Rifamycins – Obstacles and opportunities von Aristoff, Paul A, Garcia, George A, Kirchhoff, Paul D, Hollis Showalter, H.D

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Design, synthesis and prostate cancer cell-based studies of analogs of the Rho/MKL1 transcriptional pathway inhibitor, CCG-1423 von Evelyn, Chris R., Bell, Jessica L., Ryu, Jenny G., Wade, Susan M., Kocab, Andrew, Harzdorf, Nicole L., Hollis Showalter, H.D., Neubig, Richard R., Larsen, Scott D.

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Synthesis and structure–activity relationships of 2-amino-3-carboxy-4-phenylthiophenes as novel atypical protein kinase C inhibitors von Titchenell, Paul M., Hollis Showalter, H.D., Pons, Jean-François, Barber, Alistair J., Jin, Yafei, Antonetti, David A.

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Enediol mimics as inhibitors of the d-arabinose 5-phosphate isomerase (KdsD) from Francisella tularensis von Yep, Alejandra, Sorenson, Roderick J., Wilson, Michael R., Hollis Showalter, H.D., Larsen, Scott D., Keller, Paul R., Woodard, Ronald W.

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A novel synthesis of N1-(substituted)-pyrimido[5,4-e]-1,2,4-triazine-5,7(1H,6H)-diones von Turbiak, Anjanette J., Showalter, H.D. Hollis

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Synthesis and structural–activity relationships of 3-hydroxyquinazoline-2,4-dione antibacterial agents von Tran, Tuan P., Ellsworth, Edmund L., Stier, Michael A., Domagala, John M., Hollis Showalter, H.D., Gracheck, Stephen J., Shapiro, Martin A., Joannides, Themis E., Singh, Rajeshwar

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Protein cross-linking as a novel mechanism of action of a ubiquitin-activating enzyme inhibitor with anti-tumor activity von Kapuria, Vaibhav, Peterson, Luke F., Showalter, H.D. Hollis, Kirchhoff, Paul D., Talpaz, Moshe, Donato, Nicholas J.

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A roadmap for drug discovery and its translation to small molecule agents in clinical development for tuberculosis treatment von Showalter, H.D. Hollis, Denny, William A

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Characterization of rifamycin‐resistant Mycobacterium tuberculosis RNA polymerases von Gill, Sumandeep Kaur, Showalter, H.D. Hollis, Garcia, George A.

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A short, concise synthesis of queuine von Brooks, Allen F., Garcia, George A., Showalter, H.D. Hollis

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Investigation of 3-aryl-pyrimido[5,4-e][1,2,4]triazine-5,7-diones as small molecule antagonists of β-catenin/TCF transcription von Zeller, Jörg, Turbiak, Anjanette J., Powelson, Ian A., Lee, Surin, Sun, Duxin, Showalter, H.D. Hollis, Fearon, Eric R.

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Investigating the prevalence of queuine in Escherichia coli RNA via incorporation of the tritium-labeled precursor, preQ1 von Brooks, Allen F., Vélez-Martínez, Carol S., Hollis Showalter, H.D., Garcia, George A.

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A novel synthesis of N 1-(substituted)-pyrimido[5,4- e]-1,2,4-triazine-5,7(1 H,6 H)-diones von Turbiak, Anjanette J., Showalter, H.D. Hollis

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A novel synthesis of 3-(substituted)pyrimido[4,5- c]pyridazine-5,7(1 H,6 H)-diones von Turbiak, Anjanette J., Kampf, Jeff W., Hollis Showalter, H.D.

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Investigating the prevalence of queuine in Escherichia coli RNA via incorporation of the tritium-labeled precursor, preQ(1) von Brooks, Allen F, Vélez-Martínez, Carol S, Showalter, H D Hollis, Garcia, George A

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Synthesis and structure–activity relationships of novel substituted 8-amino, 8-thio, and 1,8-pyrazole congeners of antitubercular rifamycin S and rifampin von Jin, Yafei, Gill, Sumandeep K., Kirchhoff, Paul D., Wan, Baojie, Franzblau, Scott G., Garcia, George A., Showalter, H.D. Hollis

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Structure–activity relationships of 3-aminoquinazolinediones, a new class of bacterial type-2 topoisomerase (DNA gyrase and topo IV) inhibitors von Tran, Tuan P., Ellsworth, Edmund L., Sanchez, Joseph P., Watson, Brian M., Stier, Michael A., Showalter, H.D. Hollis, Domagala, John M., Shapiro, Martin A., Joannides, E. Themis, Gracheck, Stephen J., Nguyen, Dai Q., Bird, Paul, Yip, Judy, Sharadendu, Anurag, Ha, Chan, Ramezani, Saeed, Wu, Xiujuan, Singh, Rajeshwar

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Research into selective biomarkers of erythrocyte exposure to organophosphorus compounds von Aminoff, David, Bochar, Daniel A., Fuller, Amelia A., Mapp, Anna K., Showalter, H.D. Hollis, Kirchhoff, Paul D.

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Synthesis and antibacterial activity of the C-7 side chain of 3-aminoquinazolinediones von Hutchings, Kim M., Tran, Tuan P., Ellsworth, Edmund L., Watson, Brian M., Sanchez, Joseph P., Hollis Showalter, H.D., Stier, Michael A., Shapiro, Martin, Themis Joannides, E., Huband, Michael, Nguyen, Dai Q., Maiti, Samarendra, Li, Tingsheng, Tailor, Jyoti, Thomas, George, Ha, Chan, Singh, Rajeshwar

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Wnt-Pathway Directed Compound Targets Blast Crisis and Chronic Phase CML Leukemia Stem Progenitors von Peterson, Luke F, Turbiak, Anjanette J, Giannola, Diane M, Donato, Nicholas, Showalter, Hollis H.D., Fearon, Eric R, Talpaz, Moshe

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