Well-Defined Polymer-Paclitaxel Prodrugs by a Grafting-from-Drug Approach von Louage, Benoit, Nuhn, Lutz, Risseeuw, Martijn D. P., Vanparijs, Nane, De Coen, Ruben, Karalic, Izet, Van Calenbergh, Serge, De Geest, Bruno G.

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Cinnamaldehyde and cinnamaldehyde derivatives reduce virulence in Vibrio spp. by decreasing the DNA-binding activity of the quorum sensing response regulator LuxR von Brackman, Gilles, Defoirdt, Tom, Miyamoto, Carol, Bossier, Peter, Van Calenbergh, Serge, Nelis, Hans, Coenye, Tom

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Identification of a new tert -leucinate class synthetic cannabinoid in powder and “spice-like” herbal incenses: methyl 2-[[1-(5-fluoropentyl)indole-3-carbonyl]amino]-3,3-dimethyl-b... von Risseeuw, Martijn D.P, Blankaert, Peter, Coopman, Vera, Quekelberghe, Stijn Van, Calenbergh, Serge Van, Cordonnier, Jan

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4“‐O‐Alkylated α‐Galactosylceramide Analogues as iNKT‐Cell Antigens: Synthetic, Biological, and Structural Studies von Janssens, Jonas, Bitra, Aruna, Wang, Jing, Decruy, Tine, Venken, Koen, van der Eycken, Johan, Elewaut, Dirk, Zajonc, Dirk M., van Calenbergh, Serge

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Autoreactivity to Sulfatide by Human Invariant NKT Cells von Stax, Annelein M, Tuengel, Jessica, Girardi, Enrico, Kitano, Naoki, Allan, Lenka L, Liu, Victor, Zheng, Dongjun, Panenka, William J, Guillaume, Joren, Wong, Chi-Huey, van Calenbergh, Serge, Zajonc, Dirk M, van den Elzen, Peter

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Enhanced TCR footprint by a novel glycolipid increases NKT-dependent tumor protection von Aspeslagh, Sandrine, Nemčovič, Marek, Pauwels, Nora, Venken, Koen, Wang, Jing, Calenbergh, Serge Van, Zajonc, Dirk M, Elewaut, Dirk

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Synthesis of pyrrolidine-based hamamelitannin analogues as quorum sensing inhibitors in Staphylococcus aureus von Bouton, Jakob, Van Hecke, Kristof, Rasooly, Reuven, Van Calenbergh, Serge

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Galactosylsphingamides: new α-GalCer analogues to probe the F’-pocket of CD1d von Guillaume, Joren, Wang, Jing, Janssens, Jonas, Remesh, Soumya G., Risseeuw, Martijn D. P., Decruy, Tine, Froeyen, Mathy, Elewaut, Dirk, Zajonc, Dirk M., Calenbergh, Serge Van

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3D-printed wound dressings containing a fosmidomycin-derivative prevent Acinetobacter baumannii biofilm formation von van Charante, Frits, Martínez-Pérez, David, Guarch-Pérez, Clara, Courtens, Charlotte, Sass, Andrea, Choińska, Emilia, Idaszek, Joanna, Van Calenbergh, Serge, Riool, Martijn, Zaat, Sebastian A.J., Święszkowski, Wojciech, Coenye, Tom

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Design, Synthesis, and Biological Evaluation of Bivalent Ligands Targeting Dopamine D2‐Like Receptors and the μ‐Opioid Receptor von Qian, Mingcheng, Vasudevan, Lakshmi, Huysentruyt, Jelle, Risseeuw, Martijn D. P., Stove, Christophe, Vanderheyden, Patrick M. L., Van Craenenbroeck, Kathleen, Van Calenbergh, Serge

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RORγt inhibition selectively targets IL-17 producing iNKT and γδ-T cells enriched in Spondyloarthritis patients von Venken, Koen, Jacques, Peggy, Mortier, Céline, Labadia, Mark E., Decruy, Tine, Coudenys, Julie, Hoyt, Kathleen, Wayne, Anita L., Hughes, Robert, Turner, Michael, Van Gassen, Sofie, Martens, Liesbet, Smith, Dustin, Harcken, Christian, Wahle, Joseph, Wang, Chao-Ting, Verheugen, Eveline, Schryvers, Nadia, Varkas, Gaëlle, Cypers, Heleen, Wittoek, Ruth, Piette, Yves, Gyselbrecht, Lieve, Van Calenbergh, Serge, Van den Bosch, Filip, Saeys, Yvan, Nabozny, Gerald, Elewaut, Dirk

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A case of acute intoxication due to combined use of fentanyl and 3,4-dichloro-N-[2-(dimethylamino)cyclohexyl]-N-methylbenzamide (U-47700) von Coopman, Vera, Blanckaert, Peter, Van Parys, Geert, Van Calenbergh, Serge, Cordonnier, Jan

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Report on a novel emerging class of highly potent benzimidazole NPS opioids: Chemical and in vitro functional characterization of isotonitazene von Blanckaert, Peter, Cannaert, Annelies, Van Uytfanghe, Katleen, Hulpia, Fabian, Deconinck, Eric, Van Calenbergh, Serge, Stove, Christophe

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Combining tubercidin and cordycepin scaffolds results in highly active candidates to treat late-stage sleeping sickness von Hulpia, Fabian, Mabille, Dorien, Campagnaro, Gustavo D., Schumann, Gabriela, Maes, Louis, Roditi, Isabel, Hofer, Anders, de Koning, Harry P., Caljon, Guy, Van Calenbergh, Serge

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Ceramide‐Templated Macrolactams: Total Synthesis and Biological Evaluation of Macrocyclic α‐Galactosylceramide Analogues and their Aglycons von Janssens, Jonas, Van der Eycken, Johan, Van Calenbergh, Serge

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Host metabolites stimulate the bacterial proton motive force to enhance the activity of aminoglycoside antibiotics von Crabbé, Aurélie, Ostyn, Lisa, Staelens, Sorien, Rigauts, Charlotte, Risseeuw, Martijn, Dhaenens, Maarten, Daled, Simon, Van Acker, Heleen, Deforce, Dieter, Van Calenbergh, Serge, Coenye, Tom

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Regioselective Ring Opening of 1,3‐Dioxane‐Type Acetals in Carbohydrates von Janssens, Jonas, Risseeuw, Martijn D. P., Van der Eycken, Johan, Van Calenbergh, Serge

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Analytical characterization of “etonitazepyne,” a new pyrrolidinyl‐containing 2‐benzylbenzimidazole opioid sold online von Blanckaert, Peter, Balcaen, Margot, Vanhee, Céline, Risseeuw, Martijn, Canfyn, Michaël, Desmedt, Bart, Van Calenbergh, Serge, Deconinck, Eric

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Receptor-Mediated Targeting of Cathepsins in Professional Antigen Presenting Cells von Hillaert, Ulrik, Verdoes, Martijn, Florea, Bogdan I, Saragliadis, Anastasios, Habets, Kim L.L, Kuiper, Johan, Van Calenbergh, Serge, Ossendorp, Ferry, van der Marel, Gijsbert A, Driessen, Christoph, Overkleeft, Hermen S

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Hamamelitannin Analogues that Modulate Quorum Sensing as Potentiators of Antibiotics against Staphylococcus aureus von Vermote, Arno, Brackman, Gilles, Risseeuw, Martijn D. P., Vanhoutte, Bieke, Cos, Paul, Van Hecke, Kristof, Breyne, Koen, Meyer, Evelyne, Coenye, Tom, Van Calenbergh, Serge

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