Type IIA topoisomerase inhibition by a new class of antibacterial agents von Bax, Benjamin D., Chan, Pan F., Eggleston, Drake S., Fosberry, Andrew, Gentry, Daniel R., Gorrec, Fabrice, Giordano, Ilaria, Hann, Michael M., Hennessy, Alan, Hibbs, Martin, Huang, Jianzhong, Jones, Emma, Jones, Jo, Brown, Kristin Koretke, Lewis, Ceri J., May, Earl W., Saunders, Martin R., Singh, Onkar, Spitzfaden, Claus E., Shen, Carol, Shillings, Anthony, Theobald, Andrew J., Wohlkonig, Alexandre, Pearson, Neil D., Gwynn, Michael N.

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Crystal Structure of Human Cytochrome P450 2D6 von Rowland, Paul, Blaney, Frank E., Smyth, Martin G., Jones, Jo J., Leydon, Vaughan R., Oxbrow, Amanda K., Lewis, Ceri J., Tennant, Mike G., Modi, Sandeep, Eggleston, Drake S., Chenery, Richard J., Bridges, Angela M.

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Synthesis and Recognition Properties of Aromatic Amide Oligomers:  Molecular Zippers von Bisson, Adrian P, Carver, Fiona J, Eggleston, Drake S, Haltiwanger, R. Curtis, Hunter, Christopher A, Livingstone, David L, McCabe, James F, Rotger, Carmen, Rowan, Alan E

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The structure of ribonuclease P protein from Staphylococcus aureus reveals a unique binding site for single-stranded RNA von Spitzfaden, Claus, Nicholson, Neville, Jones, Jo J, Guth, Sabine, Lehr, Ruth, Prescott, Cathy D, Hegg, Lisa A, Eggleston, Drake S

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1,4-Cyclohexanecarboxylates:  Potent and Selective Inhibitors of Phosophodiesterase 4 for the Treatment of Asthma von Christensen, Siegfried B, Guider, Aimee, Forster, Cornelia J, Gleason, John G, Bender, Paul E, Karpinski, Joseph M, DeWolf, Walter E, Barnette, Mary S, Underwood, David C, Griswold, Don E, Cieslinski, Lenora B, Burman, Miriam, Bochnowicz, Steven, Osborn, Ruth R, Manning, Carol D, Grous, Marilyn, Hillegas, Leonard M, Bartus, Joan O'Leary, Ryan, M. Dominic, Eggleston, Drake S, Haltiwanger, R. Curtis, Torphy, Theodore J

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The inophyllums, novel inhibitors of HIV-1 reverse transcriptase isolated from the Malaysian tree, Calophyllum inophyllum Linn von Patil, Ashok D, Freyer, Alan J, Eggleston, Drake S, Haltiwanger, R. Curtis, Bean, Mark F, Taylor, Paul B, Caranfa, Mary Jo, Breen, Ann L, Bartus, Henry R

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Substituent effects on aromatic interactions in the solid state von Adams, Harry, Bernad Jr, Pablo L., Hembury, Guy A., Hunter, Christopher A., McCabe, James F., Eggleston, Drake S., Haltiwanger, R. Curtis, Livingstone, David J., D. M. Harris, Kenneth, Kariuki, Benson M.

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Structure and redox properties of the water-oxidation catalyst [(bpy)2(OH2)RuORu(OH2)(bpy)2]4 von Gilbert, John A, Eggleston, Drake S, Murphy, Wyatt R, Geselowitz, Daniel A, Gersten, Susan W, Hodgson, Derek J, Meyer, Thomas J

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Defining and maintaining a high quality screening collection: the GSK experience von Lane, Stephen J., Eggleston, Drake S., Brinded, Keith A., Hollerton, John C., Taylor, Nicholas L., Readshaw, Simon A.

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Non-thiazolidinedione antihyperglycaemic agents. Part 5: Asymmetric aldol synthesis of ( S)-(−)-2-oxy-3-arylpropanoic acids von Haigh, David, Birrell, Helen C, Cantello, Barrie C.C, Eggleston, Drake S, Haltiwanger, R.Curtis, Hindley, Richard M, Ramaswamy, Anantha, Stevens, Nicola C

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Design and synthesis of a C7 mimetic for the predicted .gamma.-turn conformation found in several constrained RGD antagonists von Callahan, James F, Bean, John W, Burgess, Joelle L, Eggleston, Drake S, Hwang, Shing Mei, Kopple, Kenneth D, Koster, Paul F, Nichols, Andrew, Peishoff, Catherine E

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Structure–activity analysis of truncated orexin-A analogues at the orexin-1 receptor von Darker, John G, Porter, Roderick A, Eggleston, Drake S, Smart, Darren, Brough, Stephen J, Sabido-David, Cibele, Jerman, Jeffrey C

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Metal-assisted aldol condensation of chiral .alpha.-halogenated imide enolates: a stereocontrolled chiral epoxide synthesis von Abdel-Magid, Ahmed, Pridgen, Lendon N, Eggleston, Drake S, Lantos, Ivan

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Synthesis of imidazoles via hetero-Cope rearrangements von Lantos, Ivan, Zhang, Wei Yuan, Shui, Xiuqi, Eggleston, Drake S

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Structure determination of racemic trichogin A IV using centrosymmetric crystals von Toniolo, Claudio, Peggion, Cristina, Crisma, Marco, Formaggio, Fernando, Shui, Xiuqi, Eggleston, Drake S.

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Cellular uptake and spread of the cell-permeable peptide penetratin in adult rat brain von Bolton, Sarah J., Jones, Declan N. C., Darker, John G., Eggleston, Drake S., Hunter, A. Jacqueline, Walsh, Frank S.

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Conformational Preferences in a Benzodiazepine Series of Potent Nonpeptide Fibrinogen Receptor Antagonists von Keenan, Richard M, Callahan, James F, Samanen, James M, Bondinell, William E, Calvo, Raul R, Chen, Lichong, DeBrosse, Charles, Eggleston, Drake S, Haltiwanger, R. Curtis, Hwang, Shing Mei, Jakas, Dalia R, Ku, Thomas W, Miller, William H, Newlander, Kenneth A, Nichols, Andrew, Parker, Michael F, Southhall, Linda S, Uzinskas, Irene, Vasko-Moser, Janice A, Venslavsky, Joseph W, Wong, Angela S, Huffman, William F

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Discovery of a Novel Class of Substituted Pyrrolooctahydroisoquinolines as Potent and Selective δ Opioid Agonists, Based on an Extension of the Message−Address Concept von Dondio, Giulio, Ronzoni, Silvano, Eggleston, Drake S, Artico, Marco, Petrillo, Paola, Petrone, Giuseppe, Visentin, Luciano, Farina, Carlo, Vecchietti, Vittorio, Clarke, Geoffrey D

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(E)-3-[[[[6-(2-Carboxyethenyl)-5-[[8-(4-methoxyphenyl)octyl]oxy]-2-pyridinyl]methyl]thio]methyl]benzoic Acid and Related Compounds: High Affinity Leukotriene B4 Receptor Antagonist... von Daines, Robert A, Chambers, Pamela A, Eggleston, Drake S, Foley, James J, Griswold, Don E, Haltiwanger, R. Curtis, Jakas, Dalia R, Kingsbury, William D, Martin, Lenox D

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Inhibitors of bacterial tyrosyl tRNA synthetase: synthesis of four stereoisomeric analogues of the natural product SB-219383 von Berge, John M, Copley, Royston C.B, Eggleston, Drake S, Hamprecht, Dieter W, Jarvest, Richard L, Mensah, Lucy M, O'Hanlon, Peter J, Pope, Andrew J

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