Structural understanding of non-nucleoside inhibition in an elongating herpesvirus polymerase von Hayes, Robert P., Heo, Mee Ra, Mason, Mark, Reid, John, Burlein, Christine, Armacost, Kira A., Tellers, David M., Raheem, Izzat, Shaw, Anthony W., Murray, Edward, McKenna, Philip M., Abeywickrema, Pravien, Sharma, Sujata, Soisson, Stephen M., Klein, Daniel

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Potent, Orally Bioavailable Calcitonin Gene-Related Peptide Receptor Antagonists for the Treatment of Migraine:  Discovery of N-[(3R,6S)-6-(2,3-Difluorophenyl)-2-oxo-1- (2,2,2-trif... von Paone, Daniel V, Shaw, Anthony W, Nguyen, Diem N, Burgey, Christopher S, Deng, James Z, Kane, Stefanie A, Koblan, Kenneth S, Salvatore, Christopher A, Mosser, Scott D, Johnston, Victor K, Wong, Bradley K, Miller-Stein, Cynthia M, Hershey, James C, Graham, Samuel L, Vacca, Joseph P, Williams, Theresa M

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Cerastecin Inhibition of the Lipooligosaccharide Transporter MsbA to Combat Acinetobacter baumannii : From Screening Impurity to In Vivo Efficacy von Skudlarek, Jason W, Cooke, Andrew J, Mitchell, Helen J, Babaoglu, Kerim, Shaw, Anthony W, Tong, Ling, Nomland, Ashley B, Labroli, Marc, Sha, Deyou, Mulhearn, James J, Wu, Chengwei, Li, Sarah W, Beshore, Douglas C, Hughes, Jonathan M E, Jouffroy, Matthieu, Wang, Hao, Balibar, Carl J, Painter, Ronald E, Shen, Pamela, Lange, Henry S, Ishchenko, Andrii, Chen, Yun-Ting, Klein, Daniel J, Tracy, Rodger W, Miller, Randy R, Cabalu, Tamara D, Wu, Zhe, Leithead, Andrew, Scapin, Giovanna, Hruza, Alan W, Dzhekieva, Liudmila, Bukhtiyarova, Marina, Homsher, Michelle F, Xu, Min, Bahnck-Teets, Carolyn, McKenney, David, Buevich, Alexei V, Liu, Jian, Zhang, Li-Kang, Meng, Tao, Kelly, Terri, DiNunzio, Edward, Soisson, Stephen, Cheng, Robert K Y, Hennig, Michael, Raheem, Izzat, Walker, Scott S

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Invention of novel 3-aminopiperidin-2-ones as calcitonin gene-related peptide receptor antagonists von Staas, Donnette D., Bell, Ian M., Burgey, Christopher S., Deng, James Z., Gallicchio, Steven N., Lim, John J., Paone, Daniel V., Potteiger, Craig M., Shaw, Anthony W., Stevenson, Heather, Stump, Craig A., Blair Zartman, C., Moore, Eric L., Bruno, Joseph G., Mosser, Scott D., White, Rebecca B., Kane, Stefanie A., Salvatore, Christopher A., Graham, Samuel L., Williams, Theresa M., Selnick, Harold G., Fraley, Mark E.

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Identification of second-generation P2X3 antagonists for treatment of pain von Ginnetti, Anthony T., Paone, Daniel V., Stauffer, Shaun R., Potteiger, Craig M., Shaw, Anthony W., Deng, James, Mulhearn, James J., Nguyen, Diem N., Segerdell, Carolyn, Anquandah, Juliana, Calamari, Amy, Cheng, Gong, Leitl, Michael D., Liang, Annie, Moore, Eric, Panigel, Jacqueline, Urban, Mark, Wang, Jixin, Fillgrove, Kerry, Tang, Cuyue, Cook, Sean, Kane, Stefanie, Salvatore, Christopher A., Graham, Samuel L., Burgey, Christopher S.

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Discovery of an Anion-Dependent Farnesyltransferase Inhibitor from a Phenotypic Screen von Bukhtiyarova, Marina, Cook, Erica M, Hancock, Paula J, Hruza, Alan W, Shaw, Anthony W, Adam, Gregory C, Barnard, Richard J O, McKenna, Philip M, Holloway, M Katharine, Bell, Ian M, Carroll, Steve, Cornella-Taracido, Ivan, Cox, Christopher D, Kutchukian, Peter S, Powell, David A, Strickland, Corey, Trotter, B Wesley, Tudor, Matthew, Wolkenberg, Scott, Li, Jing, Tellers, David M

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Cerastecins inhibit membrane lipooligosaccharide transport in drug-resistant Acinetobacter baumannii von Wang, Hao, Ishchenko, Andrii, Skudlarek, Jason, Shen, Pamela, Dzhekieva, Liudmila, Painter, Ronald E., Chen, Yun-Ting, Bukhtiyarova, Marina, Leithead, Andrew, Tracy, Rodger, Babaoglu, Kerim, Bahnck-Teets, Carolyn, Buevich, Alexei, Cabalu, Tamara D., Labroli, Marc, Lange, Henry, Lei, Ying, Li, Wei, Liu, Jian, Mann, Paul A., Meng, Tao, Mitchell, Helen J., Mulhearn, James, Scapin, Giovanna, Sha, Deyou, Shaw, Anthony W., Si, Qian, Tong, Ling, Wu, Chengwei, Wu, Zhe, Xiao, Jing Chen, Xu, Min, Zhang, Li-Kang, McKenney, David, Miller, Randy R., Black, Todd A., Cooke, Andrew, Balibar, Carl J., Klein, Daniel J., Raheem, Izzat, Walker, Scott S.

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Synthesis of the (3R,6S)-3-Amino-6-(2,3-difluorophenyl)azepan-2-one of Telcagepant (MK-0974), a Calcitonin Gene-Related Peptide Receptor Antagonist for the Treatment of Migraine He... von Burgey, Christopher S, Paone, Daniel V, Shaw, Anthony W, Deng, James Z, Nguyen, Diem N, Potteiger, Craig M, Graham, Samuel L, Vacca, Joseph P, Williams, Theresa M

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Rapid HATU-Mediated Solution Phase siRNA Conjugation von Aaronson, Jeffrey G, Klein, Lee J, Momose, Aaron A, O’Brien, Ann M, Shaw, Anthony W, Tucker, Thomas J, Yuan, Yu, Tellers, David M

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Examining the binding properties of MK-0974: A CGRP receptor antagonist for the acute treatment of migraine von Moore, Eric L., Burgey, Christopher S., Paone, Daniel V., Shaw, Anthony W., Tang, Yui S., Kane, Stefanie A., Salvatore, Christopher A.

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Orally bioavailable imidazoazepanes as calcitonin gene-related peptide (CGRP) receptor antagonists: Discovery of MK-2918 von Paone, Daniel V., Nguyen, Diem N., Shaw, Anthony W., Burgey, Christopher S., Potteiger, Craig M., Deng, James Z., Mosser, Scott D., Salvatore, Christopher A., Yu, Sean, Roller, Shane, Kane, Stefanie A., Selnick, Harold G., Vacca, Joseph P., Williams, Theresa M.

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Asymmetric synthesis of α,α-diaryl and α-aryl-α-heteroaryl alkylamines by organometallic additions to N-tert- butanesulfinyl ketimines von Shaw, Anthony W, deSolms, S.Jane

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Caprolactams as potent CGRP receptor antagonists for the treatment of migraine von Shaw, Anthony W., Paone, Daniel V., Nguyen, Diem N., Stump, Craig A., Burgey, Christopher S., Mosser, Scott D., Salvatore, Christopher A., Rutledge, Ruth Z., Kane, Stefanie A., Koblan, Kenneth S., Graham, Samuel L., Vacca, Joeseph P., Williams, Theresa M.

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Diaryl ether inhibitors of farnesyl-protein transferase von MacTough, Suzanne C., deSolms, S.Jane, Shaw, Anthony W., Abrams, Marc T., Ciccarone, Terrence M., Davide, Joseph P., Hamilton, Kelly A., Hutchinson, John H., Koblan, Kenneth S., Kohl, Nancy E., Lobell, Robert B., Robinson, Ronald G., Graham, Samuel L.

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Dual Protein Farnesyltransferase−Geranylgeranyltransferase-I Inhibitors as Potential Cancer Chemotherapeutic Agents von deSolms, S. Jane, Ciccarone, Terrence M, MacTough, Suzanne C, Shaw, Anthony W, Buser, Carolyn A, Ellis-Hutchings, Michelle, Fernandes, Christine, Hamilton, Kelly A, Huber, Hans E, Kohl, Nancy E, Lobell, Robert B, Robinson, Ronald G, Tsou, Nancy N, Walsh, Eileen S, Graham, Samuel L, Beese, Lorena S, Taylor, Jeffrey S

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Calcitonin gene-related peptide (CGRP) receptor antagonists: Investigations of a pyridinone template von Nguyen, Diem N., Paone, Daniel V., Shaw, Anthony W., Burgey, Christopher S., Mosser, Scott D., Johnston, Victor, Salvatore, Christopher A., Leonard, Yvonne M., Miller-Stein, Cynthia M., Kane, Stefanie A., Koblan, Kenneth S., Vacca, Joseph P., Graham, Samuel L., Williams, Theresa M.

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Progress in imaging by α‐synuclein Positron Emission Tomography von Bennacef, Idriss, Zeng, Zhizhen, Miller, Patricia J, Riffel, Kerry, Purcell, Mona L, Haley, Hyking D, Meng, Xiangjun, Yuchuan, Wang, Roecker, Anthony J, Shaw, Anthony W, Stump, Craig A, Mitchell, Helen J, Tong, Ling V, Fawaz, Maria V, Drolet, Robert E, Ma, Lei M, Marcus, Jacob, Li, Wenping, Hostetler, Eric D.

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Synthesis of tri- and tetrasubstituted imidazoles von Paone, Daniel V., Shaw, Anthony W.

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Calcium hypochlorite-mediated oxidation of primary alcohols to methyl esters von McDonald, Chriss E., Nice, Lois E., Shaw, Anthony W., Nestor, Nestor B.

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Molecular and Cellular Pharmacology: Examining the binding properties of MK-0974: A CGRP receptor antagonist for the acute treatment of migraine von Moore, Eric L, Burgey, Christopher S, Paone, Daniel V, Shaw, Anthony W, Tang, Yui S, Kane, Stefanie A, Salvatore, Christopher A

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