Development of Hamari Ligands for Practical Asymmetric Synthesis of Tailor-Made Amino Acids von Han, Jianlin, Romoff, Todd T, Moriwaki, Hiroki, Konno, Hiroyuki, Soloshonok, Vadim A

Volltext

Scale-up Synthesis of (R)- and (S)‑N‑(2-Benzoyl-4-chlorophenyl)-1-(3,4-dichlorobenzyl)pyrrolidine-2-carboxamide Hydrochloride, A Versatile Reagent for the Preparation of Tailor-Mad... von Romoff, Todd T, Palmer, Andrew B, Mansour, Noel, Creighton, Christopher J, Miwa, Toshio, Ejima, Yuki, Moriwaki, Hiroki, Soloshonok, Vadim A

Volltext

Synthesis, in vitro and in vivo activity of thiamine antagonist transketolase inhibitors von Thomas, Allen A., Le Huerou, Y., De Meese, J., Gunawardana, Indrani, Kaplan, Tomas, Romoff, Todd T., Gonzales, Stephen S., Condroski, Kevin, Boyd, Steven A., Ballard, Josh, Bernat, Bryan, DeWolf, Walter, Han, May, Lee, Patrice, Lemieux, Christine, Pedersen, Robin, Pheneger, Jed, Poch, Greg, Smith, Darin, Sullivan, Francis, Weiler, Solly, Wright, S. Kirk, Lin, Jie, Brandhuber, Barb, Vigers, Guy

Volltext

Non-charged thiamine analogs as inhibitors of enzyme transketolase von Thomas, Allen A., De Meese, J., Le Huerou, Y., Boyd, Steven A., Romoff, Todd T., Gonzales, Steven S., Gunawardana, Indrani, Kaplan, Tomas, Sullivan, Francis, Condroski, Kevin, Lyssikatos, Joseph P., Aicher, Thomas D., Ballard, Josh, Bernat, Bryan, DeWolf, Walter, Han, May, Lemieux, Christine, Smith, Darin, Weiler, Solly, Wright, S. Kirk, Vigers, Guy, Brandhuber, Barb

Volltext

Rapid and efficient syntheses of tryptophans using a continuous-flow quaternization-substitution reaction of gramines with a chiral nucleophilic glycine equivalent von Koiwa, Daichi, Ohira, Masayuki, Hiramatsu, Takahiro, Abe, Hidenori, Kawamoto, Tetsuji, Ishihara, Yuji, Ignacio, Bernardo, Mansour, Noel, Romoff, Todd

Volltext

Prodrug thiamine analogs as inhibitors of the enzyme transketolase von Le Huerou, Yvan, Gunawardana, Indrani, Thomas, Allen A., Boyd, Steven A., de Meese, Jason, deWolf, Walter, Gonzales, Steven S., Han, May, Hayter, Laura, Kaplan, Tomas, Lemieux, Christine, Lee, Patrice, Pheneger, Jed, Poch, Gregory, Romoff, Todd T., Sullivan, Francis, Weiler, Solly, Wright, S. Kirk, Lin, Jie

Volltext

Large-Scale Synthesis of the Glycine Schiff Base Ni(II) Complex Derived from (S)- and (R)-N-(2-Benzoyl-4-chlorophenyl)-1-[(3,4-dichlorophenyl)methyl]-2-pyrrolidinecarboxamide von Romoff, Todd T., Ignacio, Bernardo G., Mansour, Noel, Palmer, Andrew B., Creighton, Christopher J., Abe, Hidenori, Moriwaki, Hiroki, Han, Jianlin, Konno, Hiroyuki, Soloshonok, Vadim A.

Volltext

Mechanistic Studies of an Unusual Amide Bond Scission von Creighton, Christopher J, Romoff, Todd T, Bu, Jane H, Goodman, Murray

Volltext

Conformationally Constrained Peptides and Semipeptides Derived from RGD as Potent Inhibitors of the Platelet Fibrinogen Receptor and Platelet Aggregation von Ali, Fadia E, Bennett, Donald B, Calvo, Raul R, Elliott, John D, Hwang, Shing-Mei, Ku, Thomas W, Lago, M. Amparo, Nichols, Andrew J, Romoff, Todd T

Volltext

3-(Diethoxyphosphoryloxy)-1,2,3- benzotriazin-4(3H)-one (DEPBT):  A New Coupling Reagent with Remarkable Resistance to Racemization von Li, Haitao, Jiang, Xiaohui, Ye, Yun-hua, Fan, Chongxu, Romoff, Todd, Goodman, Murray

Volltext

Large-Scale Synthesis of the Glycine Schiff Base Ni(II) Complex Derived from (S)- and (R)‑N‑(2-Benzoyl-4-chlorophenyl)-1-[(3,4-dichloro­phenyl)­methyl]-2-pyrrolidine­carboxamide... von Romoff, Todd T, Ignacio, Bernardo G, Mansour, Noel, Palmer, Andrew B, Creighton, Christopher J, Abe, Hidenori, Moriwaki, Hiroki, Han, Jianlin, Konno, Hiroyuki, Soloshonok, Vadim A

Volltext

Identification and characterization of a potent and selective antagonist of the prostaglandin D2 receptor (94.23) von Eberhardt, Christine, Wright, Dale, Gomez, Anna, Cook, Adam, Doherty, George, Corrette, Christopher, Hunt, Kevin, Clark, Christopher, Kim, Ganghyeok, Romoff, Todd, Delisle, Kirk, Hayter, Laura, Neale, Jason, Dean, Brian, Chantry, David, Carter, Laura, Burgess, Laurence E

Volltext

Regioselectivity and kinetics of hydride transfer in substituted 1-benzyl-3-quinolinecarboxamide redox reactions von Romoff, Todd T, Sampson, Nicole S, Van Eikeren, Paul

Volltext

The in vitro pharmacological profile of SK&F 106760, a novel GPIIB/IIIA antagonist von Nichols, Andrew J., Vasko, Janice A., Valocik, Richard E., Kopaciewicz, Linda J., Storer, Barbara L., Ali, Fadia E., Romoff, Todd, Calvo, Raul, Samanen, James M.

Volltext

Solid Phase Synthesis of 3-Acyl-2,4-Pyrrolidinediones (3-Acyl Tetramic Acids) via Mild Cyclative Cleavage von Romoff, Todd T., Ma, Liang, Wang, Yongwen, Campbell, David A.

Volltext

GUANIDINYLATION REAGENTS von ROMOFF TODD T. ROMOFF TODD T, GOODMAN MURRAY GOODMAN MURRAY, FEICHTINGER KONRAD FEICHTINGER KONRAD

Volltext bestellen

Investigation of conformational specificity at GPIIb/IIIa: evaluation of conformationally constrained RGD peptides von Peishoff, Catherine E, Ali, Fadia E, Bean, John W, Calvo, Raul, D'Ambrosio, Cynthia A, Eggleston, Drake S, Kline, Tammy Page, Koster, Paul F, Hwang, S. M

Volltext

6-SUBSTITUTED PHENOXYCHROMAN CARBOXYLIC ACIS DERIVATIVES von KIM, GANGHYEOK, CORRETTE, CHRISTOPHER P, ROBERT KIRK DELISLE, DOHERTY, GEORGE A, CLARK, CHRISTOPHER T, BURGESS, LAURENCE E, ROMOFF, TODD, HUNT, KEVIN W, COOK, ADAM

Volltext bestellen

Urethane-protected N-carboxyanhydrides (UNCAs) as unique reactants for the study of intrinsic racemization tendencies in peptide synthesis von ROMOFF, TODD T., GOODMAN, MURRAY

Volltext

6-SUBSTITUTED PHENOXYCHROMAN CARBOXYLIC ACID DERIVATIVES von BURGESS, Laurence, E, DOHERTY, George, A, COOK, Adam, CORRETTE, Christopher, P, HUNT, Kevin, W, CLARK, Christopher, T, DELISLE, Robert, Kirk, ROMOFF, Todd, KIM, Ganghyeok

Volltext bestellen