Discovery of 3-Aryl-4-isoxazolecarboxamides as TGR5 Receptor Agonists von Evans, Karen A, Budzik, Brian W, Ross, Sean A, Wisnoski, David D, Jin, Jian, Rivero, Ralph A, Vimal, Mythily, Szewczyk, George R, Jayawickreme, Channa, Moncol, David L, Rimele, Thomas J, Armour, Susan L, Weaver, Susan P, Griffin, Robert J, Tadepalli, Sarva M, Jeune, Michael R, Shearer, Todd W, Chen, Zibin B, Chen, Lihong, Anderson, Donald L, Becherer, J. David, De Los Frailes, Maite, Colilla, Francisco Javier

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Identification of potent, nonabsorbable agonists of the calcium-sensing receptor for GI-specific administration von Sparks, Steven M., Spearing, Paul K., Diaz, Caroline J., Cowan, David J., Jayawickreme, Channa, Chen, Grace, Rimele, Thomas J., Generaux, Claudia, Harston, Lindsey T., Roller, Shane G.

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BMY 7378 is a selective antagonist of the D subtype of α1-adrenoceptors von Goetz, Aaron S., King, Holly K., Ward, Stuart D.C., True, Timothy A., Rimele, Thomas J., Saussy, David L.

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Discovery of 1,5-Benzodiazepines with Peripheral Cholecystokinin (CCK-A) Receptor Agonist Activity. 1. Optimization of the Agonist “Trigger” von Aquino, Christopher J, Armour, Duncan R, Berman, Judd M, Birkemo, Larry S, Carr, Robin A. E, Croom, Dallas K, Dezube, Milana, Dougherty, Robert W, Ervin, Gregory N, Grizzle, Mary K, Head, Julie E, Hirst, Gavin C, James, Michael K, Johnson, Michael F, Miller, Laurence J, Queen, Kennedy L, Rimele, Thomas J, Smith, David N, Sugg, Elizabeth E

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1,4-Benzodiazepine Peripheral Cholecystokinin (CCK-A) Receptor Agonists von Sherrill, Ronald G, Berman, Judd M, Birkemo, Lawrence, Croom, Dallas K, Dezube, Milana, Ervin, Gregory N, Grizzle, Mary K, James, Michael K, Johnson, Michael F, Queen, Kennedy L, Rimele, Thomas J, Vanmiddlesworth, Frank, Sugg, Elizabeth E

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3-[2-(N-Phenylacetamide)]-1,5-benzodiazepines:  Orally Active, Binding Selective CCK-A Agonists von Willson, Timothy M, Henke, Brad R, Momtahen, Tanya M, Myers, Peter L, Sugg, Elizabeth E, Unwalla, Rayomand J, Croom, Dallas K, Dougherty, Robert W, Grizzle, Mary K, Johnson, Michael F, Queen, Kennedy L, Rimele, Thomas J, Yingling, Jeffrey D, James, Michael K

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CCK-A Receptor Selective Antagonists Derived from the CCK-A Receptor Selective Tetrapeptide Agonist Boc-Trp-Lys(Tac)-Asp-MePhe-NH2 (A-71623) von Sugg, Elizabeth E, Kimery, Millard J, Ding, Jian Mei, Kenakin, Deborah C, Miller, Laurence J, Queen, Kennedy L, Rimele, Thomas J

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Foreword von Rimele, Thomas J

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Comparison of the β-Adrenoceptor Affinity and Selectivity of Cetamolol, Atenolol, Betaxolol, and ICI-118,551 von Rimele, Thomas J, Henry, Diane E, Giesa, Frank R, Buckley, Susan K, Geiger, Gabriella, Heaslip, Richard J, Lee, David K. H, Grimes, David

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The synthesis and pharmacological evaluation of indole congeners of the calcium entry blocker verapamil von Soll, Richard M, Parks, James A, Rimele, Thomas J, Heaslip, Richard J, Wojdan, Alexandra, Oshiro, George, Grimes, David, Asselin, André

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Indole-phenol-bioisosterism. Synthesis and antihypertensive activity of a pyrrolo analog of labetalol von Asselin, Andre A, Humber, Leslie G, Crosilla, Danilo, Oshiro, George, Wojdan, Alexandra, Grimes, David, Heaslip, Richard J, Rimele, Thomas J, Shaw, Chia Cheng

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Modification of Receptor Selectivity and Functional Activity in Cholecystokinin Peptoid Ligands von Dezube, Milana, Sugg, Elizabeth E, Birkemo, Larry S, Croom, Dallas K, Dougherty, Robert W, Ervin, Gregory N, Grizzle, Mary K, James, Michael K, Johnson, Michael F

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Binding of [3H]quinuclidinyl benzilate to intestinal mucus von Rimele, Thomas J., Gaginella, Timothy S.

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Sensitivity of the PGF2α-versus carbachol-contracted trachea to relaxation by salbutamol, forskolin and prenalterol von HEASLIP, R. J, GIESA, F. R, RIMELE, T. J, GRIMES, D

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Demonstration of the β2-adrenoceptor intrinsic efficacy of AY-28,925 using the PGF 2α-contracted guinea-pig trachea von Heaslip, Richard J., Giesa, Frank R., Rimele, Thomas J., Grimes, David

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Demonstration of the β2-adrenoceptor intrinsic efficacy of AY-28,925 using the PGF2α-contracted guinea-pig trachea von HEASLIP, R. J, GIESA, F. R, RIMELE, T. J, GRIMES, D

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Sensitivity of the PGF 2α- versus carbachol-contracted trachea to relaxation by salbutamol, forskolin and prenalterol von Heaslip, Richard J., Giesa, Frank R., Rimele, Thomas J., Grimes, David

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Binding of [ 3H]quinuclidinyl benzilate to intestinal mucus : An artifact in identification of epithelial cell muscarinic receptors von Rimele, Thomas J., Gaginella, Timothy S.

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In vivo identification of muscarinic receptors on rat colonic epithelial cells. Binding of [3H]-quinuclidinyl benzilate von Rimele, T J, Gaginella, T S

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Effect of thymoxamine on the human pupil von Lee, David A., Rimele, Thomas J., Brubaker, Richard F., Nagataki, Shigetoshi, Vanhoutte, Paul M.

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