Oxazolidine Synthesis by Complementary Stereospecific and Stereoconvergent Methods von Shaghafi, Michael B, Grote, Robin E, Jarvo, Elizabeth R

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Structure-based Design of Pyridone–Aminal eFT508 Targeting Dysregulated Translation by Selective Mitogen-activated Protein Kinase Interacting Kinases 1 and 2 (MNK1/2) Inhibition von Reich, Siegfried H, Sprengeler, Paul A, Chiang, Gary G, Appleman, James R, Chen, Joan, Clarine, Jeff, Eam, Boreth, Ernst, Justin T, Han, Qing, Goel, Vikas K, Han, Edward Z. R, Huang, Vera, Hung, Ivy N. J, Jemison, Adrianna, Jessen, Katti A, Molter, Jolene, Murphy, Douglas, Neal, Melissa, Parker, Gregory S, Shaghafi, Michael, Sperry, Samuel, Staunton, Jocelyn, Stumpf, Craig R, Thompson, Peggy A, Tran, Chinh, Webber, Stephen E, Wegerski, Christopher J, Zheng, Hong, Webster, Kevin R

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Constructing Saturated Guanidinum Heterocycles by Cycloaddition of N‑Amidinyliminium Ions with Indoles von Allred, Tyler K, Shaghafi, Michael B, Chen, Pan-Pan, Tran, Quan, Houk, K. N, Overman, Larry E

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The insulin secretory action of novel polycyclic guanidines: discovery through open innovation phenotypic screening, and exploration of structure-activity relationships von Shaghafi, Michael B, Barrett, David G, Willard, Francis S, Overman, Larry E

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Palladium-Catalyzed Conjugate Allylation Reactions of α,β-Unsaturated N-Acylpyrroles von Shaghafi, Michael B, Kohn, Benjamin L, Jarvo, Elizabeth R

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Quinolones as HCV NS5B polymerase inhibitors von Kumar, Dange V., Rai, Roopa, Brameld, Ken A., Somoza, John R., Rajagopalan, Ravi, Janc, James W., Xia, Yu M., Ton, Tony L., Shaghafi, Michael B., Hu, Huiyong, Lehoux, Isabelle, To, Nhat, Young, Wendy B., Green, Michael J.

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Abstract 5333: Combining chemoproteomics with machine learning identifies functionally active covalent fragments for hard-to-drug cancer drivers von Hermann, Johannes C., Everley, Robert, Marholz, Laura, Berberich, Matthew, Yang, Tzu-Yi, Chao, Yu-Hsin, Awol, Abduselam K., Shaghafi, Michael, Yoon, Han, Varma, Rohan, Stein, Reed, Krug, Karsten, Lachtara, Emily, Erlanson, Daniel, Varma, Chris, Webster, Kevin R.

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TARGETED AUTOPHAGY CONJUGATES AND METHODS von HERMANN, Johannes, SHAGHAFI, Michael B

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TARGETED AUTOPHAGY CONJUGATES AND METHODS von HERMANN, Johannes, SHAGHAFI, Michael B

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TARGETED AUTOPHAGY CONJUGATES AND METHODS von HERMANN, Johannes, SHAGHAFI, Michael B

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Discovery of novel hydroxy pyrazole based factor IXa inhibitor von Vijaykumar, Dange, Sprengeler, Paul A., Shaghafi, Michael, Spencer, Jeffrey R., Katz, Brad A., Yu, Christine, Rai, Roopa, Young, Wendy B., Schultz, Brian, Janc, James

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ChemInform Abstract: Oxazolidine Synthesis by Complementary Stereospecific and Stereoconvergent Methods von Shaghafi, Michael B., Grote, Robin E., Jarvo, Elizabeth R.

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TARGETED AUTOPHAGY CONJUGATES AND METHODS von HERMANN, Johannes, SHAGHAFI, Michael B

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MAGL INHIBITORS von GRICE, Cheryl A, BUZARD, Daniel J, SHAGHAFI, Michael B

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MAGL INHIBITORS von GRICE, Cheryl A, BUZARD, Daniel J, SHAGHAFI, Michael B

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MAGL inhibitors von Buzard, Daniel J, Shaghafi, Michael B, Grice, Cheryl A

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MAGL INHIBITORS von GRICE, Cheryl A, BUZARD, Daniel J, SHAGHAFI, Michael B

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Efforts toward oral bioavailability in factor VIIa inhibitors von Vijaykumar, Dange, Rai, Roopa, Shaghafi, Michael, Ton, Tony, Torkelson, Steve, Leahy, Ellen M., Riggs, Jennifer R., Hu, Huiyong, Sprengeler, Paul A., Shrader, William D., O’Bryan, Colin, Cabuslay, Ronnell, Sanford, Ellen, Gjerstadt, Erik, Liu, Liang, Sukbuntherng, Juthamas, Young, Wendy B.

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MAGL inhibitors von Buzard, Daniel J, Shaghafi, Michael B, Grice, Cheryl A

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MAGL INHIBITORS von GRICE, Cheryl A, BUZARD, Daniel J, SHAGHAFI, Michael B

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