Fructose-1,6-bisphosphatase Inhibitors. 1. Purine Phosphonic Acids as Novel AMP Mimics von Dang, Qun, Brown, Brian S, Liu, Yan, Rydzewski, Robert M, Robinson, Edward D, Poelje, Paul D. van, Reddy, M. Rami, Erion, Mark D

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Novel, Nonpeptidic Cyanamides as Potent and Reversible Inhibitors of Human Cathepsins K and L von Falgueyret, Jean-Pierre, Oballa, Renata M, Okamoto, Osamu, Wesolowski, Gregg, Aubin, Yves, Rydzewski, Robert M, Prasit, Peppi, Riendeau, Denis, Rodan, Sevgi B, Percival, M. David

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Optimization of Subsite Binding to the β5 Subunit of the Human 20S Proteasome Using Vinyl Sulfones and 2-Keto-1,3,4-oxadiazoles:  Syntheses and Cellular Properties of Potent, Selec... von Rydzewski, Robert M, Burrill, Leland, Mendonca, Rohan, Palmer, James T, Rice, Mark, Tahilramani, Ram, Bass, Kathryn E, Leung, Ling, Gjerstad, Erik, Janc, James W, Pan, Lin

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Synthesis and anti-HIV activity of 4'-azido- and 4'-methoxynucleosides von Maag, Hans, Rydzewski, Robert M, McRoberts, Mary Jane, Crawford-Ruth, Diane, Verheyden, Julien P. H, Prisbe, Ernest J

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An unexpected cyclization discovered during the synthesis of 8-substituted purines from a 4,5-diaminopyrimidine von Dang, Qun, Rydzewski, Robert M., Cashion, Daniel K., Erion, Mark D.

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Design and synthesis of selective keto-1,2,4-oxadiazole-based tryptase inhibitors von Palmer, James T., Rydzewski, Robert M., Mendonca, Rohan V., Sperandio, David, Spencer, Jeffrey R., Hirschbein, Bernard L., Lohman, Julia, Beltman, Jeri, Nguyen, Margaret, Liu, Liang

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Bis[(para-methoxy)benzyl] phosphonate prodrugs with improved stability and enhanced cell penetration von Dang, Qun, Liu, Yan, Rydzewski, Robert M., Brown, Brian S., Robinson, Edward, van Poelje, Paul D., Colby, Timothy J., Erion, Mark D.

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Peptidic 1-cyanopyrrolidines: synthesis and SAR of a series of potent, selective cathepsin inhibitors von Rydzewski, Robert M, Bryant, Clifford, Oballa, Renata, Wesolowski, Gregg, Rodan, Sevgi B, Bass, Kathryn E, Wong, Darren H

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Design and Synthesis of Tri-Ring P3 Benzamide-Containing Aminonitriles as Potent, Selective, Orally Effective Inhibitors of Cathepsin K von Palmer, James T, Bryant, Clifford, Wang, Dan-Xiong, Davis, Dana E, Setti, Eduardo L, Rydzewski, Robert M, Venkatraman, Shankar, Tian, Zong-Qiang, Burrill, Leland C, Mendonca, Rohan V, Springman, Eric, McCarter, John, Chung, Tobee, Cheung, Harry, Janc, James W, McGrath, Mary, Somoza, John R, Enriquez, Philip, Yu, Z. Walter, Strickley, Robert M, Liu, Liang, Venuti, Michael C, Percival, M. David, Falgueyret, Jean-Pierre, Prasit, Peppi, Oballa, Renata, Riendeau, Denis, Young, Robert N, Wesolowski, Gregg, Rodan, Sevgi B, Johnson, Colena, Kimmel, Donald B, Rodan, Gideon

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pH Dependence of inhibitors targeting the occluding loop of cathepsin B von Cathers, Brian E, Barrett, Cynthia, Palmer, James T, Rydzewski, Robert M

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Design and Synthesis of Tri-Ring P 3 Benzamide-Containing Aminonitriles as Potent, Selective, Orally Effective Inhibitors of Cathepsin K von Palmer, James T., Bryant, Clifford, Wang, Dan-Xiong, Davis, Dana E., Setti, Eduardo L., Rydzewski, Robert M., Venkatraman, Shankar, Tian, Zong-Qiang, Burrill, Leland C., Mendonca, Rohan V., Springman, Eric, McCarter, John, Chung, Tobee, Cheung, Harry, Janc, James W., McGrath, Mary, Somoza, John R., Enriquez, Philip, Yu, Z. Walter, Strickley, Robert M., Liu, Liang, Venuti, Michael C., Percival, M. David, Falgueyret, Jean-Pierre, Prasit, Peppi, Oballa, Renata, Riendeau, Denis, Young, Robert N., Wesolowski, Gregg, Rodan, Sevgi B., Johnson, Colena, Kimmel, Donald B., Rodan, Gideon

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An Efficient Synthetic Route to Ethyl 2-Aryl-4-hydroxy-1,3(2H,4H)- dioxoisoquinoline-4-carboxylates(1) von Semple, J. Edward, Rydzewski, Robert M., Gardner, Gary

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Synthesis and antiviral evaluation of 6'-substituted aristeromycins: potential mechanism-based inhibitors of S-adenosylhomocysteine hydrolase von Madhavan, G. V. Bindu, McGee, Danny P. C, Rydzewski, Robert M, Boehme, Richard, Martin, John C, Prisbe, Ernest J

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Optimization of subsite binding to the beta5 subunit of the human 20S proteasome using vinyl sulfones and 2-keto-1,3,4-oxadiazoles: syntheses and cellular properties of potent, sel... von Rydzewski, Robert M, Burrill, Leland, Mendonca, Rohan, Palmer, James T, Rice, Mark, Tahilramani, Ram, Bass, Kathryn E, Leung, Ling, Gjerstad, Erik, Janc, James W, Pan, Lin

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Cathepsin B inactivation attenuates hepatic apoptosis and fibrosis during cholestasis von Canbay, Ali, Higuchi, Hajime, Guicciardi, Maria E., Bronk, Steven F., Feldstein, Ariel, Taniai, Makiko, Rydzewski, Robert M., Gores, Gregory J.

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Synthesis and structure-activity relationships of a new series of antiarrhythmic agents: 4,4-disubstituted hexahydro-3H-pyrido[1,2-c]pyrimidin-3-ones and related compounds von Chorvat, Robert J, Prodan, Kathleen A, Adelstein, Gilbert W, Rydzewski, Robert M, McLaughlin, Kathleen T, Stamm, Margarete H, Frederick, Leo G, Schniepp, Henry C, Stickney, Janice L

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An allylic azide route to 4'-azido carbocyclic nucleosides. Synthesis of (.+-.)-(1'.alpha.,2'.alpha.,3'.beta.)- and (.+-.)-(1'.alpha.,2'.beta.,3'.beta.)-1-[1-azido-2-hydroxy-1-(hyd... von Maag, Hans, Rydzewski, Robert M.

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4-Substituted-5(3)-carbamoyl-3(5)-(2-deoxy-β-D-ribofuranosyl)pyrazoles. Application of Palladium Catalyzed Glycal Coupling Methodology to the Synthesis of Pyrazofurin Analogs von Erion, Mark D., Rydzewski†, Robert M.

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An Efficient Synthetic Route to Ethyl 2-Aryl-4-hydroxy-1,3(2H,4H)- dioxoisoquinoline-4-carboxylates1 von Semple, J. Edward, Rydzewski, Robert M., Gardner, Gary

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An Efficient Synthetic Route to Ethyl 2-Aryl-4-hydroxy-1,3(2 H ,4 H )- dioxoisoquinoline-4-carboxylates 1 von Semple, J. Edward, Rydzewski, Robert M., Gardner, Gary

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