Utilizing Chemical Genomics to Identify Cytochrome b as a Novel Drug Target for Chagas Disease von Khare, Shilpi, Roach, Steven L, Barnes, S Whitney, Hoepfner, Dominic, Walker, John R, Chatterjee, Arnab K, Neitz, R Jeffrey, Arkin, Michelle R, McNamara, Case W, Ballard, Jaime, Lai, Yin, Fu, Yue, Molteni, Valentina, Yeh, Vince, McKerrow, James H, Glynne, Richard J, Supek, Frantisek

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Discovery of nonsteroidal glucocorticoid receptor ligands based on 6-indole-1,2,3,4-tetrahydroquinolines von Roach, Steven L., Higuchi, Robert I., Adams, Mark E., Liu, Yan, Karanewsky, Donald S., Marschke, Keith B., Mais, Dale E., Miner, Jeffrey N., Zhi, Lin

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Synthesis and Characterization of Nonsteroidal Glucocorticoid Receptor Modulators for Multiple Myeloma von Hudson, Andrew R, Roach, Steven L, Higuchi, Robert I, Phillips, Dean P, Bissonnette, Reid P, Lamph, William W, Yen, Jean, Li, Yongkai, Adams, Mark E, Valdez, Lino J, Vassar, Angie, Cuervo, Catalina, Kallel, E. Adam, Gharbaoui, Catherine J, Mais, Dale E, Miner, Jeffrey N, Marschke, Keith B, Rungta, Deepa, Negro-Vilar, Andrés, Zhi, Lin

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Inhibition of pancreatic cancer growth by the dietary isoprenoids farnesol and geraniol von Burke, Y.D, Stark, M.J, Roach, S.L, Sen, S.E, Crowell, P.L

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Ferric Chloride Hexahydrate:  A Mild Hydrolytic Agent for the Deprotection of Acetals von Sen, Stephanie E, Roach, Steven L, Boggs, Janet K, Ewing, Gregory J, Magrath, Joe

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Lead Identification to Clinical Candidate Selection: Drugs for Chagas Disease von Neitz, R. Jeffrey, Chen, Steven, Supek, Frantisek, Yeh, Vince, Kellar, Danielle, Gut, Jiri, Bryant, Clifford, Gallardo-Godoy, Alejandra, Molteni, Valentina, Roach, Steven L., Chatterjee, Arnab K., Robertson, Stephanie, Renslo, Adam R., Arkin, Michelle, Glynne, Richard, McKerrow, James, Siqueira-Neto, Jair L.

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Tetrahydroquinoline glucocorticoid receptor agonists: Discovery of a 3-hydroxyl for improving receptor selectivity von Roach, Steven L., Higuchi, Robert I., Hudson, Andrew R., Adams, Mark E., Syka, Peter M., Mais, Dale E., Miner, Jeffrey N., Marschke, Keith B., Zhi, Lin

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Discovery of orally available tetrahydroquinoline-based glucocorticoid receptor agonists von Hudson, Andrew R., Higuchi, Robert I., Roach, Steven L., Adams, Mark E., Vassar, Angela, Syka, Peter M., Mais, Dale E., Miner, Jeffrey N., Marschke, Keith B., Zhi, Lin

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Nonsteroidal 2,3-dihydroquinoline glucocorticoid receptor agonists with reduced PEPCK activation von Hudson, Andrew R., Higuchi, Robert I., Roach, Steven L., Valdez, Lino J., Adams, Mark E., Vassar, Angie, Rungta, Deepa, Syka, Peter M., Mais, Dale E., Marschke, Keith B., Zhi, Lin

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Tetrahydroquinolin-3-yl carbamate glucocorticoid receptor agonists with reduced PEPCK activation von Roach, Steven L., Higuchi, Robert I., Hudson, Andrew R., Vassar, Angie, Grant, Virginia H.S., Lamer, Ryan, Hooper, Charlene, Rungta, Deepa, Syka, Peter M., Mais, Dale E., Marschke, Keith B., Zhi, Lin

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5 (Z) -Benzylidene -1,2 -dihydro -9 -hydroxy -10 -methoxy -2,2, 4 -trimethyl -5H-1 -aza -6 -oxa -chrysenes as non-steroidal glucocorticoid receptor modulators von ARDECKY, Robert J, HUDSON, Andrew R, LOPEZ, Francisco J, MARSCHKE, Keith B, MINER, Jeffrey N, KARANEWSKY, Donald S, NEGRO-VILAR, Andrés, LIN ZHI, PHILLIPS, Dean P, TYHONAS, John S, DECKHUT, Charlotte, LAU, Thomas L, YONGKAI LI, MARTINBOROUGH, Esther A, ROACH, Steven L, HIGUCHI, Robert I

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Zeolite-Mediated Cyclization of an Epoxide-Containing Polyene von Sen, Stephanie E, Zhang, Yan zhi, Roach, Steven L

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Biomimetic Cyclization of Enamide-Containing Polyenes as a New Route to Azapolycycles von Sen, Stephanie E, Roach, Steven L

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Utilizing Chemical Genomics to Identify Cytochrome b as a Novel Drug Target for Chagas Disease: e1005058 von Khare, Shilpi, Roach, Steven L, Barnes, S Whitney, Hoepfner, Dominic, Walker, John R, Chatterjee, Arnab K, Neitz, R Jeffrey, Arkin, Michelle R, McNamara, Case W, Ballard, Jaime, Lai, Yin, Fu, Yue, Molteni, Valentina, Yeh, Vince, McKerrow, James H, Glynne, Richard J, Supek, Frantisek

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Discovery of Non-Peptidyl Small-Molecule Human GCSF Receptor Agonists for the Potential Treatment of Neutropenia von Marschke, Keith, Rungta, Deepa, Slavin, Daniela A, Sanders, Jennifer, Roach, Steven L, Pickens, Jason C, Shen, Yixing, van Oeveren, Arjan, Hong, Mei Hua, Sun, Hong, Bissonnette, Reid P., Syka, Peter M, Zhi, Lin

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NON-Peptidyl Small Molecule EPO Receptor Agonists Are Potent Pathway Selective Inducers of Erythropoiesis von Bissonnette, Reid P., Rungta, Deepa, Hudson, Andrew R, Roach, Steven L, Hong, Mei Hua, Sun, Hong, Hu, Junlian, Ward, James N, Luo, Wen, Sanders, Jen E, Syka, Peter M, Slavin, Daniela A, Zhi, Lin, Marschke, Keith B

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A Convenient Two-Step Procedure for the Synthesis of Substituted Allylic Amines from Allylic Alcohols von Sen, Stephanie E., Roach, Steven L.

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5( Z)-Benzylidene-1,2-dihydro-9-hydroxy-10-methoxy-2,2,4-trimethyl-5 H-1-aza-6-oxa-chrysenes as non-steroidal glucocorticoid receptor modulators von Ardecky, Robert J., Hudson, Andrew R., Phillips, Dean P., Tyhonas, John S., Deckhut, Charlotte, Lau, Thomas L., Li, Yongkai, Martinborough, Esther A., Roach, Steven L., Higuchi, Robert I., Lopez, Francisco J., Marschke, Keith B., Miner, Jeffrey N., Karanewsky, Donald S., Negro-Vilar, Andrés, Zhi, Lin

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Ferric chloride, an efficient promoter of cationic polyene cyclizations von Sen, Stephanie E., Roach, Steven L., Smith, Sarah M., Zhang, Yan zhi

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Methods and compositions associated with the granulocyte colony-stimulating factor receptor von Pedram, Bijan, Marschke, Keith, Pickens, Jason C, Valdez, Lino J, Shen, Yixing, Hudson, Andrew R, Grant, Virginia H, Roach, Steven L, van Oeveren, Cornelis Arjan, Zhi, Lin

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