(−)-Rhazinilam and the diphenylpyridazinone NSC 613241: Two compounds inducing the formation of morphologically similar tubulin spirals but binding apparently to two distinct sites... von Bai, Ruoli, Hamel, Ernest

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Insight on [1,3]thiazolo[4,5-e]isoindoles as tubulin polymerization inhibitors von Spanò, Virginia, Barreca, Marilia, Rocca, Roberta, Bortolozzi, Roberta, Bai, Ruoli, Carbone, Anna, Raimondi, Maria Valeria, Piccionello, Antonio Palumbo, Montalbano, Alessandra, Alcaro, Stefano, Hamel, Ernest, Viola, Giampietro, Barraja, Paola

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12,13-Aziridinyl Epothilones. Stereoselective Synthesis of Trisubstituted Olefinic Bonds from Methyl Ketones and Heteroaromatic Phosphonates and Design, Synthesis, and Biological E... von Nicolaou, K. C, Rhoades, Derek, Wang, Yanping, Bai, Ruoli, Hamel, Ernest, Aujay, Monette, Sandoval, Joseph, Gavrilyuk, Julia

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Total Synthesis of Potent Antitumor Macrolide (-)-Zampanolide: An Oxidative Intramolecular Cyclization-Based Strategy von Ghosh, Arun K., Cheng, Xu, Bai, Ruoli, Hamel, Ernest

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Toward Highly Potent Cancer Agents by Modulating the C‑2 Group of the Arylthioindole Class of Tubulin Polymerization Inhibitors von La Regina, Giuseppe, Bai, Ruoli, Rensen, Whilelmina Maria, Di Cesare, Erica, Coluccia, Antonio, Piscitelli, Francesco, Famiglini, Valeria, Reggio, Alessia, Nalli, Marianna, Pelliccia, Sveva, Da Pozzo, Eleonora, Costa, Barbara, Granata, Ilaria, Porta, Amalia, Maresca, Bruno, Soriani, Alessandra, Iannitto, Maria Luisa, Santoni, Angela, Li, Junjie, Miranda Cona, Marlein, Chen, Feng, Ni, Yicheng, Brancale, Andrea, Dondio, Giulio, Vultaggio, Stefania, Varasi, Mario, Mercurio, Ciro, Martini, Claudia, Hamel, Ernest, Lavia, Patrizia, Novellino, Ettore, Silvestri, Romano

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Synthesis and evaluation of diaryl sulfides and diaryl selenide compounds for antitubulin and cytotoxic activity von dos Santos, Edson dos A., Hamel, Ernest, Bai, Ruoli, Burnett, James C., Tozatti, Camila Santos Suniga, Bogo, Danielle, Perdomo, Renata T., Antunes, Alexandra M.M., Marques, M. Matilde, Matos, Maria de F.C., de Lima, Dênis P.

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Discovery of Biarylaminoquinazolines as Novel Tubulin Polymerization Inhibitors von Marzaro, Giovanni, Coluccia, Antonio, Ferrarese, Alessandro, Brun, Paola, Castagliuolo, Ignazio, Conconi, Maria Teresa, La Regina, Giuseppe, Bai, Ruoli, Silvestri, Romano, Hamel, Ernest, Chilin, Adriana

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New Arylthioindoles and Related Bioisosteres at the Sulfur Bridging Group. 4. Synthesis, Tubulin Polymerization, Cell Growth Inhibition, and Molecular Modeling Studies von La Regina, Giuseppe, Sarkar, Taradas, Bai, Ruoli, Edler, Michael C, Saletti, Roberto, Coluccia, Antonio, Piscitelli, Francesco, Minelli, Lara, Gatti, Valerio, Mazzoccoli, Carmela, Palermo, Vanessa, Mazzoni, Cristina, Falcone, Claudio, Scovassi, Anna Ivana, Giansanti, Vincenzo, Campiglia, Pietro, Porta, Amalia, Maresca, Bruno, Hamel, Ernest, Brancale, Andrea, Novellino, Ettore, Silvestri, Romano

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Interactions of Halichondrin B and Eribulin with Tubulin von Bai, Ruoli, Nguyen, Tam Luong, Burnett, James C, Atasoylu, Onur, Munro, Murray H. G, Pettit, George R, Smith, Amos B, Gussio, Rick, Hamel, Ernest

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Enantioselective Synthesis of (+)-Chamaecypanone C: A Novel Microtubule Inhibitor von Dong, Suwei, Hamel, Ernest, Bai, Ruoli, Covell, David G, Beutler, John A, Porco, John A. Jr

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Synthesis, antiproliferative activity, and mechanism of action of a series of 2-{[(2 E)-3-phenylprop-2-enoyl]amino}benzamides von Raffa, Demetrio, Maggio, Benedetta, Plescia, Fabiana, Cascioferro, Stella, Plescia, Salvatore, Raimondi, Maria Valeria, Daidone, Giuseppe, Tolomeo, Manlio, Grimaudo, Stefania, Di Cristina, Antonietta, Pipitone, Rosaria Maria, Bai, Ruoli, Hamel, Ernest

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Comparison of the Activities of the Truncated Halichondrin B Analog NSC 707389 (E7389) with Those of the Parent Compound and a Proposed Binding Site on Tubulin von Dabydeen, Donnette A, Burnett, James C, Bai, Ruoli, Verdier-Pinard, Pascal, Hickford, Sarah J H, Pettit, George R, Blunt, John W, Munro, Murray H G, Gussio, Rick, Hamel, Ernest

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Synthesis and Biological Evaluation of Dihydrobenzofuran Lignans and Related Compounds as Potential Antitumor Agents that Inhibit Tubulin Polymerization von Pieters, Luc, Van Dyck, Stefaan, Gao, Mei, Bai, Ruoli, Hamel, Ernest, Vlietinck, Arnold, Lemière, Guy

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Deciphering the key heterocyclic scaffolds in targeting microtubules, kinases and carbonic anhydrases for cancer drug development von Peerzada, Mudasir Nabi, Hamel, Ernest, Bai, Ruoli, Supuran, Claudiu T., Azam, Amir

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Laulimalide and Paclitaxel: A Comparison of Their Effects on Tubulin Assembly and Their Synergistic Action When Present Simultaneously von Gapud, Eric J, Bai, Ruoli, Ghosh, Arun K, Hamel, Ernest

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Actin is the primary cellular receptor of bistramide A von Kozmin, Sergey A, Statsuk, Alexander V, Bai, Ruoli, Baryza, Jeremy L, Verma, Vishal A, Hamel, Ernest, Wender, Paul A

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(−)-RHAZINILAM AND THE DIPHENYLPYRIDAZINONE NSC 613241: TWO COMPOUNDS INDUCING THE FORMATION OF MORPHOLOGICALLY SIMILAR TUBULIN SPIRALS BUT BINDING APPARENTLY TO TWO DISTINCT SITES... von Bai, Ruoli, Hamel, Ernest

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Intracellular Activation and Deactivation of Tasidotin, an Analog of Dolastatin 15: Correlation with Cytotoxicity von Bai, Ruoli, Edler, Michael C, Bonate, Peter L, Copeland, Terry D, Pettit, George R, Ludueña, Richard F, Hamel, Ernest

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Novel Microtubule-Interacting Phenoxy Pyridine and Phenyl Sulfanyl Pyridine Analogues for Cancer Therapy von Anchoori, Ravi Kumar, Kortenhorst, Madeleine Susanne Quirine, Hidalgo, Manuel, Sarkar, Taradas, Hallur, Gurulingappa, Bai, Ruoli, Diest, Paul J. Van, Hamel, Ernest, Khan, Saeed R

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Diazonamide A and a Synthetic Structural Analog: Disruptive Effects on Mitosis and Cellular Microtubules and Analysis of Their Interactions with Tubulin von Cruz-Monserrate, Zobeida, Vervoort, Hélène C, Bai, Ruoli, Newman, David J, Howell, Stephen B, Los, Gerrit, Mullaney, Jeffrey T, Williams, Michael D, Pettit, George R, Fenical, William, Hamel, Ernest

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