Conformationally Constrained ortho-Anilino Diaryl Ureas: Discovery of 1‑(2-(1′-Neopentylspiro[indoline-3,4′-piperidine]-1-yl)phenyl)-3-(4-(trifluoromethoxy)phenyl)urea, a Potent, S... von Qiao, Jennifer X, Wang, Tammy C, Ruel, Réjean, Thibeault, Carl, L’Heureux, Alexandre, Schumacher, William A, Spronk, Steven A, Hiebert, Sheldon, Bouthillier, Gilles, Lloyd, John, Pi, Zulan, Schnur, Dora M, Abell, Lynn M, Hua, Ji, Price, Laura A, Liu, Eddie, Wu, Qimin, Steinbacher, Thomas E, Bostwick, Jeffrey S, Chang, Ming, Zheng, Joanna, Gao, Qi, Ma, Baoqing, McDonnell, Patricia A, Huang, Christine S, Rehfuss, Robert, Wexler, Ruth R, Lam, Patrick Y. S

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Discovery of Pyrrolidine-Containing GPR40 Agonists: Stereochemistry Effects a Change in Binding Mode von Jurica, Elizabeth A, Wu, Ximao, Williams, Kristin N, Hernandez, Andres S, Nirschl, David S, Rampulla, Richard A, Mathur, Arvind, Zhou, Min, Cao, Gary, Xie, Chunshan, Jacob, Biji, Cai, Hong, Wang, Tao, Murphy, Brian J, Liu, Heng, Xu, Carrie, Kunselman, Lori K, Hicks, Michael B, Sun, Qin, Schnur, Dora M, Sitkoff, Doree F, Dierks, Elizabeth A, Apedo, Atsu, Moore, Douglas B, Foster, Kimberly A, Cvijic, Mary Ellen, Panemangalore, Reshma, Flynn, Neil A, Maxwell, Brad D, Hong, Yang, Tian, Yuan, Wilkes, Jason J, Zinker, Bradley A, Whaley, Jean M, Barrish, Joel C, Robl, Jeffrey A, Ewing, William R, Ellsworth, Bruce A

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Are Target-Family-Privileged Substructures Truly Privileged? von Schnur, Dora M, Hermsmeier, Mark A, Tebben, Andrew J

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Characterization of a new class of selective nonsteroidal progesterone receptor agonists von Dong, Yu, Roberge, Jacques Y, Wang, Zhaoqing, Wang, Xiaodong, Tamasi, Joseph, Dell, Vanessa, Golla, Rajasree, Corte, James R, Liu, Yalei, Fang, Tianan, Anthony, Monique N, Schnur, Dora M, Agler, Michele L, Dickson, John K, Lawrence, R.Michael, Prack, Margaret M, Seethala, Ramakrishna, Feyen, Jean H.M

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Methods for Combinatorial and Parallel Library Design von Schnur, Dora M., Beno, Brett R., Tebben, Andrew J., Cavallaro, Cullen

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Discovery of 2-(Phenoxypyridine)-3-phenylureas as Small Molecule P2Y 1 Antagonists von Chao, Hannguang, Turdi, Huji, Herpin, Timothy F., Roberge, Jacques Y., Liu, Yalei, Schnur, Dora M., Poss, Michael A., Rehfuss, Robert, Hua, Ji, Wu, Qimin, Price, Laura A., Abell, Lynn M., Schumacher, William A., Bostwick, Jeffrey S., Steinbacher, Thomas E., Stewart, Anne B., Ogletree, Martin L., Huang, Christine S., Chang, Ming, Cacace, Angela M., Arcuri, Maredith J., Celani, Deborah, Wexler, Ruth R., Lawrence, R. Michael

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Conformationally Constrained ortho- Anilino Diaryl Ureas: Discovery of 1-(2-(1′-Neopentylspiro[indoline-3,4′-piperidine]-1-yl)phenyl)-3-(4-(trifluoromethoxy)phenyl)urea, a Potent,... von Qiao, Jennifer X., Wang, Tammy C., Ruel, Réjean, Thibeault, Carl, L’Heureux, Alexandre, Schumacher, William A., Spronk, Steven A., Hiebert, Sheldon, Bouthillier, Gilles, Lloyd, John, Pi, Zulan, Schnur, Dora M., Abell, Lynn M., Hua, Ji, Price, Laura A., Liu, Eddie, Wu, Qimin, Steinbacher, Thomas E., Bostwick, Jeffrey S., Chang, Ming, Zheng, Joanna, Gao, Qi, Ma, Baoqing, McDonnell, Patricia A., Huang, Christine S., Rehfuss, Robert, Wexler, Ruth R., Lam, Patrick Y. S.

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Discovery of 2‑(Phenoxypyridine)-3-phenylureas as Small Molecule P2Y1 Antagonists von Chao, Hannguang, Turdi, Huji, Herpin, Timothy F, Roberge, Jacques Y, Liu, Yalei, Schnur, Dora M, Poss, Michael A, Rehfuss, Robert, Hua, Ji, Wu, Qimin, Price, Laura A, Abell, Lynn M, Schumacher, William A, Bostwick, Jeffrey S, Steinbacher, Thomas E, Stewart, Anne B, Ogletree, Martin L, Huang, Christine S, Chang, Ming, Cacace, Angela M, Arcuri, Maredith J, Celani, Deborah, Wexler, Ruth R, Lawrence, R. Michael

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A molecular mechanics study of amide conformations von Schnur, Dora M, Yuh, Young H, Dalton, David R

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MM2 force field parameters for oximes von Schnur, Dora M, Dalton, David R

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Development of an internal searching algorithm for parameterization of the MM2/MM3 force fields von Schnur, Dora M., Grieshaber, Mark V., Bowen, J. Phillip

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Beyond Rhodopsin: G Protein-Coupled Receptor Structure and Modeling Incorporating the β2-adrenergic and Adenosine A2A Crystal Structures von Tebben, Andrew J., Schnur, Dora M.

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Trisubstituted heteroaromatic compounds as calcium sensing receptor modulators von Yang, Wu, Dickson, John K, Cooper, Christopher B, Dodd, Dharmpal S, Ruan, Zheming, Schnur, Dora M

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Trisubstituted heteroaromatic compounds as calcium sensing receptor modulators von COOPER CHRISTOPHER B, DODD DHARMPAL S, RUAN ZHEMING, DICKSON JOHN K, YANG WU, SCHNUR DORA M

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TRISUBSTITUTED HETEROAROMATIC COMPOUNDS AS CALCIUM SENSING RECEPTOR MODULATORS von COOPER, CHRISTOPHER, B, DICKSON, JOHN, K, DODD, DHARMPAL, S, SCHNUR, DORA, M, RUAN, ZHEMING, YANG, WU

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FÜR DIE BEHANDLUNG VON THROMBOTISCHEN LEIDEN GEEIGNETE HARNSTOFFANTAGONISTEN DES P2Y1- REZEPTORS von LAWRENCE, MICHAEL R, ROBERGE, JACQUES YVES, QIAO, JENNIFER X, LAM, PATRICK Y.S, THIBEAULT, CARL, CHAO, HANNGUANG J, RUEL, REJEAN, BOUTHILLIER, GILLES, TUERDI, HUJI, HERPIN, TIMOTHY, WANG, TAMMY C, SCHNUR, DORA M, LIU, YALEI, CLARK, CHARLES G, GUNGOR, TIMUR, L'HEUREUX, ALEXANDRE L, REHFUSS, ROBERT P

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UREA ANTAGONISTS OF P2Y1 RECEPTOR USEFUL IN THE TREATMENT OF THROMBOTIC CONDITIONS von LAWRENCE, R. MICHAEL, ROBERGE, JACQUES YVES, QIAO, JENNIFER X, LAM, PATRICK Y.S, THIBEAULT, CARL, CHAO, HANNGUANG J, RUEL, REJEAN, BOUTHILLIER, GILLES, TUERDI, HUJI, HERPIN, TIMOTHY, WANG, TAMMY C, SCHNUR, DORA M, LIU, YALEI, CLARK, CHARLES G, GUNGOR, TIMUR, L'HEUREUX, ALEXANDRE L, REHFUSS, ROBERT P

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Urea antagonists of P2Y von Chao, Hannguang J, Tuerdi, Huji, Herpin, Timothy F, Roberge, Jacques Y, Liu, Yalei, Lawrence, Michael R, Rehfuss, Robert P, Clark, Charles G, Qiao, Jennifer X, Gungor, Timur, Lam, Patrick Y. S, Wang, Tammy C, Ruel, Rejean, L'Heureux, Alexandre, Thibeault, Carl, Bouthillier, Gilles, Schnur, Dora M

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Urea antagonists of P2Y1receptor useful in the treatment of thrombotic conditions von BOUTHILLIER GILLES, LIU YALEI, HERPIN TIMOTHY F, GUNGOR TIMUR, WANG TAMMY C, ROBERGE JACQUES Y, THIBEAULT CARL, LAM PATRICK Y. S, RUEL REJEAN, CLARK CHARLES G, SCHNUR DORA M, L'HEUREUX ALEXANDRE, CHAO HANNGUANG J, TUERDI HUJI, REHFUSS ROBERT P, LAWRENCE MICHAEL R, QIAO JENNIFER X

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Trisubstituted heteroaromatic compounds as calcium sensing receptor modulators von COOPER CHRISTOPHER B, DODD DHARMPAL S, RUAN ZHEMING, DICKSON JOHN K, YANG WU, SCHNUR DORA M

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