N-(3-Fluoro-4-(4-(2-methoxy or 2,3-dichlorophenyl)piperazine-1-yl)butyl)arylcarboxamides as Selective Dopamine D3 Receptor Ligands: Critical Role of the Carboxamide Linker for D3 R... von Banala, Ashwini K, Levy, Benjamin A, Khatri, Sameer S, Furman, Cheryse A, Roof, Rebecca A, Mishra, Yogesh, Griffin, Suzy A, Sibley, David R, Luedtke, Robert R, Newman, Amy Hauck

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Identification of Small-Molecule Inhibitors of RGS4 Using a High-Throughput Flow Cytometry Protein Interaction Assay von Roman, David L, Talbot, Jeffery N, Roof, Rebecca A, Sunahara, Roger K, Traynor, John R, Neubig, Richard R

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New approaches for challenging therapeutic targets von Sharma, Karlie R., Malik, Abir, Roof, Rebecca A., Boyce, Jim P., Verma, Sharad K.

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Modification of cocaine self-administration by buspirone (buspar®): potential involvement of D3 and D4 dopamine receptors von Bergman, Jack, Roof, Rebecca A., Furman, Cheryse A., Conroy, Jennie L., Mello, Nancy K., Sibley, David R., Skolnick, Phil

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NINDS launches network to develop treatments for ultra-rare neurological diseases von Schor, Nina F., Tamiz, Amir P., Koroshetz, Walter J., Broome, Ann-Marie

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Real-time Detection of Basal and Stimulated G Protein GTPase Activity Using Fluorescent GTP Analogues von Jameson, Emily E, Roof, Rebecca A, Whorton, Matthew R, Mosberg, Henry I, Sunahara, Roger K, Neubig, Richard R, Kennedy, Robert T

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Investigation of the binding and functional properties of extended length D3 dopamine receptor-selective antagonists von Furman, Cheryse A, Roof, Rebecca A, Moritz, Amy E, Miller, Brittney N, Doyle, Trevor B, Free, R. Benjamin, Banala, Ashwini K, Paul, Noel M, Kumar, Vivek, Sibley, Christopher D, Newman, Amy Hauck, Sibley, David R

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Mechanism of Action and Structural Requirements of Constrained Peptide Inhibitors of RGS Proteins von Roof, Rebecca A., Jin, Yafei, Roman, David L., Sunahara, Roger K., Ishii, Masaru, Mosberg, Henry I., Neubig, Richard R.

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Differential modulation of mu‐opioid receptor signaling to adenylyl cyclase by regulators of G protein signaling proteins 4 or 8 and 7 in permeabilised C6 cells is Gα subtype depen... von Talbot, Jeffery N., Roman, David L., Clark, Mary J., Roof, Rebecca A., Tesmer, John J. G., Neubig, Richard R., Traynor, John R.

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Novel Peptide Ligands of RGS4 from a Focused One-Bead, One-Compound Library von Roof, Rebecca A, Sobczyk-Kojiro, Katarzyna, Turbiak, Anjanette J, Roman, David L, Pogozheva, Irina D, Blazer, Levi L, Neubig, Richard R, Mosberg, Henry I

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A covalent peptide inhibitor of RGS4 identified in a focused one-bead, one compound library screen von Roof, Rebecca A, Roman, David L, Clements, Samuel T, Sobczyk-Kojiro, Katarzyna, Blazer, Levi L, Ota, Shodai, Mosberg, Henry I, Neubig, Richard R

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Mechanistic studies with N-benzyl-1-aminobenzotriazole-inactivated CYP2B1: differential effects on the metabolism of 7-ethoxy-4-(trifluoromethyl)coumarin, testosterone, and benzphe... von Kent, Ute M, Pascual, Lise, Roof, Rebecca A, Ballou, David P, Hollenberg, Paul F

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Buspirone is a potent antagonist at D 3 and D 4 Dopamine Receptors and attenuates the reinforcing effects of cocaine in a primate model von Roof, Rebecca A, Bergman, Jack, Furman, Chersyse A., Conroy, Jennie L, Mello, Nancy K, Skolnick, Phil, Sibley, David R

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Modification of cocaine self-administration by buspirone (buspar registered ): potential involvement of D sub(3) and D sub(4) dopamine receptors von Bergman, Jack, Roof, Rebecca A, Furman, Cheryse A, Conroy, Jennie L, Mello, Nancy K, Sibley, David R, Skolnick, Phil

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High‐Throughput Screening for Novel Modulators of the D3 Dopamine Receptor von Furman, Cheryse A, Free, R. Benjamin, Roof, Rebecca A, Conroy, Jennie L, Titus, Steven A, Southall, Noel, Sibley, David R

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High‐Throughput Screening for Novel Modulators of the D1 Dopamine Receptor von Conroy, Jennie L., Hazelwood, Lisa A., Free, R. Benjamin, Roof, Rebecca A., Furman, Cheryse A., Titus, Steven A., Southall, Noel, Ferrer, Marc, Sibley, David R.

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Development of High Throughput Screening Assays for the Discovery of Functionally‐Selective D2 Dopamine Receptor Ligands von Roof, Rebecca A., Free, R. Benjamin, Duan, Lihua, Urizar, Eneko, Furman, Cheryse A., Conroy, Jennie L., Titus, Steven A., Southall, Noel, Javitch, Jonathan A., Sibley, David R.

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High‐Throughput Screening for Allosteric Modulators of the D2 Dopamine Receptor von Free, R. Benjamin, Roof, Rebecca A., Conroy, Jennie L., Furman, Cheryse A., Titus, Steven A., Southall, Noel, Ferrer, Marc, Han, Yang, Javitch, Jonathan A., Sibley, David R.

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N-(3-Fluoro-4-(4-(2-methoxy or 2,3-dichlorophenyl) piperazine-1-yl)-butyl)-aryl carboxamides as Selective Dopamine D3 Receptor Ligands: Critical Role of the Carboxamide Linker for... von Banala, Ashwini K., Levy, Benjamin A., Khatri, Sameer S., Furman, Cheryse A., Roof, Rebecca A., Mishra, Yogesh, Griffin, Suzy A., Sibley, David R., Luedtke, Robert R., Newman, Amy Hauck

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Lipid rafts and membrane cholesterol are involved in regulating D2 dopamine receptor signaling von Hazelwood, Lisa A, Romanelli, Robert J, Free, R Benjamin, Roof, Rebecca A, Javitch, Jonathan A, Neve, Kim A, Sibley, David R

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