen bond donor von Venables, Brian L., Sin, Ny, Wang, Alan Xiangdong, Sun, Li-Qiang, Tu, Yong, Hernandez, Dennis, Sheaffer, Amy, Lee, Min, Dunaj, Cindy, Zhai, Guangzhi, Barry, Diana, Friborg, Jacques, Yu, Fei, Knipe, Jay, Sandquist, Jason, Falk, Paul, Parker, Dawn, Good, Andrew C., Rajamani, Ramkumar, McPhee, Fiona, Meanwell, Nicholas A., Scola, Paul M.

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