Hydroxyl Groups in Synthetic and Natural-Product-Derived Therapeutics: A Perspective on a Common Functional Group von Cramer, Jonathan, Sager, Christoph P, Ernst, Beat

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Urinary Tract Infection: Which Conformation of the Bacterial Lectin FimH Is Therapeutically Relevant? von Mayer, Katharina, Eris, Deniz, Schwardt, Oliver, Sager, Christoph P, Rabbani, Said, Kleeb, Simon, Ernst, Beat

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Discovery of a Novel Orally Active, Selective LPA Receptor Type 1 Antagonist, 4‑(4-(2-Isopropylphenyl)-4-((2-methoxy-4-methylphenyl)carbamoyl)piperidin-1-yl)-4-oxobutanoic Acid, wi... von Lescop, Cyrille, Brotschi, Christine, Williams, Jodi T., Sager, Christoph P., Birker, Magdalena, Morrison, Keith, Froidevaux, Sylvie, Delahaye, Stéphane, Nayler, Oliver, Bolli, Martin H.

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Homodimer Architecture of QTRT2, the Noncatalytic Subunit of the Eukaryotic tRNA-Guanine Transglycosylase von Behrens, Christina, Biela, Inna, Petiot-Bécard, Stéphanie, Botzanowski, Thomas, Cianférani, Sarah, Sager, Christoph P, Klebe, Gerhard, Heine, Andreas, Reuter, Klaus

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Which Properties Allow Ligands to Open and Bind to the Transient Binding Pocket of Human Aldose Reductase? von Sandner, Anna, Ngo, Khang, Sager, Christoph P., Scheer, Frithjof, Daude, Michael, Diederich, Wibke E., Heine, Andreas, Klebe, Gerhard

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Homology modeling meets site-directed mutagenesis: An ideal combination to elucidate the topology of 17β-HSD2 von Sager, Christoph P., Weber, Susanne, Negri, Matthias, Banachowicz, Pauline, Möller, Gabriele, Adamski, Jerzy, Hartmann, Rolf W., Marchais-Oberwinkler, Sandrine

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KinITC—One Method Supports both Thermodynamic and Kinetic SARs as Exemplified on FimH Antagonists von Zihlmann, Pascal, Silbermann, Marleen, Sharpe, Timothy, Jiang, Xiaohua, Mühlethaler, Tobias, Jakob, Roman P., Rabbani, Said, Sager, Christoph P., Frei, Priska, Pang, Lijuan, Maier, Timm, Ernst, Beat

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Conformational Changes in Alkyl Chains Determine the Thermodynamic and Kinetic Binding Profiles of Carbonic Anhydrase Inhibitors von Glöckner, Steffen, Ngo, Khang, Sager, Christoph P, Hüfner-Wulsdorf, Tobias, Heine, Andreas, Klebe, Gerhard

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The price of flexibility - a case study on septanoses as pyranose mimetics von Sager, Christoph P, Fiege, Brigitte, Zihlmann, Pascal, Vannam, Raghu, Rabbani, Said, Jakob, Roman P, Preston, Roland C, Zalewski, Adam, Maier, Timm, Peczuh, Mark W, Ernst, Beat

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E-selectin ligand complexes adopt an extended high-affinity conformation von Preston, Roland C, Jakob, Roman P, Binder, Florian P C, Sager, Christoph P, Ernst, Beat, Maier, Timm

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LST-3TM12 is a member of the OATP1B family and a functional transporter von Malagnino, Vanessa, Hussner, Janine, Seibert, Isabell, Stolzenburg, Antje, Sager, Christoph P., Meyer zu Schwabedissen, Henriette E.

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What contributes to an effective mannose recognition domain? von Sager, Christoph P, Eriş, Deniz, Smieško, Martin, Hevey, Rachel, Ernst, Beat

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Improvement of Aglycone π‐Stacking Yields Nanomolar to Sub‐nanomolar FimH Antagonists von Schönemann, Wojciech, Cramer, Jonathan, Mühlethaler, Tobias, Fiege, Brigitte, Silbermann, Marleen, Rabbani, Said, Dätwyler, Philipp, Zihlmann, Pascal, Jakob, Roman P., Sager, Christoph P., Smieško, Martin, Schwardt, Oliver, Maier, Timm, Ernst, Beat

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Biochemical analyses and molecular modeling explain the functional loss of 17β-hydroxysteroid dehydrogenase 3 mutant G133R in three Tunisian patients with 46, XY Disorders of Sex D... von Engeli, Roger T., Rhouma, Bochra Ben, Sager, Christoph P., Tsachaki, Maria, Birk, Julia, Fakhfakh, Faiza, Keskes, Leila, Belguith, Neila, Odermatt, Alex

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Biochemical Analysis of Four Missense Mutations in the HSD17B3 Gene Associated With 46,XY Disorders of Sex Development in Egyptian Patients von Engeli, Roger T., Tsachaki, Maria, Hassan, Heba A., Sager, Christoph P., Essawi, Mona L., Gad, Yehia Z., Kamel, Alaa K., Mazen, Inas, Odermatt, Alex

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Drug Discovery Summit: 11th Swiss Course on Medicinal Chemistry von Frei, Priska, Navarra, Giulio, Sager, Christoph P., Silbermann, Marleen, Varga, Norbert, Wamhoff, Eike-Christian

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Drug discovery summit: 11(th) Swiss Course on Medicinal Chemistry von Frei, Priska, Navarra, Giulio, Sager, Christoph P, Silbermann, Marleen, Varga, Norbert, Wamhoff, Eike-Christian

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A survey of image labelling for computer vision applications von Sager, Christoph, Janiesch, Christian, Zschech, Patrick

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labelCloud: A Lightweight Labeling Tool for Domain-Agnostic 3D Object Detection in Point Clouds von Sager, Christoph, Zschech, Patrick, Kuhl, Niklas

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The price of flexibility - a case study on septanoses as pyranose mimeticsElectronic supplementary information (ESI) available. See DOI: 10.1039/c7sc04289b von Sager, Christoph P, Fiege, Brigitte, Zihlmann, Pascal, Vannam, Raghu, Rabbani, Said, Jakob, Roman P, Preston, Roland C, Zalewski, Adam, Maier, Timm, Peczuh, Mark W, Ernst, Beat

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