Identification of Two Novel Drosophila melanogaster Histamine-gated Chloride Channel Subunits Expressed in the Eye von Zheng, Yingcong, Hirschberg, Birgit, Yuan, Jeffrey, Wang, Alice P., Hunt, David C., Ludmerer, Steven W., Schmatz, Dennis M., Cully, Doris F.

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Apicidin: A Novel Antiprotozoal Agent that Inhibits Parasite Histone Deacetylase von Darkin-Rattray, Sandra J., Gurnett, Anne M., Myers, Robert W., Dulski, Paula M., Crumley, Tami M., Allocco, John J., Cannova, Christine, Meinke, Peter T., Colletti, Steven L., Bednarek, Maria A., Singh, Sheo B., Goetz, Michael A., Dombrowski, Anne W., Polishook, Jon D., Schmatz, Dennis M.

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Discovery of the Development Candidate N-tert-Butyl Nodulisporamide: A Safe and Efficacious Once Monthly Oral Agent for the Control of Fleas and Ticks on Companion Animals von Meinke, Peter T, Colletti, Steven L, Fisher, Michael H, Wyvratt, Matthew J, Shih, Thomas L, Ayer, Michelle B, Li, Chunshi, Lim, Julie, Ok, Dong, Salva, Steve, Warmke, Lynn M, Zakson, Michelle, Michael, Bruce F, deMontigny, Pierre, Ostlind, Dan A, Fink, David, Drag, Marlene, Schmatz, Dennis M, Shoop, Wesley L

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Design and synthesis of potent, orally bioavailable dihydroquinazolinone inhibitors of p38 MAP kinase von Stelmach, John E., Liu, Luping, Patel, Sangita B., Pivnichny, James V., Scapin, Giovanna, Singh, Suresh, Hop, Cornelis E.C.A., Wang, Zhen, Strauss, John R., Cameron, Patricia M., Nichols, Elizabeth A., O'Keefe, Stephen J., O'Neill, Edward A., Schmatz, Dennis M., Schwartz, Cheryl D., Thompson, Chris M., Zaller, Dennis M., Doherty, James B.

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Synthesis and SAR studies of very potent imidazopyridine antiprotozoal agents von Biftu, Tesfaye, Feng, Dennis, Fisher, Michael, Liang, Gui-Bai, Qian, Xiaoxia, Scribner, Andrew, Dennis, Richard, Lee, Shuliang, Liberator, Paul A., Brown, Chris, Gurnett, Anne, Leavitt, Penny S., Thompson, Donald, Mathew, John, Misura, Andrew, Samaras, Samantha, Tamas, Tamas, Sina, Joseph F., McNulty, Kathleen A., McKnight, Crystal G., Schmatz, Dennis M., Wyvratt, Matthew

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Purification and molecular characterization of cGMP-dependent protein kinase from Apicomplexan parasites. A novel chemotherapeutic target von Gurnett, Anne M, Liberator, Paul A, Dulski, Paula M, Salowe, Scott P, Donald, Robert G K, Anderson, Jennifer W, Wiltsie, Judyann, Diaz, Carmen A, Harris, Georgiana, Chang, Ben, Darkin-Rattray, Sandra J, Nare, Bakela, Crumley, Tami, Blum, Penny Sue, Misura, Andrew S, Tamas, Tamas, Sardana, Mohinder K, Yuan, Jeffrey, Biftu, Tesfaye, Schmatz, Dennis M

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Structure and Chemistry of Apicidins, a Class of Novel Cyclic Tetrapeptides without a Terminal α-Keto Epoxide as Inhibitors of Histone Deacetylase with Potent Antiprotozoal Activit... von Singh, Sheo B., Zink, Deborah L., Liesch, Jerrold M., Mosley, Ralph T., Dombrowski, Anne W., Bills, Gerald F., Darkin-Rattray, Sandra J., Schmatz, Dennis M., Goetz, Michael A.

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The discovery of a potent and selective lethal factor inhibitor for adjunct therapy of anthrax infection von Xiong, Yusheng, Wiltsie, Judyann, Woods, Andrea, Guo, Jian, Pivnichny, James V., Tang, Wei, Bansal, Alka, Cummings, Richard T., Cunningham, Barry R., Friedlander, Arthur M., Douglas, Cameron M., Salowe, Scott P., Zaller, Dennis M., Scolnick, Edward M., Schmatz, Dennis M., Bartizal, Kenneth, Hermes, Jeffrey D., MacCoss, Malcolm, Chapman, Kevin T.

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Synthesis and SAR studies of potent imidazopyridine anticoccidial agents von Liang, Gui-Bai, Qian, Xiaoxia, Feng, Dennis, Fisher, Michael, Brown, Christine M., Gurnett, Anne, Leavitt, Penny Sue, Liberator, Paul A., Misura, Andrew S., Tamas, Tamas, Schmatz, Dennis M., Wyvratt, Matthew, Biftu, Tesfaye

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N-Alkyl-4-piperidinyl-2,3-diarylpyrrole derivatives with heterocyclic substitutions as potent and broad spectrum anticoccidial agents von Liang, Gui-Bai, Qian, Xiaoxia, Feng, Dennis, Fisher, Michael, Crumley, Tami, Darkin-Rattray, Sandra J., Dulski, Paula M., Gurnett, Anne, Leavitt, Penny Sue, Liberator, Paul A., Misura, Andrew S., Samaras, Samantha, Tamas, Tamas, Schmatz, Dennis M., Wyvratt, Matthew, Biftu, Tesfaye

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Synthesis and SAR of 2-(4-fluorophenyl)-3-pyrimidin-4-ylimidazo[1,2- a]pyridine derivatives as anticoccidial agents von Feng, Dennis, Fisher, Michael, Liang, Gui-Bai, Qian, Xiaoxia, Brown, Chris, Gurnett, Anne, Leavitt, Penny Sue, Liberator, Paul A., Mathew, John, Misura, Andrew, Samaras, Samantha, Tamas, Tamas, Schmatz, Dennis M., Wyvratt, Matthew, Biftu, Tesfaye

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SAR of 3,4-Dihydropyrido[3,2- d]pyrimidone p38 inhibitors von Liu, Luping, Stelmach, John E., Natarajan, Swaminathan R., Chen, Meng-Hsin, Singh, Suresh B., Schwartz, Cheryl D., Fitzgerald, Catherine E., O'Keefe, Stephen J., Zaller, Dennis M., Schmatz, Dennis M., Doherty, James B.

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Preparation and structure-activity relationships of simplified analogs of the antifungal agent cilofungin: a total synthesis approach von Zambias, Robert A, Hammond, Milton L, Heck, James V, Bartizal, Ken, Trainor, Charlotte, Abruzzo, George, Schmatz, Dennis M, Nollstadt, Karl M

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Hybrid-Designed Inhibitors of p38 MAP Kinase Utilizing N-Arylpyridazinones von Colletti, Steven L, Frie, Jessica L, Dixon, Elizabeth C, Singh, Suresh B, Choi, Bernard K, Scapin, Giovanna, Fitzgerald, Catherine E, Kumar, Sanjeev, Nichols, Elizabeth A, O'Keefe, Stephen J, O'Neill, Edward A, Porter, Gene, Samuel, Koppara, Schmatz, Dennis M, Schwartz, Cheryl D, Shoop, Wesley L, Thompson, Chris M, Thompson, James E, Wang, Ruixiu, Woods, Andrea, Zaller, Dennis M, Doherty, James B

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Synthesis of Apicidin-Derived Quinolone Derivatives:  Parasite-Selective Histone Deacetylase Inhibitors and Antiproliferative Agents von Meinke, Peter T, Colletti, Steven L, Doss, George, Myers, Robert W, Gurnett, Anne M, Dulski, Paula M, Darkin-Rattray, Sandra J, Allocco, John J, Galuska, Stefan, Schmatz, Dennis M, Wyvratt, Matthew J, Fisher, Michael H

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Synthesis and SAR Studies of diarylpyrrole anticoccidial agents von Qian, Xiaoxia, Liang, Gui-Bai, Feng, Dennis, Fisher, Michael, Crumley, Tami, Rattray, Sandra, Dulski, Paula M., Gurnett, Anne, Leavitt, Penny Sue, Liberator, Paul A., Misura, Andrew S., Samaras, Samantha, Tamas, Tamas, Schmatz, Dennis M., Wyvratt, Matthew, Biftu, Tesfaye

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Broad spectrum antiprotozoal agents that inhibit histone deacetylase: Structure-activity relationships of apicidin. Part 1 von COLLETTI, Steven L, MYERS, Robert W, CRUMLEY, Tami M, CANNOVA, Christine, SCHMATZ, Dennis M, WYVRATT, Matthew J, FISHER, Michael H, MEINKE, Peter T, DARKIN-RATTRAY, Sandra J, GURNETT, Anne M, DULSKI, Paula M, GALUSKA, Stefan, ALLOCCO, John J, AYER, Michelle B, CHUNSHI LI, LIM, Julie

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Potent 4-aminopiperidine based antimalarial agents von Brinner, Kristin M., Powles, Mary Ann, Schmatz, Dennis M., Ellman, Jonathan A.

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Structure, Histone Deacetylase, and Antiprotozoal Activities of Apicidins B and C, Congeners of Apicidin with Proline and Valine Substitutions von Singh, Sheo B, Zink, Deborah L, Liesch, Jerrold M, Dombrowski, Anne W, Darkin-Rattray, Sandra J, Schmatz, Dennis M, Goetz, Michael A

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Hydroxylated N-alkyl-4-piperidinyl-2,3-diarylpyrrole derivatives as potent broad-spectrum anticoccidial agents von Liang, Gui-Bai, Qian, Xiaoxia, Biftu, Tesfaye, Feng, Dennis, Fisher, Michael, Crumley, Tami, Darkin-Rattray, Sandra J., Dulski, Paula M., Gurnett, Anne, Leavitt, Penny Sue, Liberator, Paul A., Misura, Andrew S., Samaras, Samantha, Tamas, Tamas, Schmatz, Dennis M., Wyvratt, Matthew

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