2,3-Dihydroxy-6-nitro-7-sulfamoyl-benzo(F)quinoxaline: A Neuroprotectant for Cerebral Ischemia von Sheardown, Malcolm J., Nielsen, Elsebet Ø., Hansen, Anker J., Jacobsen, Poul, Honoré, Tage

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ZK200775: A Phosphonate Quinoxalinedione AMPA Antagonist for Neuroprotection in Stroke and Trauma von Turski, Lechoslaw, Huth, Andreas, Sheardown, Malcolm, McDonald, Fiona, Neuhaus, Roland, Schneider, Herbert H., Dirnagl, Ulrich, Wiegand, Frank, Jacobsen, Poul, Ottow, Eckhard

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N-Substituted Adenosines as Novel Neuroprotective A1 Agonists with Diminished Hypotensive Effects von Knutsen, Lars J. S, Lau, Jesper, Petersen, Hans, Thomsen, Christian, Weis, Jan U, Shalmi, Michael, Judge, Martin E, Hansen, Anker Jon, Sheardown, Malcolm J

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Xanomeline, an M1/M4 preferring muscarinic cholinergic receptor agonist, produces antipsychotic-like activity in rats and mice von Shannon, Harlan E., Rasmussen, Kurt, Bymaster, Frank P., Hart, John C., Peters, Steven C., Swedberg, Michael D.B., Jeppesen, Lone, Sheardown, Malcolm J., Sauerberg, Per, Fink-Jensen, Anders

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Novel functional M1 selective muscarinic agonists. Synthesis and structure-activity relationships of 3-(1,2,5-thiadiazolyl)-1,2,5,6-tetrahydro-1-methylpyridines von Sauerberg, Per, Olesen, Preben H, Nielsen, Susanne, Treppendahl, Svend, Sheardown, Malcolm J, Honore, Tage, Mitch, Charles H, Ward, John S, Pike, Andrew J

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Agonist-induced functional desensitization of recombinant human 5-HT2 receptors expressed in CHO-K1 cells von Porter, Richard H.P., Malcolm, Craig S., Allen, Nicola H., Lamb, Helen, Revell, Dean F., Sheardown, Malcolm J.

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The muscarinic receptor agonist BuTAC, a novel potential antipsychotic, does not impair learning and memory in mouse passive avoidance von Rasmussen, Thøger, Fink-Jensen, Anders, Sauerberg, Per, Swedberg, Michael D.B., Thomsen, Christian, Sheardown, Malcolm J., Jeppesen, Lone, Calligaro, David O., DeLapp, Neil W., Whitesitt, Celia, Ward, John S., Shannon, Harlan E., Bymaster, Frank P.

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Muscarinic receptor agonists decrease cocaine self-administration rates in drug-naive mice von Rasmussen, Thøger, Sauerberg, Per, Nielsen, Erik B, Swedberg, Michael D.B, Thomsen, Christian, Sheardown, Malcolm J, Jeppesen, Lone, Calligaro, David O, DeLapp, Neil W, Whitesitt, Celia, Ward, John S, Shannon, Harlan E, Bymaster, Frank P, Fink-Jensen, Anders

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Vulnerability to chronic subordination stress-induced depression-like disorders in adult 129SvEv male mice von Dadomo, Harold, Sanghez, Valentina, Di Cristo, Luisana, Lori, Andrea, Ceresini, Graziano, Malinge, Isabelle, Parmigiani, Stefano, Palanza, Paola, Sheardown, Malcolm, Bartolomucci, Alessandro

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Unexpected antipsychotic-like activity with the muscarinic receptor ligand (5 R,6 R)6-(3-propylthio-1,2,5-thiadiazol-4-yl)-1-azabicyclo[3.2.1]octane von Bymaster, Frank P, Shannon, Harlan E, Rasmussen, Kurt, Delapp, Neil W, Mitch, Charles H, Ward, John S, Calligaro, David O, Ludvigsen, Thomas S, Sheardown, Malcolm J, Olesen, Preben H, Swedberg, Michael D.B, Sauerberg, Per, Fink-Jensen, Anders

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The triggering of spreading depression in the chick retina by nicotinic receptor agonists von Sheardown, Malcolm J

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Unexpected neuroprotection observed with the adenosine A2A receptor agonist CGS 21680 von Sheardown, Malcolm J., Knutsen, Lars J.S.

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Muscarinic Agonists with Antipsychotic-like Activity:  Structure−Activity Relationships of 1,2,5-Thiadiazole Analogues with Functional Dopamine Antagonist Activity von Sauerberg, Per, Jeppesen, Lone, Olesen, Preben H, Rasmussen, Thøger, Swedberg, Michael D. B, Sheardown, Malcolm J, Fink-Jensen, Anders, Thomsen, Christian, Thøgersen, Henning, Rimvall, Karin, Ward, John S, Calligaro, David O, DeLapp, Neil W, Bymaster, Frank P, Shannon, Harlan E

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1,2,5-Thiadiazole Analogues of Aceclidine as Potent m1 Muscarinic Agonists von Ward, John S, Merritt, Leander, Calligaro, David O, Bymaster, Franklin P, Shannon, Harlan E, Mitch, Charles H, Whitesitt, Celia, Brunsting, David, Sheardown, Malcolm J, Olesen, Preben H, Swedberg, Michael D. B, Jeppesen, Lone, Sauerberg, Per

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The suitability of 129SvEv mice for studying depressive-like behaviour: Both males and females develop learned helplessness von Chourbaji, Sabine, Pfeiffer, Natascha, Dormann, Christof, Brandwein, Christiane, Fradley, Rosa, Sheardown, Malcolm, Gass, P.

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Metabotropic glutamate receptor agonists reduce epileptiform activity in the rat cortex von Sheardown, Malcolm J

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Muscarinic agonists exhibit functional dopamine antagonism in unilaterally 6-OHDA lesioned rats von Fink-Jensen, Anders, Kristensen, Peter, Shannon, Harlan E, Calligaro, David O, Delapp, Neil W, Whitesitt, Cilia, Ward, John S, Thomsen, Christian, Rasmusseen, Thøger, Sheardown, Malcolm J, Jeppesen, Lone, Sauerberg, Per, Bymaster, Frank P

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Modulation of γ-aminobutyric acid responses in the rat optic nerve von Empson, Ruth M, Sheardown, Malcolm J, Newberry, Nigel R

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Chlormethiazole inhibits epileptiform activity by potentiating GABAA receptor function von EMPSON, Ruth M, GEE, Veronica J, SHEARDOWN, Malcolm J, NEWBERRY, Nigel R

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1-(1,2,5-Thiadiazol-4-yl)-4-azatricyclo[2.2.1.02,6]heptanes as New Potent Muscarinic M1 Agonists:  Structure−Activity Relationship for 3-Aryl-2-propyn-1-yloxy and 3-Aryl-2-propyn-1... von Jeppesen, Lone, Olesen, Preben H, Hansen, Lena, Sheardown, Malcolm J, Thomsen, Christian, Rasmussen, Thøger, Jensen, Anders Fink, Christensen, Michael S, Rimvall, Karin, Ward, John S, Whitesitt, Celia, Calligaro, David O, Bymaster, Frank P, Delapp, Neil W, Felder, Christian C, Shannon, Harlan E, Sauerberg, Per

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